Compile Data Set for Download or QSAR
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Found 23 Enz. Inhib. hit(s) with all data for entry = 5237
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by PDSP Ki Database
LigandPNGBDBM50021325(4-methyl-(1S,5R,13R,14S)-12-oxa-4-azapentacyclo[9....)
Affinity DataKi:  0.400nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by PDSP Ki Database
LigandPNGBDBM50000788((morphine)4-methyl-(1S,5R,13R,14S,17R)-12-oxa-4-az...)
Affinity DataKi:  0.900nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by PDSP Ki Database
LigandPNGBDBM21015((2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl...)
Affinity DataKi:  1.10nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(GUINEA PIG)
Hungarian Academy Of Sciences

Curated by PDSP Ki Database
LigandPNGBDBM50000788((morphine)4-methyl-(1S,5R,13R,14S,17R)-12-oxa-4-az...)
Affinity DataKi:  1.40nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Hungarian Academy Of Sciences

Curated by PDSP Ki Database
LigandPNGBDBM21015((2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl...)
Affinity DataKi:  2.60nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by PDSP Ki Database
LigandPNGBDBM50016847(CHEMBL337041 | Cyprodime)
Affinity DataKi:  5.40nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Hungarian Academy Of Sciences

Curated by PDSP Ki Database
LigandPNGBDBM50021325(4-methyl-(1S,5R,13R,14S)-12-oxa-4-azapentacyclo[9....)
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(GUINEA PIG)
Hungarian Academy Of Sciences

Curated by PDSP Ki Database
LigandPNGBDBM50018708(2-{2-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propio...)
Affinity DataKi:  6.30nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by PDSP Ki Database
LigandPNGBDBM50016847(CHEMBL337041 | Cyprodime)
Affinity DataKi:  8.10nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by PDSP Ki Database
LigandPNGBDBM50018708(2-{2-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propio...)
Affinity DataKi:  9.80nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Hungarian Academy Of Sciences

Curated by PDSP Ki Database
LigandPNGBDBM50016847(CHEMBL337041 | Cyprodime)
Affinity DataKi:  26.6nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by PDSP Ki Database
LigandPNGBDBM50346948(CHEMBL1795717 | CTAP-NH2)
Affinity DataKi:  43.8nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Hungarian Academy Of Sciences

Curated by PDSP Ki Database
LigandPNGBDBM50346948(CHEMBL1795717 | CTAP-NH2)
Affinity DataKi:  48.1nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by PDSP Ki Database
LigandPNGBDBM81935(CAS_105618-26-6 | NSC_3034416 | Nor-BNI)
Affinity DataKi:  172nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by PDSP Ki Database
LigandPNGBDBM50169774(2-(3,4-Dichloro-phenyl)-N-methyl-N-(2-pyrrolidin-1...)
Affinity DataKi:  288nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Hungarian Academy Of Sciences

Curated by PDSP Ki Database
LigandPNGBDBM50169774(2-(3,4-Dichloro-phenyl)-N-methyl-N-(2-pyrrolidin-1...)
Affinity DataKi:  304nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Hungarian Academy Of Sciences

Curated by PDSP Ki Database
LigandPNGBDBM81935(CAS_105618-26-6 | NSC_3034416 | Nor-BNI)
Affinity DataKi:  770nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by PDSP Ki Database
LigandPNGBDBM50000507((R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-pheny...)
Affinity DataKi:  1.19E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by PDSP Ki Database
LigandPNGBDBM50057010((S)-4-((S)-2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-phen...)
Affinity DataKi:  1.90E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by PDSP Ki Database
LigandPNGBDBM50016847(CHEMBL337041 | Cyprodime)
Affinity DataKi:  2.19E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by PDSP Ki Database
LigandPNGBDBM50041958(2-(1-{2-[2-amino-3-(4-hydroxyphenyl)propanoyl]-1,2...)
Affinity DataKi:  2.83E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(GUINEA PIG)
Hungarian Academy Of Sciences

Curated by PDSP Ki Database
LigandPNGBDBM50000507((R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-pheny...)
Affinity DataKi:  2.88E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(GUINEA PIG)
Hungarian Academy Of Sciences

Curated by PDSP Ki Database
LigandPNGBDBM50041958(2-(1-{2-[2-amino-3-(4-hydroxyphenyl)propanoyl]-1,2...)
Affinity DataKi:  7.06E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed