Affinity DataEC50: 0.00540nMAssay Description:Agonist activity at NK3R (unknown origin) transfected in CHO cells assessed as calcium influx at 10 mMMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0120nMAssay Description:Agonist activity at NK3R (unknown origin) transfected in CHO cells assessed as calcium influx at 10 mMMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0130nMAssay Description:Agonist activity at NK3R (unknown origin) transfected in CHO cells assessed as calcium influx at 10 mMMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0170nMAssay Description:Agonist activity at NK3R (unknown origin) transfected in CHO cells assessed as calcium influx at 10 mMMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0240nMAssay Description:Agonist activity at NK3R (unknown origin) transfected in CHO cells assessed as calcium influx at 10 mMMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0260nMAssay Description:Agonist activity at NK3R (unknown origin) transfected in CHO cells assessed as calcium influx at 10 mMMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0320nMAssay Description:Agonist activity at NK3R (unknown origin) transfected in CHO cells assessed as calcium influx at 10 mMMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0360nMAssay Description:Agonist activity at NK3R (unknown origin) transfected in CHO cells assessed as calcium influx at 10 mMMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0360nMAssay Description:Agonist activity at NK3R (unknown origin) transfected in CHO cells assessed as calcium influx at 10 mMMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0380nMAssay Description:Agonist activity at NK3R (unknown origin) transfected in CHO cells assessed as calcium influx at 10 mMMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0400nMAssay Description:Agonist activity at NK3R (unknown origin) transfected in CHO cells assessed as calcium influx at 10 mMMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0400nMAssay Description:Agonist activity at NK3R (unknown origin) transfected in CHO cells assessed as calcium influx at 10 mMMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0410nMAssay Description:Agonist activity at NK3R (unknown origin) transfected in CHO cells assessed as calcium influx at 10 mMMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0430nMAssay Description:Agonist activity at NK3R (unknown origin) transfected in CHO cells assessed as calcium influx at 10 mMMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0460nMAssay Description:Agonist activity at NK3R (unknown origin) transfected in CHO cells assessed as calcium influx at 10 mMMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0510nMAssay Description:Agonist activity at NK3R (unknown origin) transfected in CHO cells assessed as calcium influx at 10 mMMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0600nMAssay Description:Agonist activity at NK3R (unknown origin) transfected in CHO cells assessed as calcium influx at 10 mMMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0650nMAssay Description:Agonist activity at NK3R (unknown origin) transfected in CHO cells assessed as calcium influx at 10 mMMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0710nMAssay Description:Agonist activity at NK3R (unknown origin) transfected in CHO cells assessed as calcium influx at 10 mMMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0720nMAssay Description:Agonist activity at NK3R (unknown origin) transfected in CHO cells assessed as calcium influx at 10 mMMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0780nMAssay Description:Agonist activity at NK3R (unknown origin) transfected in CHO cells assessed as calcium influx at 10 mMMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0790nMAssay Description:Agonist activity at NK3R (unknown origin) transfected in CHO cells assessed as calcium influx at 10 mMMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0800nMAssay Description:Agonist activity at NK3R (unknown origin) transfected in CHO cells assessed as calcium influx at 10 mMMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0830nMAssay Description:Agonist activity at NK3R (unknown origin) transfected in CHO cells assessed as calcium influx at 10 mMMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0850nMAssay Description:Agonist activity at NK3R (unknown origin) transfected in CHO cells assessed as calcium influx at 10 mMMore data for this Ligand-Target Pair
Affinity DataEC50: 0.110nMAssay Description:Agonist activity at NK3R (unknown origin) transfected in CHO cells assessed as calcium influx at 10 mMMore data for this Ligand-Target Pair
Affinity DataEC50: 0.120nMAssay Description:Agonist activity at NK3R (unknown origin) transfected in CHO cells assessed as calcium influx at 10 mMMore data for this Ligand-Target Pair
Affinity DataEC50: 0.130nMAssay Description:Agonist activity at NK3R (unknown origin) transfected in CHO cells assessed as calcium influx at 10 mMMore data for this Ligand-Target Pair
Affinity DataEC50: 0.150nMAssay Description:Agonist activity at NK3R (unknown origin) transfected in CHO cells assessed as calcium influx at 10 mMMore data for this Ligand-Target Pair
Affinity DataEC50: 0.210nMAssay Description:Agonist activity at NK3R (unknown origin) transfected in CHO cells assessed as calcium influx at 10 mMMore data for this Ligand-Target Pair
Affinity DataEC50: 0.220nMAssay Description:Agonist activity at NK3R (unknown origin) transfected in CHO cells assessed as calcium influx at 10 mMMore data for this Ligand-Target Pair
Affinity DataEC50: 0.280nMAssay Description:Agonist activity at NK3R (unknown origin) transfected in CHO cells assessed as calcium influx at 10 mMMore data for this Ligand-Target Pair
Affinity DataEC50: 0.470nMAssay Description:Agonist activity at NK3R (unknown origin) transfected in CHO cells assessed as calcium influx at 10 mMMore data for this Ligand-Target Pair
Affinity DataEC50: 0.600nMAssay Description:Agonist activity at human NK3 receptor expressed in cells assessed as accumulation of [3H]inositol phosphateMore data for this Ligand-Target Pair
Affinity DataEC50: 0.710nMAssay Description:Agonist activity at wild type human NK3 receptor expressed in HEK293 cells assessed as [3H]IP accumulation after 45 minsMore data for this Ligand-Target Pair
Affinity DataEC50: 1.40nMAssay Description:Agonist activity at NK3R (unknown origin) transfected in CHO cells assessed as calcium influx at 10 mMMore data for this Ligand-Target Pair
Affinity DataEC50: 1.70nMAssay Description:Antagonist activity at human NK3 receptor expressed in CHO cells assessed as inhibition of senktide-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.80nMAssay Description:Antagonist activity at human NK3 receptor expressed in CHO cells assessed as inhibition of senktide-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.80nMAssay Description:Antagonist activity at human NK3 receptor expressed in CHO cells assessed as inhibition of senktide-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2.5nMAssay Description:Antagonist activity at human NK3 receptor expressed in CHO cells assessed as inhibition of senktide-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 3nMAssay Description:Activity at human NK3 receptor expressed in CHO cells assessed as increase in inositol phosphate generationMore data for this Ligand-Target Pair
Affinity DataEC50: 3.30nMAssay Description:Antagonist activity at human NK3 receptor expressed in CHO cells assessed as inhibition of senktide-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 3.40nMAssay Description:Agonist activity at NK3R (unknown origin) transfected in CHO cells assessed as calcium influx at 10 mMMore data for this Ligand-Target Pair
Affinity DataEC50: 3.60nMAssay Description:Antagonist activity at human NK3 receptor expressed in CHO cells assessed as inhibition of senktide-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 3.70nMAssay Description:Antagonist activity at human NK3 receptor expressed in CHO cells assessed as inhibition of senktide-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 4.90nMAssay Description:Antagonist activity at human NK3 receptor expressed in CHO cells assessed as inhibition of senktide-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 4.90nMAssay Description:Antagonist activity at human NK3 receptor expressed in CHO cells assessed as inhibition of senktide-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 5nMAssay Description:Agonist activity at NK3R (unknown origin) transfected in CHO cells assessed as calcium influx at 10 mMMore data for this Ligand-Target Pair
Affinity DataEC50: 5.10nMAssay Description:Antagonist activity at human NK3 receptor expressed in CHO cells assessed as inhibition of senktide-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 5.30nMAssay Description:Antagonist activity at human NK3 receptor expressed in CHO cells assessed as inhibition of senktide-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair