Compile Data Set for Download or QSAR
maximum 50k data
Found 241 of ec50 data for polymerid = 2125,50000659
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Mayo Clinic

Curated by ChEMBL
LigandPNGBDBM50329178((S)-3-(3-(1-(2-(isopropyl(phenyl)amino)-2-oxoethyl...)
Affinity DataEC50:  0.00200nMAssay Description:Activity at CCK1R (unknown origin) expressed in CHO cells assessed as CCK EC50 measured as intracellular calcium responses at 0.316 nM (Rvb = 7 to 14...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Mayo Clinic

Curated by ChEMBL
LigandPNGBDBM50329178((S)-3-(3-(1-(2-(isopropyl(phenyl)amino)-2-oxoethyl...)
Affinity DataEC50:  0.0100nMAssay Description:Activity at CCK1R (unknown origin) expressed in CHO cells assessed as CCK EC50 measured as intracellular calcium responses at 0.1 nM (Rvb = 7 to 14 p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Mayo Clinic

Curated by ChEMBL
LigandPNGBDBM50329178((S)-3-(3-(1-(2-(isopropyl(phenyl)amino)-2-oxoethyl...)
Affinity DataEC50:  0.0130nMAssay Description:Activity at CCK1R (unknown origin) expressed in CHO cells assessed as CCK EC50 measured as intracellular calcium responses at 0.01 nM (Rvb = 7 to 14 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Mayo Clinic

Curated by ChEMBL
LigandPNGBDBM50074832(CHEMBL156605)
Affinity DataEC50:  0.0140nMAssay Description:Activity at CCK1R (unknown origin) expressed in CHO cells assessed as CCK EC50 measured as intracellular calcium responses at 100 nM (Rvb = 7 to 14 p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Mayo Clinic

Curated by ChEMBL
LigandPNGBDBM50074832(CHEMBL156605)
Affinity DataEC50:  0.0190nMAssay Description:Activity at CCK1R (unknown origin) expressed in CHO cells assessed as CCK EC50 measured as intracellular calcium responses at 10 nM (Rvb = 7 to 14 pM...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Mayo Clinic

Curated by ChEMBL
LigandPNGBDBM50072419(2-[2,4-Dioxo-5-phenyl-3-(3-phenyl-ureido)-2,3,4,5-...)
Affinity DataEC50:  0.0200nMAssay Description:Activity at CCK1R (unknown origin) expressed in CHO cells assessed as CCK EC50 measured as intracellular calcium responses at 10 nM (Rvb = 7 to 14 pM...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Mayo Clinic

Curated by ChEMBL
LigandPNGBDBM50061829((R)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-({(S)-2-[...)
Affinity DataEC50:  0.0251nMAssay Description:Agonist activity at human CCK1R expressed in human 1321N1 cells assessed as IP1 accumulation after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Mayo Clinic

Curated by ChEMBL
LigandPNGBDBM50245189(3-((R)-3-(acetamidomethyl)-4-(1-(3-ethoxyphenyl)-2...)
Affinity DataEC50:  0.0330nMAssay Description:Agonist activity at human CCK1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Mayo Clinic

Curated by ChEMBL
LigandPNGBDBM50245188(3-((S)-3-((carboxymethoxy)methyl)-4-(1-(3-ethoxyph...)
Affinity DataEC50:  0.0340nMAssay Description:Agonist activity at human CCK1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Mus musculus)
Merck

Curated by ChEMBL
LigandPNGBDBM50245192(3-((S)-4-(1-(3-ethoxyphenyl)-2-(2-fluoro-4-methylp...)
Affinity DataEC50:  0.0340nMAssay Description:Agonist activity at mouse CCK1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Mayo Clinic

Curated by ChEMBL
LigandPNGBDBM50074832(CHEMBL156605)
Affinity DataEC50:  0.0390nMAssay Description:Activity at CCK1R (unknown origin) expressed in CHO cells assessed as CCK EC50 measured as intracellular calcium responses at 1000 nM (Rvb = 7 to 14 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Mayo Clinic

Curated by ChEMBL
LigandPNGBDBM50245182(3-((S)-3-(acetamidomethyl)-4-(1-(3-ethoxyphenyl)-2...)
Affinity DataEC50:  0.0400nMAssay Description:Agonist activity at human CCK1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Mayo Clinic

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataEC50:  0.0437nMAssay Description:Agonist activity at human CCK1R expressed in human 1321N1 cells assessed as IP1 accumulation after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Mayo Clinic

Curated by ChEMBL
LigandPNGBDBM50263226(3-(4-(1-(3-ethoxyphenyl)-2-(4-fluorophenyl)-1H-imi...)
Affinity DataEC50:  0.0480nMAssay Description:Agonist activity against human CCK1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Mayo Clinic

Curated by ChEMBL
LigandPNGBDBM50072419(2-[2,4-Dioxo-5-phenyl-3-(3-phenyl-ureido)-2,3,4,5-...)
Affinity DataEC50:  0.0510nMAssay Description:Activity at CCK1R (unknown origin) expressed in CHO cells assessed as CCK EC50 measured as intracellular calcium responses at 100 nM (Rvb = 7 to 14 p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Mayo Clinic

Curated by ChEMBL
LigandPNGBDBM50263227(3-(4-(2-(2,4-difluorophenyl)-1-(3-ethoxyphenyl)-1H...)
Affinity DataEC50:  0.0530nMAssay Description:Agonist activity against human CCK1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Mayo Clinic

Curated by ChEMBL
LigandPNGBDBM50245186(3-((S)-4-(1-(3-ethoxyphenyl)-2-p-tolyl-1H-imidazol...)
Affinity DataEC50:  0.0530nMAssay Description:Agonist activity at human CCK1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Mayo Clinic

Curated by ChEMBL
LigandPNGBDBM50245187(3-(4-(1-(3-ethoxyphenyl)-2-(2-fluoro-4-methylpheny...)
Affinity DataEC50:  0.0550nMAssay Description:Agonist activity at human CCK1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Mayo Clinic

Curated by ChEMBL
LigandPNGBDBM50245187(3-(4-(1-(3-ethoxyphenyl)-2-(2-fluoro-4-methylpheny...)
Affinity DataEC50:  0.0560nMAssay Description:Agonist activity against human CCK1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Mayo Clinic

Curated by ChEMBL
LigandPNGBDBM50517380(CHEMBL4464703)
Affinity DataEC50:  0.0603nMAssay Description:Agonist activity at human CCK1R expressed in human 1321N1 cells assessed as IP1 accumulation after 1 hr by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Mayo Clinic

Curated by ChEMBL
LigandPNGBDBM50343721(3-(4-(4-(2-fluoro-4-methylphenyl)-5-(4-methoxyphen...)
Affinity DataEC50:  0.0630nMAssay Description:Agonist activity at human CCK1 receptor expressed in CHO Flip cells assessed as increase of radio labeled inositol phosphate accumulation by Wallac m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Mayo Clinic

Curated by ChEMBL
LigandPNGBDBM50343722(3-(4-(5-(2,3-dihydrobenzo[b][1,4]dioxin-6-yl)-4-(2...)
Affinity DataEC50:  0.0650nMAssay Description:Agonist activity at human CCK1 receptor expressed in CHO Flip cells assessed as increase of radio labeled inositol phosphate accumulation by Wallac m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Mayo Clinic

Curated by ChEMBL
LigandPNGBDBM50245201(3-(((S)-1-(1-(3-ethoxyphenyl)-2-p-tolyl-1H-imidazo...)
Affinity DataEC50:  0.0650nMAssay Description:Agonist activity at human CCK1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Mayo Clinic

Curated by ChEMBL
LigandPNGBDBM50517379(CHEMBL4453982)
Affinity DataEC50:  0.0676nMAssay Description:Agonist activity at human CCK1R expressed in human 1321N1 cells assessed as IP1 accumulation after 1 hr by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Mayo Clinic

Curated by ChEMBL
LigandPNGBDBM50245192(3-((S)-4-(1-(3-ethoxyphenyl)-2-(2-fluoro-4-methylp...)
Affinity DataEC50:  0.0710nMAssay Description:Agonist activity at human CCK1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Mayo Clinic

Curated by ChEMBL
LigandPNGBDBM50245191(3-((R)-4-(1-(3-ethoxyphenyl)-2-(2-fluoro-4-methylp...)
Affinity DataEC50:  0.0740nMAssay Description:Agonist activity at human CCK1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Mayo Clinic

Curated by ChEMBL
LigandPNGBDBM50263230(3-(4-(1-(2,3-dihydrobenzo[b][1,4]dioxin-6-yl)-2-(2...)
Affinity DataEC50:  0.0770nMAssay Description:Agonist activity against human CCK1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Mayo Clinic

Curated by ChEMBL
LigandPNGBDBM50262862(3-(4-(1-(3-methoxyphenyl)-2-p-tolyl-1H-imidazole-4...)
Affinity DataEC50:  0.0780nMAssay Description:Agonist activity against human CCK1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Mayo Clinic

Curated by ChEMBL
LigandPNGBDBM50245185(3-((R)-4-(1-(3-ethoxyphenyl)-2-p-tolyl-1H-imidazol...)
Affinity DataEC50:  0.0820nMAssay Description:Agonist activity at human CCK1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Mayo Clinic

Curated by ChEMBL
LigandPNGBDBM50245205(2-((S)-1-(1-(3-ethoxyphenyl)-2-p-tolyl-1H-imidazol...)
Affinity DataEC50:  0.0890nMAssay Description:Agonist activity at human CCK1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Mayo Clinic

Curated by ChEMBL
LigandPNGBDBM50263229(3-(4-(1-(2,3-dihydrobenzo[b][1,4]dioxin-6-yl)-2-(4...)
Affinity DataEC50:  0.0930nMAssay Description:Agonist activity against human CCK1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Mayo Clinic

Curated by ChEMBL
LigandPNGBDBM50245180(3-(4-(1-(3-ethoxyphenyl)-2-p-tolyl-1H-imidazole-4-...)
Affinity DataEC50:  0.0940nMAssay Description:Agonist activity against human CCK1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Mayo Clinic

Curated by ChEMBL
LigandPNGBDBM50245180(3-(4-(1-(3-ethoxyphenyl)-2-p-tolyl-1H-imidazole-4-...)
Affinity DataEC50:  0.0940nMAssay Description:Agonist activity at human CCK1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Mayo Clinic

Curated by ChEMBL
LigandPNGBDBM50245183(3-((R)-4-(1-(3-ethoxyphenyl)-2-p-tolyl-1H-imidazol...)
Affinity DataEC50:  0.0950nMAssay Description:Agonist activity at human CCK1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Mayo Clinic

Curated by ChEMBL
LigandPNGBDBM50245195(2-(((R)-1-(1-(3-ethoxyphenyl)-2-p-tolyl-1H-imidazo...)
Affinity DataEC50:  0.0970nMAssay Description:Agonist activity at human CCK1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Mayo Clinic

Curated by ChEMBL
LigandPNGBDBM50245181(3-((R)-3-((carboxymethoxy)methyl)-4-(1-(3-ethoxyph...)
Affinity DataEC50:  0.0970nMAssay Description:Agonist activity at human CCK1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Mayo Clinic

Curated by ChEMBL
LigandPNGBDBM50245202(CHEMBL503331 | N-(((R)-1-(1-(3-ethoxyphenyl)-2-p-t...)
Affinity DataEC50:  0.0970nMAssay Description:Agonist activity at human CCK1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Mayo Clinic

Curated by ChEMBL
LigandPNGBDBM50245190(3-((S)-4-(1-(3-ethoxyphenyl)-2-(2-fluoro-4-methylp...)
Affinity DataEC50:  0.100nMAssay Description:Agonist activity at human CCK1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Mayo Clinic

Curated by ChEMBL
LigandPNGBDBM50245196(CHEMBL450443 | N-(((S)-1-(1-(3-ethoxyphenyl)-2-p-t...)
Affinity DataEC50:  0.100nMAssay Description:Agonist activity at human CCK1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Mayo Clinic

Curated by ChEMBL
LigandPNGBDBM50517371(CHEMBL4475304)
Affinity DataEC50:  0.107nMAssay Description:Agonist activity at human CCK1R expressed in human 1321N1 cells assessed as IP1 accumulation after 1 hr by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Mayo Clinic

Curated by ChEMBL
LigandPNGBDBM50517355(CHEMBL4471525)
Affinity DataEC50:  0.107nMAssay Description:Agonist activity at human CCK1R expressed in human 1321N1 cells assessed as IP1 accumulation after 1 hr by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Mayo Clinic

Curated by ChEMBL
LigandPNGBDBM50517331(CHEMBL4467338)
Affinity DataEC50:  0.110nMAssay Description:Agonist activity at human CCK1R expressed in human 1321N1 cells assessed as IP1 accumulation after 1 hr by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Mus musculus)
Merck

Curated by ChEMBL
LigandPNGBDBM50245186(3-((S)-4-(1-(3-ethoxyphenyl)-2-p-tolyl-1H-imidazol...)
Affinity DataEC50:  0.110nMAssay Description:Agonist activity at mouse CCK1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Mus musculus)
Merck

Curated by ChEMBL
LigandPNGBDBM50245205(2-((S)-1-(1-(3-ethoxyphenyl)-2-p-tolyl-1H-imidazol...)
Affinity DataEC50:  0.110nMAssay Description:Agonist activity at mouse CCK1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Mayo Clinic

Curated by ChEMBL
LigandPNGBDBM50517339(CHEMBL4551834)
Affinity DataEC50:  0.115nMAssay Description:Agonist activity at human CCK1R expressed in human 1321N1 cells assessed as IP1 accumulation after 1 hr by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Mayo Clinic

Curated by ChEMBL
LigandPNGBDBM50517356(CHEMBL4557012)
Affinity DataEC50:  0.115nMAssay Description:Agonist activity at human CCK1R expressed in human 1321N1 cells assessed as IP1 accumulation after 1 hr by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Mayo Clinic

Curated by ChEMBL
LigandPNGBDBM50263186((1-(2,3-dihydrobenzo[b][1,4]dioxin-6-yl)-2-p-tolyl...)
Affinity DataEC50:  0.120nMAssay Description:Agonist activity against human CCK1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Mus musculus)
Merck

Curated by ChEMBL
LigandPNGBDBM50343722(3-(4-(5-(2,3-dihydrobenzo[b][1,4]dioxin-6-yl)-4-(2...)
Affinity DataEC50:  0.120nMAssay Description:Agonist activity at mouse CCK1 receptor expressed in CHO Flip cells assessed as increase in radio labeled inositol phosphate accumulation by Wallac m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Mayo Clinic

Curated by ChEMBL
LigandPNGBDBM50072419(2-[2,4-Dioxo-5-phenyl-3-(3-phenyl-ureido)-2,3,4,5-...)
Affinity DataEC50:  0.120nMAssay Description:Activity at CCK1R (unknown origin) expressed in CHO cells assessed as CCK EC50 measured as intracellular calcium responses at 1000 nM (Rvb = 7 to 14 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Mayo Clinic

Curated by ChEMBL
LigandPNGBDBM50380728(CHEMBL2017835)
Affinity DataEC50:  0.120nMAssay Description:Agonist activity at human CCK1R T3.28V, T3.29S mutant expressed in CHO cells assessed as intracellular calcium response by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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