Affinity DataEC50: 0.0200nMAssay Description:Agonist activity at delta-opioid receptor in mouse vas deferensMore data for this Ligand-Target Pair
Affinity DataEC50: 0.331nMAssay Description:Negative logarithm of the molar concentration of delta receptor was determined in mouse vas deferensMore data for this Ligand-Target Pair
Affinity DataEC50: 0.360nMAssay Description:Effective concentration was measured towards delta opioid receptor using mouse vas deferens(MVD, delta) bioassay in vitroMore data for this Ligand-Target Pair
Affinity DataEC50: 0.660nMAssay Description:Effective concentration was measured towards delta opioid receptor using mouse vas deferens(MVD, delta) bioassay in vitroMore data for this Ligand-Target Pair
Affinity DataEC50: 0.830nMAssay Description:Agonist activity at mouse delta opioid receptor-1 expressed in CHO cell membranes assessed as [35S]GTPgammaS binding incubated for 60 mins by scintil...More data for this Ligand-Target Pair
Affinity DataEC50: 0.900nMAssay Description:Activity against delta opioid receptor by stimulation of [35S]GTPgammaS binding in CHO-hgamma cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 1.80nMAssay Description:In vitro bioassay data to determine the effective concentration required for antagonistic activity against Opioid receptor delta 1 in functional assa...More data for this Ligand-Target Pair
Affinity DataEC50: 1.80nMAssay Description:Tested for electrically induced smooth muscle contractions from mouse vas deferens expressed in delta opioid receptorsMore data for this Ligand-Target Pair
Affinity DataEC50: 2.10nMAssay Description:Agonist activity at mouse cloned delta opioid receptor expressed in CHO cells after 60 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2.60nMAssay Description:Agonist activity at delta-opioid receptor in mouse vas deferensMore data for this Ligand-Target Pair
Affinity DataEC50: 3nMAssay Description:Activity against delta opioid receptor by stimulation of [35S]GTPgammaS binding in CHO-hgamma cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 3nMAssay Description:Agonist activity at delta-opioid receptor in mouse vas deferensMore data for this Ligand-Target Pair
Affinity DataEC50: 4.10nMAssay Description:Effective concentration was measured towards delta opioid receptor using mouse vas deferens(MVD, delta) bioassay in vitroMore data for this Ligand-Target Pair
Affinity DataEC50: 4.10nMAssay Description:In vitro bioassay data to determine the effective concentration required for antagonistic activity against Opioid receptor delta 1 in functional assa...More data for this Ligand-Target Pair
Affinity DataEC50: 4.40nMAssay Description:Agonist activity at mouse DOR expressed in CHO cells after 1.5 hrs by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 7.10nMAssay Description:Agonist activity at mouse delta opioid receptor expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 7.70nMAssay Description:Agonist activity at mouse delta opioid receptor expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 9.10nMAssay Description:Agonist activity at mouse cloned delta opioid receptor expressed in CHO cells after 60 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 10nMAssay Description:Agonist activity at mouse delta opioid receptor-1 expressed in CHO cell membranes assessed as [35S]GTPgammaS binding incubated for 60 mins by scintil...More data for this Ligand-Target Pair
Affinity DataEC50: 19nMAssay Description:Activity against delta opioid receptor by stimulation of [35S]GTPgammaS binding in CHO-hgamma cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 22nMAssay Description:Activity against delta opioid receptor by stimulation of [35S]GTPgammaS binding in CHO-hgamma cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 33nMAssay Description:Agonist activity at mouse DOR expressed in CHO cells after 1.5 hrs by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 35nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electric-field induced measured after 5 minsMore data for this Ligand-Target Pair
Affinity DataEC50: 37nMAssay Description:Activity against delta opioid receptor by stimulation of [35S]GTPgammaS binding in CHO-hgamma cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 74nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electric-field induced measured after 5 minsMore data for this Ligand-Target Pair
Affinity DataEC50: 91nMAssay Description:Agonist activity at mouse delta opioid receptor expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 99nMAssay Description:Agonist activity at mouse DOR expressed in CHO cells after 1.5 hrs by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 108nMAssay Description:Agonist activity at mouse DOR expressed in CHO cells after 1.5 hrs by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 126nMAssay Description:Agonist activity at DOR in CD1 mouse vas deferens assessed as inhibition of EFS-induced contractions incubated for 60 minsMore data for this Ligand-Target Pair
Affinity DataEC50: 135nMAssay Description:Activity against delta opioid receptor by stimulation of [35S]GTPgammaS binding in CHO-hgamma cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 140nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electric-field induced measured after 5 minsMore data for this Ligand-Target Pair
Affinity DataEC50: 168nMAssay Description:Effective concentration was measured towards delta opioid receptor using mouse vas deferens(MVD, delta) bioassay in vitroMore data for this Ligand-Target Pair
Affinity DataEC50: 170nMAssay Description:In vitro bioassay data to determine the effective concentration required for antagonistic activity against Opioid receptor delta 1 in functional assa...More data for this Ligand-Target Pair
Affinity DataEC50: 174nMAssay Description:Tested for electrically induced smooth muscle contractions from mouse vas deferens expressed in delta opioid receptorsMore data for this Ligand-Target Pair
Affinity DataEC50: 210nMAssay Description:Tested for electrically induced smooth muscle contractions from mouse vas deferens expressed in delta opioid receptorsMore data for this Ligand-Target Pair
Affinity DataEC50: 210nMAssay Description:Tested for electrically induced smooth muscle contractions from mouse vas deferens expressed in delta opioid receptorsMore data for this Ligand-Target Pair
Affinity DataEC50: 360nMAssay Description:Agonist activity at mouse delta opioid receptor expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 500nMAssay Description:Activity against delta opioid receptor by stimulation of [35S]GTPgammaS binding in CHO-hgamma cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 730nMAssay Description:Activity against delta opioid receptor by stimulation of [35S]GTPgammaS binding in CHO-hgamma cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 830nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
Affinity DataEC50: >1.50E+3nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
Affinity DataEC50: >1.50E+3nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
Affinity DataEC50: >1.50E+3nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
Affinity DataEC50: 2.20E+3nMAssay Description:In vitro bioassay data to determine the effective concentration required for antagonistic activity against Opioid receptor delta 1 in functional assa...More data for this Ligand-Target Pair
Affinity DataEC50: 7.94E+3nMAssay Description:Antagonist activity at DOR in CD1 mouse vas deferens assessed as pEC50 for DPDPE-induced inhibition of EFS-evoked contractions at 1 uM incubated for ...More data for this Ligand-Target Pair
Affinity DataEC50: 1.26E+5nMAssay Description:Antagonist activity at DOR in CD1 mouse vas deferens assessed as pEC50 for DPDPE-induced inhibition of EFS-evoked contractions at 1 uM incubated for ...More data for this Ligand-Target Pair
Affinity DataEC50: 1.58E+5nMAssay Description:Agonist activity at DOR in CD1 mouse vas deferens assessed as inhibition of EFS-induced contractions incubated for 60 minsMore data for this Ligand-Target Pair