TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of Toledo
Curated by ChEMBL
University Of Toledo
Curated by ChEMBL
Affinity DataKd: 0.0300nMAssay Description:Binding of [3H]-QNB to HM1 receptor was evaluated by saturation binding assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of Toledo
Curated by ChEMBL
University Of Toledo
Curated by ChEMBL
Affinity DataKd: 0.0400nMAssay Description:Binding of [3H]-QNB to HM1 receptor was evaluated by saturation binding assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of Toledo
Curated by ChEMBL
University Of Toledo
Curated by ChEMBL
Affinity DataKd: 0.170nMAssay Description:Displacement of [3H]N-methylscopolamine from human muscarinic acetylcholine M1 receptor stably expressed in CHO cells by radioligand competition bind...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of Toledo
Curated by ChEMBL
University Of Toledo
Curated by ChEMBL
Affinity DataKd: 0.170nMAssay Description:Displacement of [3H]N-methylscopolamine from human muscarinic acetylcholine M1 receptor stably expressed in CHO cells by radioligand competition bind...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of Toledo
Curated by ChEMBL
University Of Toledo
Curated by ChEMBL
Affinity DataKd: 0.170nMAssay Description:Displacement of [3H]N-methylscopolamine from human muscarinic acetylcholine M1 receptor stably expressed in CHO cells by radioligand competition bind...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of Toledo
Curated by ChEMBL
University Of Toledo
Curated by ChEMBL
Affinity DataKd: 0.170nMAssay Description:Displacement of [3H]N-methylscopolamine from human muscarinic acetylcholine M1 receptor stably expressed in CHO cells by radioligand competition bind...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of Toledo
Curated by ChEMBL
University Of Toledo
Curated by ChEMBL
Affinity DataKd: 0.200nMAssay Description:Antagonist activity at human recombinant muscarinic M1 receptor expressed in CHO cells assessed as inhibition of acetylcholine-induced calcium mobili...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of Toledo
Curated by ChEMBL
University Of Toledo
Curated by ChEMBL
Affinity DataKd: 0.813nMAssay Description:Displacement of [3H]-UR-SK259 human muscarinic M1 receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of Toledo
Curated by ChEMBL
University Of Toledo
Curated by ChEMBL
Affinity DataKd: 1.5nMAssay Description:Displacement of [3H]-QNB from muscarinic receptor 1 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of Toledo
Curated by ChEMBL
University Of Toledo
Curated by ChEMBL
Affinity DataKd: 2.51nMAssay Description:Antagonist activity at human recombinant muscarinic M1 receptor expressed in CHO cells assessed as inhibition of acetylcholine-induced intracellular ...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of Toledo
Curated by ChEMBL
University Of Toledo
Curated by ChEMBL
Affinity DataKd: 2.70nMAssay Description:Displacement of [3H]-QNB from muscarinic receptor 1 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of Toledo
Curated by ChEMBL
University Of Toledo
Curated by ChEMBL
Affinity DataKd: 3.40nMAssay Description:Displacement of [3H]-QNB from muscarinic receptor 1 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of Toledo
Curated by ChEMBL
University Of Toledo
Curated by ChEMBL
Affinity DataKd: 4.10nMAssay Description:Apparent dissociation constant for human muscarinic receptor M1 from FRET based binding assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of Toledo
Curated by ChEMBL
University Of Toledo
Curated by ChEMBL
Affinity DataKd: 4.90nMAssay Description:Displacement of [3H]-QNB from rat brain stem muscarinic receptor 2 (M2)More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of Toledo
Curated by ChEMBL
University Of Toledo
Curated by ChEMBL
Affinity DataKd: 4.92nMAssay Description:Displacement of [3H]-QNB from muscarinic receptor 1 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of Toledo
Curated by ChEMBL
University Of Toledo
Curated by ChEMBL
Affinity DataKd: 5nMAssay Description:Displacement of [3H]-QNB from muscarinic receptor 1 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of Toledo
Curated by ChEMBL
University Of Toledo
Curated by ChEMBL
Affinity DataKd: 5.20nMAssay Description:Displacement of [3H]-QNB from muscarinic receptor 1 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of Toledo
Curated by ChEMBL
University Of Toledo
Curated by ChEMBL
Affinity DataKd: 6.5nMAssay Description:Binding affinity to human muscarinic M1 receptor expressed in CHO-K9 cells incubated in dark at 22 degree C for 2 hrs by FACSCalibur flow cytometric ...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of Toledo
Curated by ChEMBL
University Of Toledo
Curated by ChEMBL
Affinity DataKd: 10nMAssay Description:Binding affinity to human muscarinic M1 receptor expressed in CHO-K9 cells incubated in dark measured after 60 mins by Hoechst H33342 dye based confo...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of Toledo
Curated by ChEMBL
University Of Toledo
Curated by ChEMBL
Affinity DataKd: 12nMAssay Description:Displacement of [3H]-QNB from muscarinic receptor 1 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of Toledo
Curated by ChEMBL
University Of Toledo
Curated by ChEMBL
Affinity DataKd: 13nMAssay Description:Apparent dissociation constant for human muscarinic receptor M1 from FRET based binding assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of Toledo
Curated by ChEMBL
University Of Toledo
Curated by ChEMBL
Affinity DataKd: 13nMAssay Description:Apparent dissociation constant for human muscarinic receptor M1 from FRET based binding assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of Toledo
Curated by ChEMBL
University Of Toledo
Curated by ChEMBL
Affinity DataKd: 14nMAssay Description:Apparent dissociation constant for human muscarinic receptor M1 from FRET based binding assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of Toledo
Curated by ChEMBL
University Of Toledo
Curated by ChEMBL
Affinity DataKd: 15.8nMAssay Description:Antagonist activity at human recombinant muscarinic M1 receptor expressed in CHO cells assessed as inhibition of acetylcholine-induced intracellular ...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of Toledo
Curated by ChEMBL
University Of Toledo
Curated by ChEMBL
Affinity DataKd: 15.8nMAssay Description:Antagonist activity at human recombinant muscarinic M1 receptor expressed in CHO cells assessed as inhibition of acetylcholine-induced intracellular ...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of Toledo
Curated by ChEMBL
University Of Toledo
Curated by ChEMBL
Affinity DataKd: 19nMAssay Description:Apparent dissociation constant for human muscarinic receptor M1 from FRET based binding assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of Toledo
Curated by ChEMBL
University Of Toledo
Curated by ChEMBL
Affinity DataKd: 20nMAssay Description:Apparent dissociation constant for human muscarinic receptor M1 from FRET based binding assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of Toledo
Curated by ChEMBL
University Of Toledo
Curated by ChEMBL
Affinity DataKd: 22nMAssay Description:Apparent dissociation constant for human muscarinic receptor M1 from FRET based binding assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of Toledo
Curated by ChEMBL
University Of Toledo
Curated by ChEMBL
Affinity DataKd: 24nMAssay Description:Displacement of [3H]-QNB from muscarinic receptor 1 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of Toledo
Curated by ChEMBL
University Of Toledo
Curated by ChEMBL
Affinity DataKd: 26nMAssay Description:Binding affinity to human muscarinic M1 receptor expressed in CHO-K9 cells incubated in dark measured after 60 mins by Hoechst H33342 dye based confo...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of Toledo
Curated by ChEMBL
University Of Toledo
Curated by ChEMBL
Affinity DataKd: 31.6nMAssay Description:Antagonist activity at human recombinant muscarinic M1 receptor expressed in CHO cells assessed as inhibition of acetylcholine-induced intracellular ...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of Toledo
Curated by ChEMBL
University Of Toledo
Curated by ChEMBL
Affinity DataKd: 36nMAssay Description:Apparent dissociation constant for human muscarinic receptor M1 from FRET based binding assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of Toledo
Curated by ChEMBL
University Of Toledo
Curated by ChEMBL
Affinity DataKd: 39.8nMAssay Description:Antagonist activity at human recombinant muscarinic M1 receptor expressed in CHO cells assessed as inhibition of acetylcholine-induced intracellular ...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of Toledo
Curated by ChEMBL
University Of Toledo
Curated by ChEMBL
Affinity DataKd: 72nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 acetylcholine receptor expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of Toledo
Curated by ChEMBL
University Of Toledo
Curated by ChEMBL
Affinity DataKd: 74nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 acetylcholine receptor expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of Toledo
Curated by ChEMBL
University Of Toledo
Curated by ChEMBL
Affinity DataKd: 79.4nMAssay Description:Antagonist activity at human recombinant muscarinic M1 receptor expressed in CHO cells assessed as inhibition of acetylcholine-induced intracellular ...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of Toledo
Curated by ChEMBL
University Of Toledo
Curated by ChEMBL
Affinity DataKd: 79.4nMAssay Description:Antagonist activity at human recombinant muscarinic M1 receptor expressed in CHO cells assessed as inhibition of acetylcholine-induced intracellular ...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of Toledo
Curated by ChEMBL
University Of Toledo
Curated by ChEMBL
Affinity DataKd: 126nMAssay Description:Antagonist activity at human recombinant muscarinic M1 receptor expressed in CHO cells assessed as inhibition of acetylcholine-induced intracellular ...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of Toledo
Curated by ChEMBL
University Of Toledo
Curated by ChEMBL
Affinity DataKd: 141nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 acetylcholine receptor expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of Toledo
Curated by ChEMBL
University Of Toledo
Curated by ChEMBL
Affinity DataKd: 148nMAssay Description:Binding affinity against M1 receptor expressed in CHO-K1 cells transfected with human muscarinic receptor sequence using radioligand [3H]-quinuclidin...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of Toledo
Curated by ChEMBL
University Of Toledo
Curated by ChEMBL
Affinity DataKd: 151nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 acetylcholine receptor expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of Toledo
Curated by ChEMBL
University Of Toledo
Curated by ChEMBL
Affinity DataKd: 151nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 acetylcholine receptor expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of Toledo
Curated by ChEMBL
University Of Toledo
Curated by ChEMBL
Affinity DataKd: 158nMAssay Description:Antagonist activity at human recombinant muscarinic M1 receptor expressed in CHO cells assessed as inhibition of acetylcholine-induced intracellular ...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of Toledo
Curated by ChEMBL
University Of Toledo
Curated by ChEMBL
Affinity DataKd: 166nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 acetylcholine receptor expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of Toledo
Curated by ChEMBL
University Of Toledo
Curated by ChEMBL
Affinity DataKd: 167nMAssay Description:Binding affinity against M1 receptor expressed in CHO-K1 cells transfected with human muscarinic receptor sequence using radioligand [3H]-quinuclidin...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of Toledo
Curated by ChEMBL
University Of Toledo
Curated by ChEMBL
Affinity DataKd: 168nMAssay Description:Displacement of [3H]-QNB from muscarinic receptor 1 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of Toledo
Curated by ChEMBL
University Of Toledo
Curated by ChEMBL
Affinity DataKd: 423nMAssay Description:Binding affinity against M1 receptor expressed in CHO-K1 cells transfected with human muscarinic receptor sequence using radioligand [3H]-quinuclidin...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of Toledo
Curated by ChEMBL
University Of Toledo
Curated by ChEMBL
Affinity DataKd: 490nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 acetylcholine receptor expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of Toledo
Curated by ChEMBL
University Of Toledo
Curated by ChEMBL
Affinity DataKd: 494nMAssay Description:Binding affinity against M1 receptor expressed in CHO-K1 cells transfected with human muscarinic receptor sequence using radioligand [3H]-quinuclidin...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of Toledo
Curated by ChEMBL
University Of Toledo
Curated by ChEMBL
Affinity DataKd: 605nMAssay Description:Binding affinity against M1 receptor expressed in CHO-K1 cells transfected with human muscarinic receptor sequence using radioligand [3H]-quinuclidin...More data for this Ligand-Target Pair