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maximum 50k data
Found 86 Enz. Inhib. hit(s) with all data for entry = 50048909
TargetType-1 angiotensin II receptor A/B(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230906(CHEMBL308261)
Affinity DataIC50:  0.410nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230919(CHEMBL307844 | CI-996)
Affinity DataIC50:  0.580nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230891(CHEMBL76166)
Affinity DataIC50:  0.800nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230883(CHEMBL309089)
Affinity DataIC50:  0.820nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230915(CHEMBL76169)
Affinity DataIC50:  0.900nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230887(CHEMBL306259)
Affinity DataIC50:  1nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230912(CHEMBL72922)
Affinity DataIC50:  1.20nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230886(CHEMBL307455)
Affinity DataIC50:  1.40nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230882(CARBOXYLIC ACID METABOLITE | CHEBI:74125 | E-3174)
Affinity DataIC50:  1.60nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230882(CARBOXYLIC ACID METABOLITE | CHEBI:74125 | E-3174)
Affinity DataIC50:  1.60nMAssay Description:Tested for inhibitory concentration against AT1 receptor binding affinity in rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230910(CHEMBL306066)
Affinity DataIC50:  1.60nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1/Type-2 angiotensin II receptor(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230882(CARBOXYLIC ACID METABOLITE | CHEBI:74125 | E-3174)
Affinity DataIC50:  1.80nMAssay Description:Inhibitory concentration against [125I]angiotensin II(AII) induced contraction in rabbit aorta by 50%More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230877(CHEMBL70371)
Affinity DataIC50:  2.40nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1/Type-2 angiotensin II receptor(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230883(CHEMBL309089)
Affinity DataIC50:  2.40nMAssay Description:Inhibitory concentration against [125I]angiotensin II(AII) induced contraction in rabbit aorta by 50%More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230900(CHEMBL73433)
Affinity DataIC50:  2.5nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1/Type-2 angiotensin II receptor(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230891(CHEMBL76166)
Affinity DataIC50:  2.60nMAssay Description:Inhibitory concentration against [125I]angiotensin II(AII) induced contraction in rabbit aorta by 50%More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230902(CHEMBL75518)
Affinity DataIC50:  2.80nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230893(CHEMBL308031)
Affinity DataIC50:  2.80nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1/Type-2 angiotensin II receptor(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230887(CHEMBL306259)
Affinity DataIC50:  2.90nMAssay Description:Inhibitory concentration against [125I]angiotensin II(AII) induced contraction in rabbit aorta by 50%More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1/Type-2 angiotensin II receptor(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230906(CHEMBL308261)
Affinity DataIC50:  3.30nMAssay Description:Inhibitory concentration against [125I]angiotensin II(AII) induced contraction in rabbit aorta by 50%More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230881(CHEMBL308779)
Affinity DataIC50:  3.30nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230908(CHEMBL443269 | DuP-532)
Affinity DataIC50:  3.40nMAssay Description:Tested for inhibitory concentration against AT1 receptor binding affinity in rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230897(CHEMBL275652)
Affinity DataIC50:  3.60nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230909(CHEMBL306852)
Affinity DataIC50:  3.60nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1/Type-2 angiotensin II receptor(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230919(CHEMBL307844 | CI-996)
Affinity DataIC50:  3.80nMAssay Description:Inhibitory concentration against [125I]angiotensin II(AII) induced contraction in rabbit aorta by 50%More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230914(CHEMBL431390)
Affinity DataIC50:  3.90nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230888(CHEMBL306612)
Affinity DataIC50:  4nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1/Type-2 angiotensin II receptor(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230877(CHEMBL70371)
Affinity DataIC50:  4nMAssay Description:Inhibitory concentration against [125I]angiotensin II(AII) induced contraction in rabbit aorta by 50%More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1/Type-2 angiotensin II receptor(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230915(CHEMBL76169)
Affinity DataIC50:  4.5nMAssay Description:Inhibitory concentration against [125I]angiotensin II(AII) induced contraction in rabbit aorta by 50%More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1/Type-2 angiotensin II receptor(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230893(CHEMBL308031)
Affinity DataIC50:  4.80nMAssay Description:Inhibitory concentration against [125I]angiotensin II(AII) induced contraction in rabbit aorta by 50%More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM82258(CAS_114798-26-4 | Losartan | NSC_3961)
Affinity DataIC50:  5nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM82258(CAS_114798-26-4 | Losartan | NSC_3961)
Affinity DataIC50:  5nMAssay Description:Tested for inhibitory concentration against AT1 receptor binding affinity in rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1/Type-2 angiotensin II receptor(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230912(CHEMBL72922)
Affinity DataIC50:  5.40nMAssay Description:Inhibitory concentration against [125I]angiotensin II(AII) induced contraction in rabbit aorta by 50%More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230899(CHEMBL75935)
Affinity DataIC50:  5.60nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1/Type-2 angiotensin II receptor(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230910(CHEMBL306066)
Affinity DataIC50:  7nMAssay Description:Inhibitory concentration against [125I]angiotensin II(AII) induced contraction in rabbit aorta by 50%More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230885(CHEMBL72453)
Affinity DataIC50:  8.80nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1/Type-2 angiotensin II receptor(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230918(CHEMBL73084)
Affinity DataIC50:  9nMAssay Description:Inhibitory concentration against [125I]angiotensin II(AII) induced contraction in rabbit aorta by 50%More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230911(CHEMBL306949)
Affinity DataIC50:  11nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230918(CHEMBL73084)
Affinity DataIC50:  11nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230890(CHEMBL73646)
Affinity DataIC50:  12nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230907(CHEMBL76393)
Affinity DataIC50:  14nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230879(CHEMBL309094)
Affinity DataIC50:  15nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1/Type-2 angiotensin II receptor(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230900(CHEMBL73433)
Affinity DataIC50:  18nMAssay Description:Inhibitory concentration against [125I]angiotensin II(AII) induced contraction in rabbit aorta by 50%More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1/Type-2 angiotensin II receptor(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230911(CHEMBL306949)
Affinity DataIC50:  19nMAssay Description:Inhibitory concentration against [125I]angiotensin II(AII) induced contraction in rabbit aorta by 50%More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230916(CHEMBL76330)
Affinity DataIC50:  19nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230896(CHEMBL308961)
Affinity DataIC50:  21nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1/Type-2 angiotensin II receptor(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230881(CHEMBL308779)
Affinity DataIC50:  21nMAssay Description:Inhibitory concentration against [125I]angiotensin II(AII) induced contraction in rabbit aorta by 50%More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230892(CHEMBL73725)
Affinity DataIC50:  22nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230913(CHEMBL75092)
Affinity DataIC50:  22nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230920(CHEMBL307284)
Affinity DataIC50:  23nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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