TargetATP-dependent Clp protease proteolytic subunit(Escherichia coli (strain K12))
University Of Oklahoma Cobre In Structural Biology
Curated by ChEMBL
University Of Oklahoma Cobre In Structural Biology
Curated by ChEMBL
Affinity DataEC50: 100nMAssay Description:Activation of Escherichia coli BLR (DE3) ClpP using Abz-DFAPKMALVPYNO2 as substrate assessed as degradation of substrate peptide preincubated for 15 ...More data for this Ligand-Target Pair
TargetATP-dependent Clp protease proteolytic subunit(Escherichia coli (strain K12))
University Of Oklahoma Cobre In Structural Biology
Curated by ChEMBL
University Of Oklahoma Cobre In Structural Biology
Curated by ChEMBL
Affinity DataEC50: 1.20E+3nMAssay Description:Activation of Escherichia coli BLR (DE3) ClpP using FITC-beta casein as substrate assessed as degradation of substrate peptide preincubated for 15 mi...More data for this Ligand-Target Pair
TargetATP-dependent Clp protease proteolytic subunit(Staphylococcus aureus (strain NCTC 8325))
Sichuan University
Curated by ChEMBL
Sichuan University
Curated by ChEMBL
Affinity DataEC50: 1.27E+3nMAssay Description:Binding affinity to N-terminal His6-sumo-tagged full length Staphylococcus aureus ClpP expressed in Escherichia coli BL2 (DE3) assessed as shifting o...More data for this Ligand-Target Pair
TargetATP-dependent Clp protease proteolytic subunit(Staphylococcus aureus (strain NCTC 8325))
Sichuan University
Curated by ChEMBL
Sichuan University
Curated by ChEMBL
Affinity DataEC50: 1.40E+3nMAssay Description:Inhibition of ClpP in methicillin-resistant Staphylococcus aureus ATCC 33591 assessed as reduction in bacteria-induced hemolysis of sheep erythrocyte...More data for this Ligand-Target Pair
TargetATP-dependent Clp protease proteolytic subunit(Staphylococcus aureus (strain NCTC 8325))
Sichuan University
Curated by ChEMBL
Sichuan University
Curated by ChEMBL
Affinity DataEC50: 2.60E+3nMAssay Description:Inhibition of ClpP in methicillin-resistant Staphylococcus aureus ATCC 33591 assessed as reduction in bacteria-induced hemolysis of sheep erythrocyte...More data for this Ligand-Target Pair
TargetATP-dependent Clp protease proteolytic subunit(Staphylococcus aureus (strain NCTC 8325))
Sichuan University
Curated by ChEMBL
Sichuan University
Curated by ChEMBL
Affinity DataEC50: 3.30E+3nMAssay Description:Inhibition of ClpP in methicillin-resistant Staphylococcus aureus ATCC 33591 assessed as reduction in bacteria-induced hemolysis of sheep erythrocyte...More data for this Ligand-Target Pair
TargetATP-dependent Clp protease proteolytic subunit(Staphylococcus aureus (strain NCTC 8325))
Sichuan University
Curated by ChEMBL
Sichuan University
Curated by ChEMBL
Affinity DataEC50: 3.40E+3nMAssay Description:Inhibition of recombinant Staphylococcus aureus NCTC 8325 peptidase activity of clpP expressed in Escherichia coli BL21 after 10 mins using SLY-AMC a...More data for this Ligand-Target Pair
TargetATP-dependent Clp protease proteolytic subunit(Staphylococcus aureus (strain NCTC 8325))
Sichuan University
Curated by ChEMBL
Sichuan University
Curated by ChEMBL
Affinity DataEC50: 3.60E+3nMAssay Description:Inhibition of ClpP in methicillin-resistant Staphylococcus aureus ATCC 33591 assessed as reduction in bacteria-induced hemolysis of sheep erythrocyte...More data for this Ligand-Target Pair
TargetATP-dependent Clp protease proteolytic subunit(Staphylococcus aureus (strain NCTC 8325))
Sichuan University
Curated by ChEMBL
Sichuan University
Curated by ChEMBL
Affinity DataEC50: 4.50E+3nMAssay Description:Inhibition of recombinant Staphylococcus aureus NCTC 8325 peptidase activity of clpP expressed in Escherichia coli BL21 after 10 mins using SLY-AMC a...More data for this Ligand-Target Pair
TargetATP-dependent Clp protease proteolytic subunit(Staphylococcus aureus (strain NCTC 8325))
Sichuan University
Curated by ChEMBL
Sichuan University
Curated by ChEMBL
Affinity DataEC50: 5.40E+3nMAssay Description:Inhibition of recombinant Staphylococcus aureus NCTC 8325 peptidase activity of clpP expressed in Escherichia coli BL21 after 10 mins using SLY-AMC a...More data for this Ligand-Target Pair
TargetATP-dependent Clp protease proteolytic subunit(Staphylococcus aureus (strain NCTC 8325))
Sichuan University
Curated by ChEMBL
Sichuan University
Curated by ChEMBL
Affinity DataEC50: 9.60E+3nMAssay Description:Inhibition of ClpP in methicillin-resistant Staphylococcus aureus ATCC 33591 assessed as reduction in bacteria-induced hemolysis of sheep erythrocyte...More data for this Ligand-Target Pair
TargetATP-dependent Clp protease proteolytic subunit(Staphylococcus aureus (strain NCTC 8325))
Sichuan University
Curated by ChEMBL
Sichuan University
Curated by ChEMBL
Affinity DataEC50: 1.48E+4nMAssay Description:Inhibition of ClpP in methicillin-resistant Staphylococcus aureus ATCC 33591 assessed as reduction in bacteria-induced hemolysis of sheep erythrocyte...More data for this Ligand-Target Pair
TargetATP-dependent Clp protease proteolytic subunit(Staphylococcus aureus (strain NCTC 8325))
Sichuan University
Curated by ChEMBL
Sichuan University
Curated by ChEMBL
Affinity DataEC50: 1.99E+4nMAssay Description:Binding affinity to N-terminal His6-sumo-tagged full length Staphylococcus aureus ClpP expressed in Escherichia coli BL2 (DE3) assessed as shifting o...More data for this Ligand-Target Pair
TargetATP-dependent Clp protease proteolytic subunit(Escherichia coli (strain K12))
University Of Oklahoma Cobre In Structural Biology
Curated by ChEMBL
University Of Oklahoma Cobre In Structural Biology
Curated by ChEMBL
Affinity DataEC50: 2.22E+4nMAssay Description:Activation of Escherichia coli BLR (DE3) ClpP using FITC-beta casein as substrate assessed as degradation of substrate peptide preincubated for 15 mi...More data for this Ligand-Target Pair
TargetATP-dependent Clp protease proteolytic subunit(Staphylococcus aureus (strain NCTC 8325))
Sichuan University
Curated by ChEMBL
Sichuan University
Curated by ChEMBL
Affinity DataEC50: 2.35E+4nMAssay Description:Inhibition of ClpP in methicillin-resistant Staphylococcus aureus ATCC 33591 assessed as reduction in bacteria-induced hemolysis of sheep erythrocyte...More data for this Ligand-Target Pair
TargetATP-dependent Clp protease proteolytic subunit(Escherichia coli (strain K12))
University Of Oklahoma Cobre In Structural Biology
Curated by ChEMBL
University Of Oklahoma Cobre In Structural Biology
Curated by ChEMBL
Affinity DataEC50: 2.54E+4nMAssay Description:Activation of Escherichia coli BLR (DE3) ClpP using Abz-DFAPKMALVPYNO2 as substrate assessed as degradation of substrate peptide preincubated for 15 ...More data for this Ligand-Target Pair
TargetATP-dependent Clp protease proteolytic subunit(Escherichia coli (strain K12))
University Of Oklahoma Cobre In Structural Biology
Curated by ChEMBL
University Of Oklahoma Cobre In Structural Biology
Curated by ChEMBL
Affinity DataEC50: 3.96E+4nMAssay Description:Activation of Escherichia coli BLR (DE3) ClpP using Abz-DFAPKMALVPYNO2 as substrate assessed as degradation of substrate peptide preincubated for 15 ...More data for this Ligand-Target Pair
TargetATP-dependent Clp protease proteolytic subunit(Escherichia coli (strain K12))
University Of Oklahoma Cobre In Structural Biology
Curated by ChEMBL
University Of Oklahoma Cobre In Structural Biology
Curated by ChEMBL
Affinity DataEC50: 8.75E+4nMAssay Description:Activation of Escherichia coli BLR (DE3) ClpP using FITC-beta casein as substrate assessed as degradation of substrate peptide preincubated for 15 mi...More data for this Ligand-Target Pair