Compile Data Set for Download or QSAR
maximum 50k data
Found 63 Enz. Inhib. hit(s) with all data for entry = 5280
TargetAlpha-2C adrenergic receptor(RAT)
Centre De Recherches De Croissy

Curated by PDSP Ki Database
LigandPNGBDBM85709(S18616)
Affinity DataKi:  0.159nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2A adrenergic receptor [16-465](Rattus norvegicus (rat))
Centre De Recherches De Croissy

Curated by PDSP Ki Database
LigandPNGBDBM85709(S18616)
Affinity DataKi:  0.251nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Centre De Recherches De Croissy

Curated by PDSP Ki Database
LigandPNGBDBM85709(S18616)
Affinity DataKi:  0.251nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Centre De Recherches De Croissy

Curated by PDSP Ki Database
LigandPNGBDBM85709(S18616)
Affinity DataKi:  0.316nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Centre De Recherches De Croissy

Curated by PDSP Ki Database
LigandPNGBDBM85709(S18616)
Affinity DataKi:  0.346nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Centre De Recherches De Croissy

Curated by PDSP Ki Database
LigandPNGBDBM85709(S18616)
Affinity DataKi:  0.562nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Centre De Recherches De Croissy

Curated by PDSP Ki Database
LigandPNGBDBM85709(S18616)
Affinity DataKi:  0.631nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2C adrenergic receptor(RAT)
Centre De Recherches De Croissy

Curated by PDSP Ki Database
LigandPNGBDBM50241196((R)-5-(1-(2,3-dimethylphenyl)ethyl)-1H-imidazole |...)
In DepthDetails PubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Centre De Recherches De Croissy

Curated by PDSP Ki Database
LigandPNGBDBM50241196((R)-5-(1-(2,3-dimethylphenyl)ethyl)-1H-imidazole |...)
Affinity DataKi:  2.00nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Centre De Recherches De Croissy

Curated by PDSP Ki Database
LigandPNGBDBM50241196((R)-5-(1-(2,3-dimethylphenyl)ethyl)-1H-imidazole |...)
Affinity DataKi:  2.04nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Centre De Recherches De Croissy

Curated by PDSP Ki Database
LigandPNGBDBM50241196((R)-5-(1-(2,3-dimethylphenyl)ethyl)-1H-imidazole |...)
Affinity DataKi:  2.51nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Centre De Recherches De Croissy

Curated by PDSP Ki Database
LigandPNGBDBM50241196((R)-5-(1-(2,3-dimethylphenyl)ethyl)-1H-imidazole |...)
Affinity DataKi:  3.16nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Centre De Recherches De Croissy

Curated by PDSP Ki Database
LigandPNGBDBM85709(S18616)
Affinity DataKi:  3.98nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Centre De Recherches De Croissy

Curated by PDSP Ki Database
LigandPNGBDBM85709(S18616)
Affinity DataKi:  4.37nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Centre De Recherches De Croissy

Curated by PDSP Ki Database
LigandPNGBDBM85709(S18616)
Affinity DataKi:  6.03nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Centre De Recherches De Croissy

Curated by PDSP Ki Database
LigandPNGBDBM85709(S18616)
Affinity DataKi:  6.31nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Centre De Recherches De Croissy

Curated by PDSP Ki Database
LigandPNGBDBM50241196((R)-5-(1-(2,3-dimethylphenyl)ethyl)-1H-imidazole |...)
Affinity DataKi:  15.1nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Centre De Recherches De Croissy

Curated by PDSP Ki Database
LigandPNGBDBM50241196((R)-5-(1-(2,3-dimethylphenyl)ethyl)-1H-imidazole |...)
Affinity DataKi:  15.8nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Centre De Recherches De Croissy

Curated by PDSP Ki Database
LigandPNGBDBM50241196((R)-5-(1-(2,3-dimethylphenyl)ethyl)-1H-imidazole |...)
Affinity DataKi:  19.5nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Centre De Recherches De Croissy

Curated by PDSP Ki Database
LigandPNGBDBM85709(S18616)
Affinity DataKi:  20.0nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Centre De Recherches De Croissy

Curated by PDSP Ki Database
LigandPNGBDBM85709(S18616)
Affinity DataKi:  25.1nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2A adrenergic receptor [16-465](Rattus norvegicus (rat))
Centre De Recherches De Croissy

Curated by PDSP Ki Database
LigandPNGBDBM50016897(2-(2,6-dichloroanilino)-1,3-diazacyclopentene-(2) ...)
Affinity DataKi:  25.1nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNischarin(BOVINE)
Centre De Recherches De Croissy

Curated by PDSP Ki Database
LigandPNGBDBM50016897(2-(2,6-dichloroanilino)-1,3-diazacyclopentene-(2) ...)
Affinity DataKi:  31.6nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Centre De Recherches De Croissy

Curated by PDSP Ki Database
LigandPNGBDBM50016897(2-(2,6-dichloroanilino)-1,3-diazacyclopentene-(2) ...)
Affinity DataKi:  31.6nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2C adrenergic receptor(RAT)
Centre De Recherches De Croissy

Curated by PDSP Ki Database
LigandPNGBDBM50016897(2-(2,6-dichloroanilino)-1,3-diazacyclopentene-(2) ...)
Affinity DataKi:  31.6nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Centre De Recherches De Croissy

Curated by PDSP Ki Database
LigandPNGBDBM50016897(2-(2,6-dichloroanilino)-1,3-diazacyclopentene-(2) ...)
Affinity DataKi:  35.5nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Centre De Recherches De Croissy

Curated by PDSP Ki Database
LigandPNGBDBM50016897(2-(2,6-dichloroanilino)-1,3-diazacyclopentene-(2) ...)
Affinity DataKi:  39.8nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNischarin(BOVINE)
Centre De Recherches De Croissy

Curated by PDSP Ki Database
LigandPNGBDBM85709(S18616)
Affinity DataKi:  39.8nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNischarin(RAT)
Centre De Recherches De Croissy

Curated by PDSP Ki Database
LigandPNGBDBM50241196((R)-5-(1-(2,3-dimethylphenyl)ethyl)-1H-imidazole |...)
Affinity DataKi:  50.1nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Centre De Recherches De Croissy

Curated by PDSP Ki Database
LigandPNGBDBM50016897(2-(2,6-dichloroanilino)-1,3-diazacyclopentene-(2) ...)
Affinity DataKi:  50.1nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Centre De Recherches De Croissy

Curated by PDSP Ki Database
LigandPNGBDBM50016897(2-(2,6-dichloroanilino)-1,3-diazacyclopentene-(2) ...)
Affinity DataKi:  63.1nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Centre De Recherches De Croissy

Curated by PDSP Ki Database
LigandPNGBDBM50241196((R)-5-(1-(2,3-dimethylphenyl)ethyl)-1H-imidazole |...)
Affinity DataKi:  63.1nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Centre De Recherches De Croissy

Curated by PDSP Ki Database
LigandPNGBDBM50241196((R)-5-(1-(2,3-dimethylphenyl)ethyl)-1H-imidazole |...)
Affinity DataKi:  79.4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Centre De Recherches De Croissy

Curated by PDSP Ki Database
LigandPNGBDBM85709(S18616)
Affinity DataKi:  79.4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNischarin(RAT)
Centre De Recherches De Croissy

Curated by PDSP Ki Database
LigandPNGBDBM85709(S18616)
Affinity DataKi:  79.4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Centre De Recherches De Croissy

Curated by PDSP Ki Database
LigandPNGBDBM50016897(2-(2,6-dichloroanilino)-1,3-diazacyclopentene-(2) ...)
Affinity DataKi:  100nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
Centre De Recherches De Croissy

Curated by PDSP Ki Database
LigandPNGBDBM85709(S18616)
Affinity DataKi:  100nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Centre De Recherches De Croissy

Curated by PDSP Ki Database
LigandPNGBDBM50016897(2-(2,6-dichloroanilino)-1,3-diazacyclopentene-(2) ...)
Affinity DataKi:  126nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNischarin(BOVINE)
Centre De Recherches De Croissy

Curated by PDSP Ki Database
LigandPNGBDBM50241196((R)-5-(1-(2,3-dimethylphenyl)ethyl)-1H-imidazole |...)
Affinity DataKi:  200nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Centre De Recherches De Croissy

Curated by PDSP Ki Database
LigandPNGBDBM50241196((R)-5-(1-(2,3-dimethylphenyl)ethyl)-1H-imidazole |...)
Affinity DataKi:  200nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Centre De Recherches De Croissy

Curated by PDSP Ki Database
LigandPNGBDBM50016897(2-(2,6-dichloroanilino)-1,3-diazacyclopentene-(2) ...)
Affinity DataKi:  309nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Centre De Recherches De Croissy

Curated by PDSP Ki Database
LigandPNGBDBM50016897(2-(2,6-dichloroanilino)-1,3-diazacyclopentene-(2) ...)
Affinity DataKi:  316nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
Centre De Recherches De Croissy

Curated by PDSP Ki Database
LigandPNGBDBM50016897(2-(2,6-dichloroanilino)-1,3-diazacyclopentene-(2) ...)
Affinity DataKi:  316nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Centre De Recherches De Croissy

Curated by PDSP Ki Database
LigandPNGBDBM50016897(2-(2,6-dichloroanilino)-1,3-diazacyclopentene-(2) ...)
Affinity DataKi:  316nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Centre De Recherches De Croissy

Curated by PDSP Ki Database
LigandPNGBDBM50241196((R)-5-(1-(2,3-dimethylphenyl)ethyl)-1H-imidazole |...)
Affinity DataKi:  316nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
Centre De Recherches De Croissy

Curated by PDSP Ki Database
LigandPNGBDBM50241196((R)-5-(1-(2,3-dimethylphenyl)ethyl)-1H-imidazole |...)
Affinity DataKi:  316nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Centre De Recherches De Croissy

Curated by PDSP Ki Database
LigandPNGBDBM50241196((R)-5-(1-(2,3-dimethylphenyl)ethyl)-1H-imidazole |...)
Affinity DataKi:  316nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Centre De Recherches De Croissy

Curated by PDSP Ki Database
LigandPNGBDBM35234(DL-[7-3H]norepinephrine | NOREPINEPHRINE | Noradre...)
Affinity DataKi:  331nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Centre De Recherches De Croissy

Curated by PDSP Ki Database
LigandPNGBDBM35234(DL-[7-3H]norepinephrine | NOREPINEPHRINE | Noradre...)
Affinity DataKi:  398nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Centre De Recherches De Croissy

Curated by PDSP Ki Database
LigandPNGBDBM50016897(2-(2,6-dichloroanilino)-1,3-diazacyclopentene-(2) ...)
Affinity DataKi:  501nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
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