TargetVitamin D3 receptor(Homo sapiens (Human))
Universidad de Santiago de Compostela
Curated by ChEMBL
Universidad de Santiago de Compostela
Curated by ChEMBL
Affinity DataIC50: 1.24nMAssay Description:Binding affinity to VDR assessed as inhibition of fluorescent ligand by fluorescence polarization competition assayMore data for this Ligand-Target Pair
TargetVitamin D3 receptor(Homo sapiens (Human))
Universidad de Santiago de Compostela
Curated by ChEMBL
Universidad de Santiago de Compostela
Curated by ChEMBL
Affinity DataIC50: 15.7nMAssay Description:Binding affinity to VDR assessed as inhibition of fluorescent ligand by fluorescence polarization competition assayMore data for this Ligand-Target Pair
TargetVitamin D3 receptor(Homo sapiens (Human))
Universidad de Santiago de Compostela
Curated by ChEMBL
Universidad de Santiago de Compostela
Curated by ChEMBL
Affinity DataIC50: 20.9nMAssay Description:Binding affinity to VDR assessed as inhibition of fluorescent ligand by fluorescence polarization competition assayMore data for this Ligand-Target Pair
TargetVitamin D3 receptor(Homo sapiens (Human))
Universidad de Santiago de Compostela
Curated by ChEMBL
Universidad de Santiago de Compostela
Curated by ChEMBL
Affinity DataIC50: 27.3nMAssay Description:Binding affinity to VDR assessed as inhibition of fluorescent ligand by fluorescence polarization competition assayMore data for this Ligand-Target Pair
TargetVitamin D3 receptor(Homo sapiens (Human))
Universidad de Santiago de Compostela
Curated by ChEMBL
Universidad de Santiago de Compostela
Curated by ChEMBL
Affinity DataEC50: 3.28nMAssay Description:Agonist activity at VDR in human MCF7 cells assessed as transcription of CYP24A1 gene after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetVitamin D3 receptor(Homo sapiens (Human))
Universidad de Santiago de Compostela
Curated by ChEMBL
Universidad de Santiago de Compostela
Curated by ChEMBL
Affinity DataEC50: 5.74nMAssay Description:Agonist activity at VDR in human MCF7 cells assessed as transcription of CYP24A1 gene after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetVitamin D3 receptor(Homo sapiens (Human))
Universidad de Santiago de Compostela
Curated by ChEMBL
Universidad de Santiago de Compostela
Curated by ChEMBL
Affinity DataEC50: 9.04nMAssay Description:Agonist activity at VDR in human MCF7 cells assessed as transcription of CYP24A1 gene after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetVitamin D3 receptor(Homo sapiens (Human))
Universidad de Santiago de Compostela
Curated by ChEMBL
Universidad de Santiago de Compostela
Curated by ChEMBL
Affinity DataEC50: 8.19nMAssay Description:Agonist activity at VDR in human MCF7 cells assessed as transcription of CYP24A1 gene after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
