Compile Data Set for Download or QSAR
maximum 50k data
Found 14 Enz. Inhib. hit(s) with all data for entry = 50010761
TargetThrombospondin-1(Homo sapiens)
Southern Research Institute

Curated by ChEMBL
LigandPNGBDBM50541838(CHEMBL4649483)
Affinity DataIC50:  0.380nMAssay Description:Inhibition of TSP1 in human myeloma cells assessed reduction in TGFbeta activity incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetThrombospondin-1(Homo sapiens)
Southern Research Institute

Curated by ChEMBL
LigandPNGBDBM50541831(CHEMBL4644535)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of TSP1 in human myeloma cells assessed reduction in TGFbeta activity incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetThrombospondin-1(Homo sapiens)
Southern Research Institute

Curated by ChEMBL
LigandPNGBDBM50541837(CHEMBL4642848)
Affinity DataIC50:  1.70nMAssay Description:Inhibition of TSP1 in human myeloma cells assessed reduction in TGFbeta activity incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThrombospondin-1(Homo sapiens)
Southern Research Institute

Curated by ChEMBL
LigandPNGBDBM50541836(CHEMBL4642780)
Affinity DataIC50:  2nMAssay Description:Inhibition of TSP1 in human myeloma cells assessed reduction in TGFbeta activity incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThrombospondin-1(Homo sapiens)
Southern Research Institute

Curated by ChEMBL
LigandPNGBDBM50541828(CHEMBL4633877)
Affinity DataIC50:  2.20nMAssay Description:Inhibition of TSP1 in human myeloma cells assessed reduction in TGFbeta activity incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThrombospondin-1(Homo sapiens)
Southern Research Institute

Curated by ChEMBL
LigandPNGBDBM50541833(CHEMBL4636492)
Affinity DataIC50:  2.90nMAssay Description:Inhibition of TSP1 in human myeloma cells assessed reduction in TGFbeta activity incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThrombospondin-1(Homo sapiens)
Southern Research Institute

Curated by ChEMBL
LigandPNGBDBM50541832(CHEMBL4648099)
Affinity DataIC50:  3.30nMAssay Description:Inhibition of TSP1 in human myeloma cells assessed reduction in TGFbeta activity incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThrombospondin-1(Homo sapiens)
Southern Research Institute

Curated by ChEMBL
LigandPNGBDBM50541830(CHEMBL4647669)
Affinity DataIC50:  4.40nMAssay Description:Inhibition of TSP1 in human myeloma cells assessed reduction in TGFbeta activity incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetThrombospondin-1(Homo sapiens)
Southern Research Institute

Curated by ChEMBL
LigandPNGBDBM50541826(CHEMBL4644244)
Affinity DataIC50:  5.20nMAssay Description:Inhibition of TSP1 in human myeloma cells assessed reduction in TGFbeta activity incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThrombospondin-1(Homo sapiens)
Southern Research Institute

Curated by ChEMBL
LigandPNGBDBM50541839(CHEMBL4649293)
Affinity DataIC50:  7.60nMAssay Description:Inhibition of TSP1 in human myeloma cells assessed reduction in TGFbeta activity incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThrombospondin-1(Homo sapiens)
Southern Research Institute

Curated by ChEMBL
LigandPNGBDBM50541827(CHEMBL4644046)
Affinity DataIC50:  9.5nMAssay Description:Inhibition of TSP1 in human myeloma cells assessed reduction in TGFbeta activity incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThrombospondin-1(Homo sapiens)
Southern Research Institute

Curated by ChEMBL
LigandPNGBDBM50541834(CHEMBL4644197)
Affinity DataIC50:  13nMAssay Description:Inhibition of TSP1 in human myeloma cells assessed reduction in TGFbeta activity incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThrombospondin-1(Homo sapiens)
Southern Research Institute

Curated by ChEMBL
LigandPNGBDBM50541835(CHEMBL4645518)
Affinity DataIC50:  14nMAssay Description:Inhibition of TSP1 in human myeloma cells assessed reduction in TGFbeta activity incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThrombospondin-1(Homo sapiens)
Southern Research Institute

Curated by ChEMBL
LigandPNGBDBM50541829(CHEMBL4638959)
Affinity DataIC50:  15nMAssay Description:Inhibition of TSP1 in human myeloma cells assessed reduction in TGFbeta activity incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed