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Compile Data Set for Download or QSAR

Found 4 hits of ec50 data for polymerid = 50002102,50005707,6236   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
C-C chemokine receptor type 3


(Homo sapiens (Human))
BDBM50100021
PNG
((S)-2-[(Naphthalene-1-carbonyl)-amino]-3-(4-nitro-...)
Show SMILES COC(=O)[C@H](Cc1ccc(cc1)[N+]([O-])=O)NC(=O)c1cccc2ccccc12
Show InChI InChI=1S/C21H18N2O5/c1-28-21(25)19(13-14-9-11-16(12-10-14)23(26)27)22-20(24)18-8-4-6-15-5-2-3-7-17(15)18/h2-12,19H,13H2,1H3,(H,22,24)/t19-/m0/s1
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PC sid
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Article
PubMed
n/an/an/an/a 780n/an/an/an/a



Kindai University

Curated by ChEMBL


Assay Description
Antagonist activity at human EGFP-fused CCR3 expressed in mouse L1.2 cells assessed as inhibition of CCL11-induced chemotaxis measured after 1.5 hrs ...


J Nat Prod 79: 2005-13 (2016)


Article DOI: 10.1021/acs.jnatprod.6b00262
BindingDB Entry DOI: 10.7270/Q2MW2K39
More data for this
Ligand-Target Pair
C-C chemokine receptor type 3


(Homo sapiens (Human))
BDBM50202470
PNG
(CHEMBL3922119)
Show SMILES COc1ccc(cc1OC)[C@@H](OC(C)=O)[C@H](C)Oc1c(OC)cc(CC=C)cc1OC
Show InChI InChI=1S/C24H30O7/c1-8-9-17-12-21(28-6)24(22(13-17)29-7)30-15(2)23(31-16(3)25)18-10-11-19(26-4)20(14-18)27-5/h8,10-15,23H,1,9H2,2-7H3/t15-,23-/m0/s1
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PubMed
n/an/an/an/a 1.40E+3n/an/an/an/a



Kindai University

Curated by ChEMBL


Assay Description
Antagonist activity at human EGFP-fused CCR3 expressed in mouse L1.2 cells assessed as inhibition of CCL11-induced chemotaxis measured after 1.5 hrs ...


J Nat Prod 79: 2005-13 (2016)


Article DOI: 10.1021/acs.jnatprod.6b00262
BindingDB Entry DOI: 10.7270/Q2MW2K39
More data for this
Ligand-Target Pair
C-C chemokine receptor type 3


(Homo sapiens (Human))
BDBM50202471
PNG
(CHEMBL3949874)
Show SMILES COc1cc(cc(OC)c1O)[C@H](O)[C@@H](C)Oc1c(OC)cc(CC=C)cc1OC
Show InChI InChI=1S/C22H28O7/c1-7-8-14-9-18(27-5)22(19(10-14)28-6)29-13(2)20(23)15-11-16(25-3)21(24)17(12-15)26-4/h7,9-13,20,23-24H,1,8H2,2-6H3/t13-,20-/m1/s1
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PubMed
n/an/an/an/a 1.50E+3n/an/an/an/a



Kindai University

Curated by ChEMBL


Assay Description
Antagonist activity at human EGFP-fused CCR3 expressed in mouse L1.2 cells assessed as inhibition of CCL11-induced chemotaxis measured after 1.5 hrs ...


J Nat Prod 79: 2005-13 (2016)


Article DOI: 10.1021/acs.jnatprod.6b00262
BindingDB Entry DOI: 10.7270/Q2MW2K39
More data for this
Ligand-Target Pair
C-C chemokine receptor type 3


(Homo sapiens (Human))
BDBM50202469
PNG
(CHEMBL3906647)
Show SMILES COc1cc(\C=C\C)cc2[C@@H](C)[C@@H](Oc12)c1cc(OC)c(O)c(OC)c1
Show InChI InChI=1S/C21H24O5/c1-6-7-13-8-15-12(2)20(26-21(15)18(9-13)25-5)14-10-16(23-3)19(22)17(11-14)24-4/h6-12,20,22H,1-5H3/b7-6+/t12-,20-/m1/s1
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Article
PubMed
n/an/an/an/a 1.60E+3n/an/an/an/a



Kindai University

Curated by ChEMBL


Assay Description
Antagonist activity at human EGFP-fused CCR3 expressed in mouse L1.2 cells assessed as inhibition of CCL11-induced chemotaxis measured after 1.5 hrs ...


J Nat Prod 79: 2005-13 (2016)


Article DOI: 10.1021/acs.jnatprod.6b00262
BindingDB Entry DOI: 10.7270/Q2MW2K39
More data for this
Ligand-Target Pair