Compile Data Set for Download or QSAR
maximum 50k data
Found 17 Enz. Inhib. hit(s) with all data for entry = 50036818
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50089269(CHEMBL276192 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2...)
Affinity DataKi:  0.0200nMAssay Description:Inhibition of [125I]BH-CCK-8 binding to Cholecystokinin type A receptor of rat pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50061828(CHEMBL76248 | CID44356929 | N-(1-Carbamoyl-2-pheny...)
Affinity DataKi:  0.0300nMAssay Description:Inhibition of [125I]BH-CCK-8 binding to Cholecystokinin type A receptor of rat pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50089268(CHEMBL267861 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2...)
Affinity DataKi:  0.0500nMAssay Description:Inhibition of [125I]BH-CCK-8 binding to Cholecystokinin type A receptor of rat pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataKi:  0.0900nMAssay Description:Inhibition of [125I]BH-CCK-8 binding to Cholecystokinin type A receptor of rat pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataKi:  0.410nMAssay Description:Binding affinity towards Cholecystokinin type B receptor in rat cortex synaptosomes using [125I]BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50089276(CHEMBL430608 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2...)
Affinity DataKi:  0.980nMAssay Description:Inhibition of [125I]BH-CCK-8 binding to Cholecystokinin type A receptor of rat pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50089275(CHEMBL384303 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2...)
Affinity DataKi:  3.40nMAssay Description:Inhibition of [125I]BH-CCK-8 binding to Cholecystokinin type A receptor of rat pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50089277(CHEMBL311187 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-({...)
Affinity DataKi:  4.20nMAssay Description:Inhibition of [125I]BH-CCK-8 binding to Cholecystokinin type A receptor of rat pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50089272(CHEMBL312359 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2...)
Affinity DataKi:  19nMAssay Description:Inhibition of [125I]BH-CCK-8 binding to Cholecystokinin type A receptor of rat pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50089275(CHEMBL384303 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2...)
Affinity DataKi:  36nMAssay Description:Binding affinity towards Cholecystokinin type B receptor in rat cortex synaptosomes using [125I]BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50089270(CHEMBL308622 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2...)
Affinity DataKi:  51nMAssay Description:Inhibition of [125I]BH-CCK-8 binding to Cholecystokinin type A receptor of rat pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50089276(CHEMBL430608 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2...)
Affinity DataKi:  84nMAssay Description:Binding affinity towards Cholecystokinin type B receptor in rat cortex synaptosomes using [125I]BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50089269(CHEMBL276192 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2...)
Affinity DataKi:  123nMAssay Description:Binding affinity towards Cholecystokinin type B receptor in rat cortex synaptosomes using [125I]BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50089272(CHEMBL312359 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2...)
Affinity DataKi:  150nMAssay Description:Binding affinity towards Cholecystokinin type B receptor in rat cortex synaptosomes using [125I]BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50089268(CHEMBL267861 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2...)
Affinity DataKi:  200nMAssay Description:Binding affinity towards Cholecystokinin type B receptor in rat cortex synaptosomes using [125I]BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50061828(CHEMBL76248 | CID44356929 | N-(1-Carbamoyl-2-pheny...)
Affinity DataKi:  224nMAssay Description:Binding affinity towards Cholecystokinin type B receptor in rat cortex synaptosomes using [125I]BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50089277(CHEMBL311187 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-({...)
Affinity DataKi:  960nMAssay Description:Binding affinity towards Cholecystokinin type B receptor in rat cortex synaptosomes using [125I]BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed