Compile Data Set for Download or QSAR
maximum 50k data
Found 53 Enz. Inhib. hit(s) with all data for entry = 50037015
TargetDelta-type opioid receptor(MOUSE)
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50370067(CHEMBL1237164)
Affinity DataKi:  0.0300nMAssay Description:Antagonist activity of compound on agonist stimulated [35S]GTP-gamma-S binding on delta-opioid receptorMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(MOUSE)
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50370067(CHEMBL1237164)
Affinity DataKi:  0.220nMAssay Description:Displacement of [3H]DADLE at delta-opioid receptorMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(MOUSE)
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50098674((E)-17-(2-butenyl)-6,7-dehydro-4,5alpha-epoxy-3,14...)
Affinity DataKi:  0.680nMAssay Description:Antagonist activity of compound on agonist stimulated [35S]GTP-gamma-S binding on delta-opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50221416(22-methyl-(2S,13R)-14-oxa-11,22-diazaheptacyclo[13...)
Affinity DataKi:  0.800nMAssay Description:Displacement of [3H]DADLE at delta-opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50098673(17-(2-methyl-2-propenyl)-6,7-dehydro-4,5alpha-epox...)
Affinity DataKi:  1.20nMAssay Description:Antagonist activity of compound on agonist stimulated [35S]GTP-gamma-S binding on delta-opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50098677(17-propyl-6,7-dehydro-4,5alpha-epoxy-3,14-dihydrox...)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]DADLE at delta-opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50098680(17-ethyl-6,7-dehydro-4,5alpha-epoxy-3,14-dihydroxy...)
Affinity DataKi:  3.20nMAssay Description:Antagonist activity of compound on SNC 80 stimulated [35S]GTP-gamma-S binding to delta-opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50098683(17-(2-methylpropyl)-6,7-dehydro-4,5alpha-epoxy-3,1...)
Affinity DataKi:  3.80nMAssay Description:Displacement of [3H]DADLE at delta-opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50370067(CHEMBL1237164)
Affinity DataKi:  4.30nMAssay Description:Antagonist activity of compound on agonist stimulated [35S]GTP-gamma-S binding on mu-opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50370067(CHEMBL1237164)
Affinity DataKi:  4.70nMAssay Description:Antagonist activity of compound on U50,488H stimulated [35S]GTP-gamma-S binding to opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50098673(17-(2-methyl-2-propenyl)-6,7-dehydro-4,5alpha-epox...)
Affinity DataKi:  4.70nMAssay Description:Displacement of [3H]DADLE at delta-opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50098676(17-(3-methylbutyl)-6,7-dehydro-4,5alpha-epoxy-3,14...)
Affinity DataKi:  4.80nMAssay Description:Displacement of [3H]DADLE at delta-opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50098680(17-ethyl-6,7-dehydro-4,5alpha-epoxy-3,14-dihydroxy...)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]DADLE at delta-opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50098674((E)-17-(2-butenyl)-6,7-dehydro-4,5alpha-epoxy-3,14...)
Affinity DataKi:  7.40nMAssay Description:Displacement of [3H]DADLE at delta-opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50098681(17-butyl-6,7-dehydro-4,5alpha-epoxy-3,14-dihydroxy...)
Affinity DataKi:  8.40nMAssay Description:Displacement of [3H]DADLE at delta-opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50098675(17-pentyl-6,7-dehydro-4,5alpha-epoxy-3,14-dihydrox...)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]DADLE at delta-opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50098679(17-(3-methyl-2-butenyl)-6,7-dehydro-4,5alpha-epoxy...)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]DADLE at delta-opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50098672(17-hexyl-6,7-dehydro-4,5alpha-epoxy-3,14-dihydroxy...)
Affinity DataKi:  26nMAssay Description:Displacement of [3H]DADLE at delta-opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50370067(CHEMBL1237164)
Affinity DataKi:  27nMAssay Description:Displacement of [3H]DAMGO at mu-opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50098674((E)-17-(2-butenyl)-6,7-dehydro-4,5alpha-epoxy-3,14...)
Affinity DataKi:  30nMAssay Description:Antagonist activity of compound on agonist stimulated [35S]GTP-gamma-S binding on mu-opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50370067(CHEMBL1237164)
Affinity DataKi:  30nMAssay Description:Displacement of [3H]U-69593 at opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50098678(17-(1-methylethyl)-6,7-dehydro-4,5alpha-epoxy-3,14...)
Affinity DataKi:  33nMAssay Description:Displacement of [3H]DADLE at delta-opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50221416(22-methyl-(2S,13R)-14-oxa-11,22-diazaheptacyclo[13...)
Affinity DataKi:  66nMAssay Description:Displacement of [3H]DAMGO at mu-opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50098682(17-heptyl-6,7-dehydro-4,5alpha-epoxy-3,14-dihydrox...)
Affinity DataKi:  79nMAssay Description:Displacement of [3H]DADLE at delta-opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50098674((E)-17-(2-butenyl)-6,7-dehydro-4,5alpha-epoxy-3,14...)
Affinity DataKi:  118nMAssay Description:Antagonist activity of compound on U50,488H stimulated [35S]GTP-gamma-S binding to opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50098673(17-(2-methyl-2-propenyl)-6,7-dehydro-4,5alpha-epox...)
Affinity DataKi:  200nMAssay Description:Antagonist activity of compound on agonist stimulated [35S]GTP-gamma-S binding on mu-opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50098680(17-ethyl-6,7-dehydro-4,5alpha-epoxy-3,14-dihydroxy...)
Affinity DataKi:  290nMAssay Description:Antagonist activity of compound on DAMGO stimulated [35S]GTP-gamma-S binding to mu-opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50098677(17-propyl-6,7-dehydro-4,5alpha-epoxy-3,14-dihydrox...)
Affinity DataKi:  380nMAssay Description:Displacement of [3H]U-69593 at opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50098683(17-(2-methylpropyl)-6,7-dehydro-4,5alpha-epoxy-3,1...)
Affinity DataKi:  650nMAssay Description:Displacement of [3H]U-69593 at opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50098676(17-(3-methylbutyl)-6,7-dehydro-4,5alpha-epoxy-3,14...)
Affinity DataKi:  670nMAssay Description:Displacement of [3H]U-69593 at opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50098677(17-propyl-6,7-dehydro-4,5alpha-epoxy-3,14-dihydrox...)
Affinity DataKi:  710nMAssay Description:Displacement of [3H]DAMGO at mu-opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50098673(17-(2-methyl-2-propenyl)-6,7-dehydro-4,5alpha-epox...)
Affinity DataKi:  740nMAssay Description:Antagonist activity of compound on U50,488H stimulated [35S]GTP-gamma-S binding to opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50098681(17-butyl-6,7-dehydro-4,5alpha-epoxy-3,14-dihydroxy...)
Affinity DataKi:  900nMAssay Description:Displacement of [3H]U-69593 at opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50098674((E)-17-(2-butenyl)-6,7-dehydro-4,5alpha-epoxy-3,14...)
Affinity DataKi:  960nMAssay Description:Displacement of [3H]U-69593 at opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50098680(17-ethyl-6,7-dehydro-4,5alpha-epoxy-3,14-dihydroxy...)
Affinity DataKi: >1.00E+3nMAssay Description:Antagonist activity of compound on U50,488H stimulated [35S]GTP-gamma-S binding to opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50098674((E)-17-(2-butenyl)-6,7-dehydro-4,5alpha-epoxy-3,14...)
Affinity DataKi:  1.20E+3nMAssay Description:Displacement of [3H]DAMGO at mu-opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50098681(17-butyl-6,7-dehydro-4,5alpha-epoxy-3,14-dihydroxy...)
Affinity DataKi:  1.30E+3nMAssay Description:Displacement of [3H]DAMGO at mu-opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50098676(17-(3-methylbutyl)-6,7-dehydro-4,5alpha-epoxy-3,14...)
Affinity DataKi:  1.30E+3nMAssay Description:Displacement of [3H]DAMGO at mu-opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50098675(17-pentyl-6,7-dehydro-4,5alpha-epoxy-3,14-dihydrox...)
Affinity DataKi:  2.00E+3nMAssay Description:Displacement of [3H]U-69593 at opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50098680(17-ethyl-6,7-dehydro-4,5alpha-epoxy-3,14-dihydroxy...)
Affinity DataKi:  2.50E+3nMAssay Description:Displacement of [3H]DAMGO at mu-opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50098683(17-(2-methylpropyl)-6,7-dehydro-4,5alpha-epoxy-3,1...)
Affinity DataKi:  2.60E+3nMAssay Description:Displacement of [3H]DAMGO at mu-opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50098679(17-(3-methyl-2-butenyl)-6,7-dehydro-4,5alpha-epoxy...)
Affinity DataKi:  2.80E+3nMAssay Description:Displacement of [3H]DAMGO at mu-opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50098675(17-pentyl-6,7-dehydro-4,5alpha-epoxy-3,14-dihydrox...)
Affinity DataKi:  2.80E+3nMAssay Description:Displacement of [3H]DAMGO at mu-opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50098680(17-ethyl-6,7-dehydro-4,5alpha-epoxy-3,14-dihydroxy...)
Affinity DataKi:  3.00E+3nMAssay Description:Displacement of [3H]U-69593 at opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50098672(17-hexyl-6,7-dehydro-4,5alpha-epoxy-3,14-dihydroxy...)
Affinity DataKi:  3.10E+3nMAssay Description:Displacement of [3H]U-69593 at opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50098679(17-(3-methyl-2-butenyl)-6,7-dehydro-4,5alpha-epoxy...)
Affinity DataKi:  3.20E+3nMAssay Description:Displacement of [3H]U-69593 at opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50098673(17-(2-methyl-2-propenyl)-6,7-dehydro-4,5alpha-epox...)
Affinity DataKi:  3.80E+3nMAssay Description:Displacement of [3H]U-69593 at opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50098682(17-heptyl-6,7-dehydro-4,5alpha-epoxy-3,14-dihydrox...)
Affinity DataKi:  4.60E+3nMAssay Description:Displacement of [3H]DAMGO at mu-opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50098672(17-hexyl-6,7-dehydro-4,5alpha-epoxy-3,14-dihydroxy...)
Affinity DataKi:  4.60E+3nMAssay Description:Displacement of [3H]DAMGO at mu-opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50098678(17-(1-methylethyl)-6,7-dehydro-4,5alpha-epoxy-3,14...)
Affinity DataKi:  6.20E+3nMAssay Description:Displacement of [3H]U-69593 at opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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