Compile Data Set for Download or QSAR
maximum 50k data
Found 367 of ic50 data for polymerid = 5286
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50112200(CHEMBL300056 | N-(2-(2-iodo-5-methoxy-1-methyl-1H-...)
Affinity DataIC50:  0.0891nMAssay Description:Displacement of [125I]iodomelatonin from MT3/QR2 melatonin binding site expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50112208(CHEMBL300728 | N-(2-(2-iodo-5-methoxy-1-methyl-4-n...)
Affinity DataIC50:  0.129nMAssay Description:Displacement of [125I]iodomelatonin from MT3/QR2 melatonin binding site expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50112203(CHEMBL52559 | N-(2-(2-iodo-5-methoxy-4-nitro-1H-in...)
Affinity DataIC50:  0.200nMAssay Description:Displacement of [125I]iodomelatonin from MT3/QR2 melatonin binding site expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50413646(CHEMBL511675)
Affinity DataIC50:  0.302nMAssay Description:Displacement of [125I]iodomelatonin from MT3/QR2 melatonin binding site expressed in CHO cellsMore data for this Ligand-Target Pair
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50112201(CHEMBL53622 | N-(2-(5-methoxy-1-methyl-4-nitro-1H-...)
Affinity DataIC50:  0.309nMAssay Description:Displacement of [125I]iodomelatonin from MT3/QR2 melatonin binding site expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50342769(CHEMBL1770214 | N-[2-(7-methoxycarbonylamino-napht...)
Affinity DataIC50:  0.390nMAssay Description:Binding affinity to human MT3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50112206(CHEMBL300195 | N-(2-(5-methoxy-4-nitro-1H-indol-3-...)
Affinity DataIC50:  1.20nMAssay Description:Displacement of [125I]iodomelatonin from MT3/QR2 melatonin binding site expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50260394(5-MCA-NAT | 5-methoxycarbonylamino-N-acetyltryptam...)
Affinity DataIC50:  2.70nMAssay Description:Binding affinity to low affinity melatonin (MT3) site of quinone reductase 2More data for this Ligand-Target Pair
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50066960(CHEMBL33700 | N-(2-(5-methoxy-1-methyl-1H-indol-3-...)
Affinity DataIC50:  2.82nMAssay Description:Displacement of [125I]iodomelatonin from MT3/QR2 melatonin binding site expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50413645(CHEMBL457126)
Affinity DataIC50:  3.02nMAssay Description:Displacement of [125I]iodomelatonin from MT3/QR2 melatonin binding site expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50363378(CHEMBL1945729)
Affinity DataIC50:  4.10nMAssay Description:Inhibition of human quinone reductase 2 using NMeH as substrate by MTT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50342774(CHEMBL1738752 | N-[2-(7-methylsulfamoyl-naphth-1-y...)
Affinity DataIC50:  4.90nMAssay Description:Binding affinity to human MT3 receptorMore data for this Ligand-Target Pair
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50317140(5-(2-(diethylamino)ethylamino)-7-hydroxy-8,9-dimet...)
Affinity DataIC50:  6nMAssay Description:Inhibition of human recombinant NQO2 assessed as reduction of DCPIP by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50413650(CHEMBL465378)
Affinity DataIC50:  7.76nMAssay Description:Displacement of [125I]iodomelatonin from MT3/QR2 melatonin binding site expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM29568(CHEMBL2 | PRAZOSIN | PRAZOSIN HYDROCHLORIDE | [3H]...)
Affinity DataIC50:  7.80nMAssay Description:Binding affinity to human low affinity melatonin (MT3) site of quinone reductase 2More data for this Ligand-Target Pair
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50008356(5-(2-(diethylamino)ethylamino)-8-methoxy-1-methyl-...)
Affinity DataIC50:  9nMAssay Description:Inhibition of human recombinant NQO2 assessed as reduction of DCPIP by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50342775(CHEMBL457992 | N-(2-(7-(N-methylsulfamoyl)naphthal...)
Affinity DataIC50:  9.10nMAssay Description:Binding affinity to human MT3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50342775(CHEMBL457992 | N-(2-(7-(N-methylsulfamoyl)naphthal...)
Affinity DataIC50:  9.12nMAssay Description:Displacement of [125I]iodomelatonin from MT3/QR2 melatonin binding site expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50515994(CHEMBL4514167)
Affinity DataIC50:  10nMAssay Description:Inhibition of recombinant human NQO2 expressed in Escherichia coli using DCPIP as substrate by spectrophotometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50260410(CHEMBL493424 | N-(2-(5-Methoxycarbonylamino-benzo[...)
Affinity DataIC50:  11.0nMAssay Description:Displacement of [125I]iodomelatonin from MT3/QR2 melatonin binding site expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50413654(CHEMBL457541)
Affinity DataIC50:  11.0nMAssay Description:Displacement of [125I]iodomelatonin from MT3/QR2 melatonin binding site expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50413640(CHEMBL455339)
Affinity DataIC50:  12.0nMAssay Description:Displacement of [125I]iodomelatonin from MT3/QR2 melatonin binding site expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50515978(CHEMBL1967497)
Affinity DataIC50:  13nMAssay Description:Inhibition of recombinant human NQO2 expressed in Escherichia coli using DCPIP as substrate by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50354527(CHEMBL1836819)
Affinity DataIC50:  14nMAssay Description:Inhibition of human recombinant NQO2 assessed as reduction of DCPIP by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50413643(CHEMBL495399)
Affinity DataIC50:  14.1nMAssay Description:Displacement of [125I]iodomelatonin from MT3/QR2 melatonin binding site expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50413652(CHEMBL457539)
Affinity DataIC50:  14.1nMAssay Description:Displacement of [125I]iodomelatonin from MT3/QR2 melatonin binding site expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50515995(CHEMBL4435240)
Affinity DataIC50:  15nMAssay Description:Inhibition of recombinant human NQO2 expressed in Escherichia coli using DCPIP as substrate by spectrophotometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50150962(CHEMBL3770366)
Affinity DataIC50:  15nMAssay Description:Inhibition of human recombinant NQO2 using DCPIPas substrate and NRH as cofactor measured for 1 min by spectrophotometry in the absence of BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50150963(CHEMBL3770674)
Affinity DataIC50:  15nMAssay Description:Inhibition of human recombinant NQO2 using DCPIPas substrate and NRH as cofactor measured for 1 min by spectrophotometry in the absence of BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50413644(CHEMBL446329)
Affinity DataIC50:  15.8nMAssay Description:Displacement of [125I]iodomelatonin from MT3/QR2 melatonin binding site expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50008344(5-(2-(diethylamino)ethylamino)-8-hydroxy-1-methyl-...)
Affinity DataIC50:  16nMAssay Description:Inhibition of human recombinant NQO2 assessed as reduction of DCPIP by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50317138(5-(2-(diethylamino)ethylamino)-7,10-dimethoxy-6H-i...)
Affinity DataIC50:  17nMAssay Description:Inhibition of human recombinant NQO2 assessed as reduction of DCPIP by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50515985(CHEMBL1237241 | TCMDC-142036)
Affinity DataIC50:  18nMAssay Description:Inhibition of recombinant human NQO2 expressed in Escherichia coli using DCPIP as substrate by spectrophotometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50342770(CHEMBL456727 | N-(2-(7-(methylthio)naphthalen-1-yl...)
Affinity DataIC50:  18nMAssay Description:Binding affinity to human MT3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50260398(CHEMBL494566 | N-(2-(5-Methoxycarbonyl-benzo[b]fur...)
Affinity DataIC50:  18.2nMAssay Description:Displacement of [125I]iodomelatonin from MT3/QR2 melatonin binding site expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50342770(CHEMBL456727 | N-(2-(7-(methylthio)naphthalen-1-yl...)
Affinity DataIC50:  18.2nMAssay Description:Displacement of [125I]iodomelatonin from MT3/QR2 melatonin binding site expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50342772(CHEMBL458209 | N-(2-(7-(methylsulfonyl)naphthalen-...)
Affinity DataIC50:  20.9nMAssay Description:Displacement of [125I]iodomelatonin from MT3/QR2 melatonin binding site expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50342772(CHEMBL458209 | N-(2-(7-(methylsulfonyl)naphthalen-...)
Affinity DataIC50:  21nMAssay Description:Binding affinity to human MT3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50260407(CHEMBL521826 | N-(2-(5-Methoxycarbonylamino-benzo[...)
Affinity DataIC50:  22.9nMAssay Description:Displacement of [125I]iodomelatonin from MT3/QR2 melatonin binding site expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50413639(CHEMBL456691)
Affinity DataIC50:  24.0nMAssay Description:Displacement of [125I]iodomelatonin from MT3/QR2 melatonin binding site expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50150962(CHEMBL3770366)
Affinity DataIC50:  24nMAssay Description:Inhibition of human recombinant NQO2 using DCPIPas substrate and NRH as cofactor measured for 1 min by spectrophotometry in the prsence of BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50151002(CHEMBL3770215)
Affinity DataIC50:  27nMAssay Description:Inhibition of human recombinant NQO2 using DCPIPas substrate and NRH as cofactor measured for 1 min by spectrophotometry in the absence of BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50150963(CHEMBL3770674)
Affinity DataIC50:  28nMAssay Description:Inhibition of human recombinant NQO2 using DCPIPas substrate and NRH as cofactor measured for 1 min by spectrophotometry in the prsence of BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50413649(CHEMBL443636)
Affinity DataIC50:  28.2nMAssay Description:Displacement of [125I]iodomelatonin from MT3/QR2 melatonin binding site expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50037241(CHEMBL34348 | N-(2-(7-methoxynaphthalen-1-yl)ethyl...)
Affinity DataIC50:  28.8nMAssay Description:Displacement of [125I]iodomelatonin from MT3/QR2 melatonin binding site expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50317139(5-(2-(diethylamino)ethylamino)-7-hydroxy-10-methox...)
Affinity DataIC50:  31nMAssay Description:Inhibition of human recombinant NQO2 assessed as reduction of DCPIP by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50342773(CHEMBL457763 | N-(2-(7-sulfamoylnaphthalen-1-yl)et...)
Affinity DataIC50:  32nMAssay Description:Binding affinity to human MT3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50342773(CHEMBL457763 | N-(2-(7-sulfamoylnaphthalen-1-yl)et...)
Affinity DataIC50:  32.4nMAssay Description:Displacement of [125I]iodomelatonin from MT3/QR2 melatonin binding site expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50388602(FURAMIDINE)
Affinity DataIC50:  35nMAssay Description:Inhibition of human recombinant NQO2 using DCPIPas substrate and NRH as cofactor measured for 1 min by spectrophotometry in the absence of BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50388602(FURAMIDINE)
Affinity DataIC50:  35nMAssay Description:Inhibition of recombinant human NQO2 assessed as change in rate of decolouration of DCPIP measured over 1 min by spectrophotometric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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