Compile Data Set for Download or QSAR
maximum 50k data
Found 468 of ec50 data for polymerid = 49000892,49000894,49000895
TargetOxytocin receptor(Homo sapiens (Human))
Institute Of Neuroscience

Curated by ChEMBL
LigandPNGBDBM50536275(CHEMBL4520203)
Affinity DataEC50:  0.00100nMAssay Description:Agonist activity at human oxytocin receptor C47A mutant high affinity site expressed in HEK293 cells coexpressing Rluc8-tagged Galphaq, N-terminal GF...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Institute Of Neuroscience

Curated by ChEMBL
LigandPNGBDBM50536278(CHEMBL4520170)
Affinity DataEC50:  0.00100nMAssay Description:Agonist activity at human oxytocin receptor high affinity site expressed in HEK293 cells coexpressing Rluc8-tagged Galphaq, N-terminal GFP-tagged Gga...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Institute Of Neuroscience

Curated by ChEMBL
LigandPNGBDBM50536279(CHEMBL4567752)
Affinity DataEC50:  0.00100nMAssay Description:Agonist activity at human oxytocin receptor C47A mutant high affinity site expressed in HEK293 cells coexpressing Rluc8-tagged Galphaq, N-terminal GF...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Institute Of Neuroscience

Curated by ChEMBL
LigandPNGBDBM50536277(CHEMBL4541104)
Affinity DataEC50:  0.00300nMAssay Description:Agonist activity at human oxytocin receptor high affinity site expressed in HEK293 cells coexpressing Rluc8-tagged Galphaq, N-terminal GFP-tagged Gga...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Institute Of Neuroscience

Curated by ChEMBL
LigandPNGBDBM50536277(CHEMBL4541104)
Affinity DataEC50:  0.00300nMAssay Description:Agonist activity at human oxytocin receptor high affinity site expressed in HEK293 cells coexpressing Rluc8-tagged Galphaq, N-terminal GFP-tagged Gga...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Institute Of Neuroscience

Curated by ChEMBL
LigandPNGBDBM50205990(CHEMBL395429 | OXYTOCIN)
Affinity DataEC50:  0.00460nMAssay Description:Agonist activity at human OTR receptor expressed in HEK293 cells assessed as intracellular calcium level measured at 3 secs interval for 5 mins by fu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Institute Of Neuroscience

Curated by ChEMBL
LigandPNGBDBM50240674(CHEMBL4097965)
Affinity DataEC50:  0.00500nMAssay Description:Agonist activity at human OTR expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Institute Of Neuroscience

Curated by ChEMBL
LigandPNGBDBM50240613(CHEMBL4074974)
Affinity DataEC50:  0.00500nMAssay Description:Agonist activity at human OTR expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Institute Of Neuroscience

Curated by ChEMBL
LigandPNGBDBM50240638(CHEMBL4066368)
Affinity DataEC50:  0.00700nMAssay Description:Agonist activity at human OTR expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Institute Of Neuroscience

Curated by ChEMBL
LigandPNGBDBM50044752(CHEMBL3353956)
Affinity DataEC50:  0.00700nMAssay Description:Agonist activity at human OTR expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Institute Of Neuroscience

Curated by ChEMBL
LigandPNGBDBM50240632(CHEMBL4070222)
Affinity DataEC50:  0.00700nMAssay Description:Agonist activity at human OTR expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Institute Of Neuroscience

Curated by ChEMBL
LigandPNGBDBM50240633(CHEMBL4093631)
Affinity DataEC50:  0.00700nMAssay Description:Agonist activity at human OTR expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Institute Of Neuroscience

Curated by ChEMBL
LigandPNGBDBM50240651(CHEMBL3276119)
Affinity DataEC50:  0.00700nMAssay Description:Agonist activity at human OTR expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Institute Of Neuroscience

Curated by ChEMBL
LigandPNGBDBM50240610(CHEMBL4101658)
Affinity DataEC50:  0.00700nMAssay Description:Agonist activity at human OTR expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Institute Of Neuroscience

Curated by ChEMBL
LigandPNGBDBM50240636(CHEMBL4104080)
Affinity DataEC50:  0.00800nMAssay Description:Agonist activity at human OTR expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Institute Of Neuroscience

Curated by ChEMBL
LigandPNGBDBM50205990(CHEMBL395429 | OXYTOCIN)
Affinity DataEC50:  0.00800nMAssay Description:Agonist activity at human OTR expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Institute Of Neuroscience

Curated by ChEMBL
LigandPNGBDBM50044676(CHEMBL439044)
Affinity DataEC50:  0.00900nMAssay Description:Agonist activity at human OTR expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Institute Of Neuroscience

Curated by ChEMBL
LigandPNGBDBM50240634(CHEMBL4074335)
Affinity DataEC50:  0.00900nMAssay Description:Agonist activity at human OTR expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Institute Of Neuroscience

Curated by ChEMBL
LigandPNGBDBM50044677(CHEBI:59204 | Carbetocin)
Affinity DataEC50:  0.0100nMAssay Description:Agonist activity at recombinant human OTR expressed in HEK293 cells assessed as increase in intracellular calcium level measured at 3 secs interval f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetOxytocin receptor(Homo sapiens (Human))
Institute Of Neuroscience

Curated by ChEMBL
LigandPNGBDBM50044773(CHEMBL3353932)
Affinity DataEC50:  0.0100nMAssay Description:Agonist activity at human oxytocin receptor expressed in CHO-K1 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Institute Of Neuroscience

Curated by ChEMBL
LigandPNGBDBM50044771(CHEMBL3353939)
Affinity DataEC50:  0.0100nMAssay Description:Agonist activity at human oxytocin receptor expressed in CHO-K1 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Institute Of Neuroscience

Curated by ChEMBL
LigandPNGBDBM50044770(CHEMBL3353940)
Affinity DataEC50:  0.0100nMAssay Description:Agonist activity at human oxytocin receptor expressed in CHO-K1 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Institute Of Neuroscience

Curated by ChEMBL
LigandPNGBDBM50044763(CHEMBL3353946)
Affinity DataEC50:  0.0100nMAssay Description:Agonist activity at human oxytocin receptor expressed in CHO-K1 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Institute Of Neuroscience

Curated by ChEMBL
LigandPNGBDBM50044761(CHEMBL3353948)
Affinity DataEC50:  0.0100nMAssay Description:Agonist activity at human oxytocin receptor expressed in CHO-K1 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Institute Of Neuroscience

Curated by ChEMBL
LigandPNGBDBM50044752(CHEMBL3353956)
Affinity DataEC50:  0.0100nMAssay Description:Agonist activity at human oxytocin receptor expressed in CHO-K1 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Institute Of Neuroscience

Curated by ChEMBL
LigandPNGBDBM50240630(CHEMBL4102192)
Affinity DataEC50:  0.0100nMAssay Description:Agonist activity at human OTR expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Institute Of Neuroscience

Curated by ChEMBL
LigandPNGBDBM50044775(CHEMBL3353930)
Affinity DataEC50:  0.0100nMAssay Description:Agonist activity at human oxytocin receptor expressed in CHO-K1 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Institute Of Neuroscience

Curated by ChEMBL
LigandPNGBDBM50205990(CHEMBL395429 | OXYTOCIN)
Affinity DataEC50:  0.0100nMAssay Description:Agonist activity at recombinant human OTR expressed in HEK293 cells assessed as increase in intracellular calcium level measured at 3 secs interval f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Institute Of Neuroscience

Curated by ChEMBL
LigandPNGBDBM50044742(CHEMBL3354579)
Affinity DataEC50:  0.0100nMAssay Description:Agonist activity at human oxytocin receptor expressed in CHO-K1 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Institute Of Neuroscience

Curated by ChEMBL
LigandPNGBDBM50536279(CHEMBL4567752)
Affinity DataEC50:  0.0110nMAssay Description:Agonist activity at human oxytocin receptor V43A/C47A double mutant high affinity site expressed in HEK293 cells coexpressing Rluc8-tagged Galphaq, N...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Institute Of Neuroscience

Curated by ChEMBL
LigandPNGBDBM50536278(CHEMBL4520170)
Affinity DataEC50:  0.0120nMAssay Description:Agonist activity at human oxytocin receptor high affinity site expressed in HEK293 cells coexpressing Rluc8-tagged Galphaq, N-terminal GFP-tagged Gga...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Institute Of Neuroscience

Curated by ChEMBL
LigandPNGBDBM50240672(CHEMBL4095930)
Affinity DataEC50:  0.0130nMAssay Description:Agonist activity at human OTR expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Institute Of Neuroscience

Curated by ChEMBL
LigandPNGBDBM50240644(CHEMBL3277916)
Affinity DataEC50:  0.0130nMAssay Description:Agonist activity at human OTR expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Institute Of Neuroscience

Curated by ChEMBL
LigandPNGBDBM50240607(CHEMBL4093931)
Affinity DataEC50:  0.0130nMAssay Description:Agonist activity at human OTR expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Institute Of Neuroscience

Curated by ChEMBL
LigandPNGBDBM50240629(CHEMBL4084223)
Affinity DataEC50:  0.0140nMAssay Description:Agonist activity at human OTR expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Institute Of Neuroscience

Curated by ChEMBL
LigandPNGBDBM50240663(CHEMBL4078856)
Affinity DataEC50:  0.0150nMAssay Description:Agonist activity at human OTR expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Institute Of Neuroscience

Curated by ChEMBL
LigandPNGBDBM50044754(CHEMBL3353955)
Affinity DataEC50:  0.0200nMAssay Description:Agonist activity at human oxytocin receptor expressed in CHO-K1 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Institute Of Neuroscience

Curated by ChEMBL
LigandPNGBDBM50044727(CHEMBL3354592)
Affinity DataEC50:  0.0200nMAssay Description:Agonist activity at human oxytocin receptor expressed in CHO-K1 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Institute Of Neuroscience

Curated by ChEMBL
LigandPNGBDBM50044750(CHEMBL3354571)
Affinity DataEC50:  0.0200nMAssay Description:Agonist activity at human oxytocin receptor expressed in CHO-K1 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Institute Of Neuroscience

Curated by ChEMBL
LigandPNGBDBM50240673(CHEMBL4096848)
Affinity DataEC50:  0.0210nMAssay Description:Agonist activity at human OTR expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Institute Of Neuroscience

Curated by ChEMBL
LigandPNGBDBM50044686(CHEMBL3354594)
Affinity DataEC50:  0.0250nMAssay Description:Agonist activity at recombinant human OTR expressed in HEK293 cells assessed as increase in intracellular calcium level measured at 3 secs interval f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Institute Of Neuroscience

Curated by ChEMBL
LigandPNGBDBM50240675(CHEMBL4101771)
Affinity DataEC50:  0.0270nMAssay Description:Agonist activity at human OTR expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Institute Of Neuroscience

Curated by ChEMBL
LigandPNGBDBM50240631(CHEMBL4065273)
Affinity DataEC50:  0.0270nMAssay Description:Agonist activity at human OTR expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Institute Of Neuroscience

Curated by ChEMBL
LigandPNGBDBM50523555(CHEMBL4474284)
Affinity DataEC50:  0.0280nMAssay Description:Agonist activity at recombinant human OTR expressed in HEK293 cells assessed as increase in intracellular calcium level measured at 3 secs interval f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Institute Of Neuroscience

Curated by ChEMBL
LigandPNGBDBM50240628(CHEMBL4094454)
Affinity DataEC50:  0.0300nMAssay Description:Agonist activity at human OTR expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Institute Of Neuroscience

Curated by ChEMBL
LigandPNGBDBM50044768(CHEMBL3353942)
Affinity DataEC50:  0.0300nMAssay Description:Agonist activity at human oxytocin receptor expressed in CHO-K1 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Institute Of Neuroscience

Curated by ChEMBL
LigandPNGBDBM50523557(CHEMBL4583231)
Affinity DataEC50:  0.0310nMAssay Description:Agonist activity at recombinant human OTR expressed in HEK293 cells assessed as increase in intracellular calcium level measured at 3 secs interval f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Institute Of Neuroscience

Curated by ChEMBL
LigandPNGBDBM50240604(CHEMBL4092971)
Affinity DataEC50:  0.0310nMAssay Description:Agonist activity at human OTR expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Institute Of Neuroscience

Curated by ChEMBL
LigandPNGBDBM50044683(CHEMBL3354597)
Affinity DataEC50:  0.0400nMAssay Description:Agonist activity at human oxytocin receptor expressed in CHO-K1 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Institute Of Neuroscience

Curated by ChEMBL
LigandPNGBDBM50044676(CHEMBL439044)
Affinity DataEC50:  0.0400nMAssay Description:Agonist activity at human OTR expressed in CHO cells assessed as increase in calcium flux after 60 to 120 mins by fluo-4 dye based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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