Compile Data Set for Download or QSAR
maximum 50k data
Found 76 Enz. Inhib. hit(s) with all data for entry = 50048109
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM100152(7-methoxy-1-methyl-9H-beta-carboline;hydrochloride...)
Affinity DataIC50:  29nMAssay Description:Inhibition of DYRK1A (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM100152(7-methoxy-1-methyl-9H-beta-carboline;hydrochloride...)
Affinity DataIC50:  72nMAssay Description:Inhibition of CLK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50204658(CHEMBL3908596)
Affinity DataIC50:  700nMAssay Description:Inhibition of CLK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50204646(CHEMBL3962894)
Affinity DataIC50:  890nMAssay Description:Inhibition of CLK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50204644(CHEMBL3935442)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of CLK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50204647(CHEMBL3917542)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of CLK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50204653(CHEMBL3945429)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of CLK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I delta/epsilon(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM100152(7-methoxy-1-methyl-9H-beta-carboline;hydrochloride...)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of CK1 delta/epsilon (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50204659(CHEMBL3923825)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of CLK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50204658(CHEMBL3908596)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of DYRK1A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50204646(CHEMBL3962894)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of DYRK1A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50204644(CHEMBL3935442)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of DYRK1A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50204653(CHEMBL3945429)
Affinity DataIC50:  4.70E+3nMAssay Description:Inhibition of DYRK1A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50204659(CHEMBL3923825)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of DYRK1A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50204647(CHEMBL3917542)
Affinity DataIC50:  8.90E+3nMAssay Description:Inhibition of DYRK1A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50204643(CHEMBL3921647)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of GSK-3 alpha/beta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I delta/epsilon(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50204644(CHEMBL3935442)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CK1 delta/epsilon (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50204643(CHEMBL3921647)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CLK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50204649(CHEMBL3936539)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of DYRK1A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50204650(CHEMBL3912662)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of DYRK1A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50204642(CHEMBL3985735)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CLK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I delta/epsilon(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50204650(CHEMBL3912662)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CK1 delta/epsilon (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I delta/epsilon(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50204655(CHEMBL3902603)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CK1 delta/epsilon (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM100152(7-methoxy-1-methyl-9H-beta-carboline;hydrochloride...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of GSK-3 alpha/beta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50204654(CHEMBL3893635)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of DYRK1A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50204659(CHEMBL3923825)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of GSK-3 alpha/beta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I delta/epsilon(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50204643(CHEMBL3921647)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CK1 delta/epsilon (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I delta/epsilon(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50204652(CHEMBL3974565)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CK1 delta/epsilon (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50204657(CHEMBL3930589)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of DYRK1A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50204660(CHEMBL3939584)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of DYRK1A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50204644(CHEMBL3935442)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of GSK-3 alpha/beta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50204652(CHEMBL3974565)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of GSK-3 alpha/beta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50204655(CHEMBL3902603)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of DYRK1A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50204656(CHEMBL3903644)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CLK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50204645(CHEMBL3957926)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of DYRK1A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50204651(CHEMBL3911609)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of GSK-3 alpha/beta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I delta/epsilon(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50204658(CHEMBL3908596)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CK1 delta/epsilon (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50204650(CHEMBL3912662)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CLK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50204653(CHEMBL3945429)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of GSK-3 alpha/beta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50204656(CHEMBL3903644)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of GSK-3 alpha/beta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I delta/epsilon(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50204647(CHEMBL3917542)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CK1 delta/epsilon (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50204652(CHEMBL3974565)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CLK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I delta/epsilon(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50204653(CHEMBL3945429)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CK1 delta/epsilon (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50204649(CHEMBL3936539)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of GSK-3 alpha/beta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50204647(CHEMBL3917542)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of GSK-3 alpha/beta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I delta/epsilon(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50204656(CHEMBL3903644)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CK1 delta/epsilon (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50204650(CHEMBL3912662)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of GSK-3 alpha/beta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50204643(CHEMBL3921647)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of DYRK1A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I delta/epsilon(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50204642(CHEMBL3985735)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CK1 delta/epsilon (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50204658(CHEMBL3908596)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of GSK-3 alpha/beta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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