Compile Data Set for Download or QSAR
Found 27 Enz. Inhib. hit(s) with all data for entry = 50012029
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Celltech R&D Inc.

Curated by ChEMBL
LigandPNGBDBM50102222(1-(2-Bromo-phenyl)-3-(7-cyano-3H-benzotriazol-4-yl...)
Affinity DataIC50:  10nMAssay Description:Displacement of [125I]-IL-8 from CHO cell membranes expressing human CX3C chemokine receptor 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Celltech R&D Inc.

Curated by ChEMBL
LigandPNGBDBM50113628(CHEMBL431511 | [5-(4-Fluoro-phenylcarbamoyl)-pyrid...)
Affinity DataIC50:  32nMAssay Description:Displacement of [125I]-IL-8 from CHO cell membranes expressing human CX3C chemokine receptor 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1/2(Homo sapiens (Human))
Celltech R&D Inc.

Curated by ChEMBL
LigandPNGBDBM50113628(CHEMBL431511 | [5-(4-Fluoro-phenylcarbamoyl)-pyrid...)
Affinity DataIC50:  42nMAssay Description:Inhibition against GRO-alpha driven human neutrophil chemotaxisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1/2(Homo sapiens (Human))
Celltech R&D Inc.

Curated by ChEMBL
LigandPNGBDBM50219799(CHEMBL36535)
Affinity DataIC50:  43nMAssay Description:Inhibition against GRO-alpha driven human neutrophil chemotaxisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1/2(Homo sapiens (Human))
Celltech R&D Inc.

Curated by ChEMBL
LigandPNGBDBM50219797(CHEMBL36934)
Affinity DataIC50:  46nMAssay Description:Inhibition against GRO-alpha driven human neutrophil chemotaxisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1/2(Homo sapiens (Human))
Celltech R&D Inc.

Curated by ChEMBL
LigandPNGBDBM50219796(CHEMBL39464)
Affinity DataIC50:  50nMAssay Description:Inhibition against GRO-alpha driven human neutrophil chemotaxisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1/2(Homo sapiens (Human))
Celltech R&D Inc.

Curated by ChEMBL
LigandPNGBDBM50219800(CHEMBL432475)
Affinity DataIC50:  83nMAssay Description:Inhibition against GRO-alpha driven human neutrophil chemotaxisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1/2(Homo sapiens (Human))
Celltech R&D Inc.

Curated by ChEMBL
LigandPNGBDBM50219806(CHEMBL291140)
Affinity DataIC50:  94nMAssay Description:Inhibition against GRO-alpha driven human neutrophil chemotaxisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1/2(Homo sapiens (Human))
Celltech R&D Inc.

Curated by ChEMBL
LigandPNGBDBM50219809(CHEMBL36643)
Affinity DataIC50:  110nMAssay Description:Inhibition against GRO-alpha driven human neutrophil chemotaxisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Celltech R&D Inc.

Curated by ChEMBL
LigandPNGBDBM50102225(CHEMBL39740 | N'-(3-[2,2']Bithiophenyl-5-yl-6,7-di...)
Affinity DataIC50:  110nMAssay Description:Displacement of [125I]-IL-8 from CHO cell membranes expressing human CX3C chemokine receptor 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1/2(Homo sapiens (Human))
Celltech R&D Inc.

Curated by ChEMBL
LigandPNGBDBM50219811(CHEMBL39710)
Affinity DataIC50:  160nMAssay Description:Inhibition against GRO-alpha driven human neutrophil chemotaxisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1/2(Homo sapiens (Human))
Celltech R&D Inc.

Curated by ChEMBL
LigandPNGBDBM50219812(CHEMBL36842)
Affinity DataIC50:  200nMAssay Description:Inhibition against GRO-alpha driven human neutrophil chemotaxisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1/2(Homo sapiens (Human))
Celltech R&D Inc.

Curated by ChEMBL
LigandPNGBDBM50219808(CHEMBL288527)
Affinity DataIC50:  220nMAssay Description:Inhibition against GRO-alpha driven human neutrophil chemotaxisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1/2(Homo sapiens (Human))
Celltech R&D Inc.

Curated by ChEMBL
LigandPNGBDBM50219794(CHEMBL289656)
Affinity DataIC50:  220nMAssay Description:Inhibition against GRO-alpha driven human neutrophil chemotaxisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1/2(Homo sapiens (Human))
Celltech R&D Inc.

Curated by ChEMBL
LigandPNGBDBM50219810(CHEMBL288876)
Affinity DataIC50:  360nMAssay Description:Inhibition against GRO-alpha driven human neutrophil chemotaxisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1/2(Homo sapiens (Human))
Celltech R&D Inc.

Curated by ChEMBL
LigandPNGBDBM50219795(CHEMBL40080)
Affinity DataIC50:  410nMAssay Description:Inhibition against GRO-alpha driven human neutrophil chemotaxisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1/2(Homo sapiens (Human))
Celltech R&D Inc.

Curated by ChEMBL
LigandPNGBDBM50219789(CHEMBL40955)
Affinity DataIC50:  680nMAssay Description:Inhibition against GRO-alpha driven human neutrophil chemotaxisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1/2(Homo sapiens (Human))
Celltech R&D Inc.

Curated by ChEMBL
LigandPNGBDBM50219793(CHEMBL289789)
Affinity DataIC50:  760nMAssay Description:Inhibition against GRO-alpha driven human neutrophil chemotaxisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1/2(Homo sapiens (Human))
Celltech R&D Inc.

Curated by ChEMBL
LigandPNGBDBM50219790(CHEMBL39937)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition against GRO-alpha driven human neutrophil chemotaxisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Celltech R&D Inc.

Curated by ChEMBL
LigandPNGBDBM50113636(CHEMBL39835 | [5-(4-Fluoro-phenylcarbamoyl)-pyridi...)
Affinity DataIC50:  1.20E+3nMAssay Description:Displacement of [125I]-IL-8 from CHO cell membranes expressing human CX3C chemokine receptor 2 (CXCR2 filter mat binding assay)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1/2(Homo sapiens (Human))
Celltech R&D Inc.

Curated by ChEMBL
LigandPNGBDBM50219801(CHEMBL40558)
Affinity DataIC50:  2.70E+3nMAssay Description:Inhibition against GRO-alpha driven human neutrophil chemotaxisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1/2(Homo sapiens (Human))
Celltech R&D Inc.

Curated by ChEMBL
LigandPNGBDBM50219798(CHEMBL39988)
Affinity DataIC50:  5.10E+3nMAssay Description:Inhibition against GRO-alpha driven human neutrophil chemotaxisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1/2(Homo sapiens (Human))
Celltech R&D Inc.

Curated by ChEMBL
LigandPNGBDBM50219792(CHEMBL40114)
Affinity DataIC50:  1.25E+4nMAssay Description:Inhibition against GRO-alpha driven human neutrophil chemotaxisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1/2(Homo sapiens (Human))
Celltech R&D Inc.

Curated by ChEMBL
LigandPNGBDBM50219788(CHEMBL36797)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition against GRO-alpha driven human neutrophil chemotaxisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1/2(Homo sapiens (Human))
Celltech R&D Inc.

Curated by ChEMBL
LigandPNGBDBM50219791(CHEMBL35938)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition against GRO-alpha driven human neutrophil chemotaxisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1/2(Homo sapiens (Human))
Celltech R&D Inc.

Curated by ChEMBL
LigandPNGBDBM50113636(CHEMBL39835 | [5-(4-Fluoro-phenylcarbamoyl)-pyridi...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition against GRO-alpha driven human neutrophil chemotaxisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1/2(Homo sapiens (Human))
Celltech R&D Inc.

Curated by ChEMBL
LigandPNGBDBM50219807(CHEMBL288457)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition against GRO-alpha driven human neutrophil chemotaxisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed