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Found 10 Enz. Inhib. hit(s) with all data for entry = 50038383
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Stanford University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50375695(CHEMBL270984)
Affinity DataKi:  0.0190nMAssay Description:Displacement of [3H]deltorphin2 from delta opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Stanford University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50375694(CHEMBL244265)
Affinity DataKi:  0.172nMAssay Description:Displacement of [3H]deltorphin2 from delta opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Stanford University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50375696(CHEMBL269842)
Affinity DataKi:  0.248nMAssay Description:Displacement of [3H]deltorphin2 from delta opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Stanford University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50375695(CHEMBL270984)
Affinity DataKi:  2.75nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Stanford University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50375696(CHEMBL269842)
Affinity DataKi:  13.2nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Stanford University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50375694(CHEMBL244265)
Affinity DataKi:  41.2nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Stanford University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50375696(CHEMBL269842)
Affinity DataIC50:  50.6nMAssay Description:Agonist activity at mu opioid receptor in Hartley guinea pig assessed as inhibition of electrically evoked-contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Stanford University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50375694(CHEMBL244265)
Affinity DataIC50:  1.92E+3nMAssay Description:Agonist activity at mu opioid receptor in Hartley guinea pig assessed as inhibition of electrically evoked-contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Stanford University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50375696(CHEMBL269842)
Affinity DataIC50:  5.18E+3nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically evoked-contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Stanford University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50375695(CHEMBL270984)
Affinity DataIC50: >1.00E+4nMAssay Description:Agonist activity at mu opioid receptor in Hartley guinea pig assessed as inhibition of electrically evoked-contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed