Compile Data Set for Download or QSAR
maximum 50k data
Found 13 of kd data for polymerid = 2104,49000778,49000780
TargetSubstance-P receptor(Rattus norvegicus (rat))
Rochester

Curated by ChEMBL
LigandPNGBDBM50002462(1,3-Diethyl-2-[3-(1,3,3-trimethyl-1,3-dihydro-indo...)
Affinity DataKd:  0.180nMAssay Description:Scatchard analysis at concentration of the 3 uM :Apparent affinity constant (Kd) against tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50000041((+) (2-Methoxy-benzyl)-(2-phenyl-piperidin-3-yl)-a...)
Affinity DataKd:  0.320nMAssay Description:Evaluated for the binding affinity towards NK1 receptor in the striatal membranes of guinea pigMore data for this Ligand-Target Pair
TargetSubstance-P receptor(Rattus norvegicus (rat))
Rochester

Curated by ChEMBL
LigandPNGBDBM50002462(1,3-Diethyl-2-[3-(1,3,3-trimethyl-1,3-dihydro-indo...)
Affinity DataKd:  0.970nMAssay Description:Scatchard analysis at concentration of the 1 uM :Apparent affinity constant (Kd) against tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Rochester

Curated by ChEMBL
LigandPNGBDBM50002462(1,3-Diethyl-2-[3-(1,3,3-trimethyl-1,3-dihydro-indo...)
Affinity DataKd:  1.5nMAssay Description:Scatchard analysis at concentration of the 10 uM :Apparent affinity constant (Kd) against tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50403168(CHEMBL367312)
Affinity DataKd:  39.8nMAssay Description:The compound was evaluated in vitro for the antagonistic activity against substance P receptor in guinea pig myenteric plexus longitudinal muscle str...More data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-P receptor(GUINEA PIG)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50406736(CHEMBL406142)
Affinity DataKd:  100nMAssay Description:Tested for antagonist activity toward NK-1 receptor in guinea pig ileum against the agonist eledoisinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50403167(CHEMBL172794)
Affinity DataKd:  126nMAssay Description:The compound was evaluated in vitro for the antagonistic activity against Tachykinin receptor 1 in guinea pig myenteric plexus longitudinal muscle st...More data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-P receptor(GUINEA PIG)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50403165(CHEMBL424567)
Affinity DataKd:  200nMAssay Description:The compound was evaluated in vitro for the antagonistic activity against substance P receptor in guinea pig myenteric plexus longitudinal muscle str...More data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-P receptor(GUINEA PIG)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50406739(CHEMBL266884)
Affinity DataKd:  251nMAssay Description:Tested for antagonist activity toward NK-1 receptor in guinea pig ileum against the agonist eledoisinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50403166(CHEMBL170299)
Affinity DataKd:  398nMAssay Description:The compound was evaluated in vitro for the antagonistic activity against substance P receptor in guinea pig myenteric plexus longitudinal muscle str...More data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-P receptor(GUINEA PIG)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50403170(CHEMBL435717)
Affinity DataKd:  501nMAssay Description:The compound was evaluated in vitro for the antagonistic activity against substance P receptor in guinea pig myenteric plexus longitudinal muscle str...More data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-P receptor(GUINEA PIG)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50403169(CHEMBL405167)
Affinity DataKd:  1.26E+3nMAssay Description:The compound was evaluated in vitro for the antagonistic activity against substance P receptor in guinea pig myenteric plexus longitudinal muscle str...More data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-P receptor(GUINEA PIG)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50406733(CHEMBL2370702)
Affinity DataKd:  2.00E+3nMAssay Description:Tested for antagonist activity toward NK-1 receptor in guinea pig ileum against the agonist eledoisin (mean +/-, n=4)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed