Compile Data Set for Download or QSAR
maximum 50k data
Found 8 of ec50 data for polymerid = 49000302
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50275902(CHEMBL525577 | D-Phe-Gln-Trp-Ala-Val-b-Ala-His-Phe...)
Affinity DataEC50:  0.0600nMAssay Description:Agonist activity at recombinant gastrin releasing peptide receptor (unknown origin) expressed in baculovirus-transduced HEK293 cells assessed as intr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM85484(Bombesin)
Affinity DataEC50:  0.258nMAssay Description:Displacement of 125I[Tyr4]-bombesin from GRPR expressed in human PC3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50374870(CHEMBL272335)
Affinity DataEC50:  0.373nMAssay Description:Displacement of 125I[Tyr4]-bombesin from GRPR expressed in human PC3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50127532(CHEMBL438926 | Val-Pro-Leu-Pro-Ala-Gly-Gly-Gly-Thr...)
Affinity DataEC50:  34nMAssay Description:Effective concentration required against gastrin releasing peptide receptor (GRP-R) in CHO cells by using FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50071745(CHEMBL403317 | Compound NMB | Gly-Asn-Leu-Trp-Ala-...)
Affinity DataEC50:  41nMAssay Description:Effective concentration required against gastrin releasing peptide receptor (GRP-R) in CHO cells by using FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50127519(CHEMBL262992 | [D-Tyr6-, Beta-Ala11, Phe13, Nle14]...)
Affinity DataEC50:  84nMAssay Description:Effective concentration required against gastrin releasing peptide receptor (GRP-R) in CHO cells by using FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50127535(2-[2-(4-Chloro-phenyl)-acetylamino]-pentanedioic a...)
Affinity DataEC50:  1.22E+4nMAssay Description:Effective concentration required against gastrin releasing peptide receptor (GRP-R) in CHO cells by using FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50127522(2-Phenylacetylamino-pentanedioic acid 5-amide 1-{[...)
Affinity DataEC50:  1.91E+4nMAssay Description:Effective concentration required against gastrin releasing peptide receptor (GRP-R) in CHO cells by using FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed