Affinity DataEC50: 0.0490nMAssay Description:Antagonist activity at human recombinant NK1 receptor expressed in CHO cells assessed as inhibition of NPS-induced intracellular calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0575nMAssay Description:Antagonist activity at human recombinant NK1 receptor expressed in CHO cells assessed as inhibition of NPS-induced intracellular calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataEC50: 0.600nMAssay Description:Agonist activity at wild type human NK1 receptor expressed in HEK293 cells assessed as increase in [3H]IP accumulation after 20 minsMore data for this Ligand-Target Pair
Affinity DataEC50: 0.600nMAssay Description:Agonist activity at bfSPR to produce increase in intracellular [Ca2+]More data for this Ligand-Target Pair
Affinity DataEC50: 0.600nMAssay Description:SP-induced [Ca2+] mobilization in CHO cells expressing human Tachykinin receptor 1More data for this Ligand-Target Pair
Affinity DataEC50: 0.600nMAssay Description:SP-induced [Ca2+] mobilization in CHO cells expressing human Tachykinin receptor 1More data for this Ligand-Target Pair
Affinity DataEC50: 1nMAssay Description:Agonist activity at bfSPR to produce increase in intracellular [Ca2+]More data for this Ligand-Target Pair
Affinity DataEC50: 5nMAssay Description:Tested for the biological activity and selectivity against NK-1 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 11nMAssay Description:Tested for the biological activity and selectivity against NK-1 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 13.5nMAssay Description:Agonist activity at bfSPR to produce increase in intracellular [Ca2+]More data for this Ligand-Target Pair
Affinity DataEC50: 14nMAssay Description:SP-induced [Ca2+] mobilization in CHO cells expressing human Tachykinin receptor 1More data for this Ligand-Target Pair
Affinity DataEC50: 14nMAssay Description:SP-induced [Ca2+] mobilization in CHO cells expressing human Tachykinin receptor 1More data for this Ligand-Target Pair
Affinity DataEC50: 14nMAssay Description:Agonist activity at bfSPR to produce increase in intracellular [Ca2+]More data for this Ligand-Target Pair
Affinity DataEC50: 24.4nMAssay Description:Displacement of [3H]SR140333 from human recombinant NK1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 180nMAssay Description:Tested for the biological activity and selectivity against NK-1 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 5.30E+3nMAssay Description:Binding affinity to NK1R (unknown origin) expressed in HEK293 cells assessed as reduction in cell viability incubated for 96 hrs by MTT assayMore data for this Ligand-Target Pair
Affinity DataEC50: 7.20E+3nMAssay Description:Binding affinity to NK1R (unknown origin) expressed in HEK293 cells assessed as reduction in cell viability incubated for 96 hrs by MTT assayMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Tested for the biological activity and selectivity against NK-1 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: >5.00E+4nMAssay Description:Agonist activity at NK1 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 3.50E+5nMAssay Description:Partial agonist activity at His6-tagged NK1 receptor (unknown origin) expressed in CHO cells assessed as IP1 accumulation measured after 30 mins by H...More data for this Ligand-Target Pair