Compile Data Set for Download or QSAR
maximum 50k data
Found 9 Enz. Inhib. hit(s) with all data for entry = 50004201
TargetReverse transcriptase(Human immunodeficiency virus 1)
Afmb-Cnrs-Esil

Curated by ChEMBL
LigandPNGBDBM50479983(Adefovir Diphosphate)
Affinity DataIC50:  8.30E+3nMAssay Description:Inhibition of HIV1 wild type reverse transcriptase p66/p51 expressed in Escherichia coli using calf thymus DNA substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Afmb-Cnrs-Esil

Curated by ChEMBL
LigandPNGBDBM50479984(CHEMBL2448398)
Affinity DataIC50:  1.45E+4nMAssay Description:Inhibition of HIV1 wild type reverse transcriptase p66/p51 expressed in Escherichia coli using calf thymus DNA substrateMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Afmb-Cnrs-Esil

Curated by ChEMBL
LigandPNGBDBM50479985(CHEMBL2448397)
Affinity DataIC50:  1.70E+4nMAssay Description:Inhibition of HIV1 wild type reverse transcriptase p66/p51 expressed in Escherichia coli using calf thymus DNA substrateMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Afmb-Cnrs-Esil

Curated by ChEMBL
LigandPNGBDBM50478158(Tenofovir diphospahte | tenofovir diphosphate)
Affinity DataIC50:  2.20E+4nMAssay Description:Inhibition of HIV1 wild type reverse transcriptase p66/p51 expressed in Escherichia coli using calf thymus DNA substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Afmb-Cnrs-Esil

Curated by ChEMBL
LigandPNGBDBM50479985(CHEMBL2448397)
Affinity DataKd:  6.50E+3nMAssay Description:Binding affinity to HIV1 wild type reverse transcriptase p66/p51 expressed in Escherichia coli assessed as incorporation of drug to DNA by gel electr...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Afmb-Cnrs-Esil

Curated by ChEMBL
LigandPNGBDBM50478158(Tenofovir diphospahte | tenofovir diphosphate)
Affinity DataKd:  2.30E+4nMAssay Description:Binding affinity to HIV1 wild type reverse transcriptase p66/p51 expressed in Escherichia coli assessed as incorporation of drug to DNA by gel electr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Afmb-Cnrs-Esil

Curated by ChEMBL
LigandPNGBDBM50118233(2'-deoxyadenosine 5'-(tetrahydrogen triphosphate) ...)
Affinity DataKd:  7.50E+3nMAssay Description:Binding affinity to HIV1 wild type reverse transcriptase p66/p51 expressed in Escherichia coli assessed as incorporation of drug to DNA by gel electr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Afmb-Cnrs-Esil

Curated by ChEMBL
LigandPNGBDBM50479984(CHEMBL2448398)
Affinity DataKd:  3.30E+4nMAssay Description:Binding affinity to HIV1 wild type reverse transcriptase p66/p51 expressed in Escherichia coli assessed as incorporation of drug to DNA by gel electr...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Afmb-Cnrs-Esil

Curated by ChEMBL
LigandPNGBDBM50479983(Adefovir Diphosphate)
Affinity DataKd:  7.90E+3nMAssay Description:Binding affinity to HIV1 wild type reverse transcriptase p66/p51 expressed in Escherichia coli assessed as incorporation of drug to DNA by gel electr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed