Found 206 of kd data for polymerid = 2130,2135,4341,5768 TargetAdenosine receptor A3(Homo sapiens (Human))
National And Kapodistrian University Of Athens
Curated by ChEMBL
National And Kapodistrian University Of Athens
Curated by ChEMBL
Affinity DataKd: 0.0776nMAssay Description:Binding affinity to Nluc-A3R (unknown origin) expressed in HEK293 cells by nanoBRET assayMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
National And Kapodistrian University Of Athens
Curated by ChEMBL
National And Kapodistrian University Of Athens
Curated by ChEMBL
Affinity DataKd: 0.0977nMAssay Description:Binding affinity to wild type A3R (unknown origin) expressed in Flp-In-CHO cells assessed as dissociation constant by by Schild analysisMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
National And Kapodistrian University Of Athens
Curated by ChEMBL
National And Kapodistrian University Of Athens
Curated by ChEMBL
Affinity DataKd: 0.158nMAssay Description:Antagonist activity at human recombinant adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKd: 0.170nMAssay Description:Binding affinity to human adenosine A2B receptorMore data for this Ligand-Target Pair
Affinity DataKd: 0.220nMAssay Description:The membranes prepared from Flp-In HEK cells transfected with adenosine receptors were used in binding assays. Nonspecific binding was determined in ...More data for this Ligand-Target Pair
3D Structure (crystal)Affinity DataKd: 0.220nMpH: 7.4 T: 2°CAssay Description:The membranes prepared from Flp-In HEK cells transfected with adenosine receptors were used in binding assays. Nonspecific binding was determined in ...More data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
National And Kapodistrian University Of Athens
Curated by ChEMBL
National And Kapodistrian University Of Athens
Curated by ChEMBL
Affinity DataKd: 0.331nMAssay Description:Antagonist activity at human adenosine A3 receptor expressed in forskolin-stimulated CHO cells assessed as inhibition of NECA-induced CRE-SPAP gene t...More data for this Ligand-Target Pair
Affinity DataKd: 0.403nMAssay Description:Binding affinity to human recombinant adenosine A2B receptor expressed in CHO cells by saturation experimentMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
National And Kapodistrian University Of Athens
Curated by ChEMBL
National And Kapodistrian University Of Athens
Curated by ChEMBL
Affinity DataKd: 0.437nMAssay Description:Antagonist activity at human adenosine A3 receptor expressed in forskolin-stimulated CHO cells assessed as inhibition of NECA-induced CRE-SPAP gene t...More data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
National And Kapodistrian University Of Athens
Curated by ChEMBL
National And Kapodistrian University Of Athens
Curated by ChEMBL
Affinity DataKd: 0.460nMAssay Description:Binding affinity to human adenosine A3R expressed in CHO cells membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
National And Kapodistrian University Of Athens
Curated by ChEMBL
National And Kapodistrian University Of Athens
Curated by ChEMBL
Affinity DataKd: 0.550nMAssay Description:Binding affinity to human adenosine A3 receptor expressed in HEK293 cells measured by radioligand binding assayMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
National And Kapodistrian University Of Athens
Curated by ChEMBL
National And Kapodistrian University Of Athens
Curated by ChEMBL
Affinity DataKd: 0.550nMAssay Description:Binding affinity to adenosine A3R (unknown origin)More data for this Ligand-Target Pair
Affinity DataKd: 0.652nMAssay Description:Binding affinity to human recombinant adenosine A2B receptor expressed in CHO cells by kinetic experimentMore data for this Ligand-Target Pair
Affinity DataKd: 0.700nMAssay Description:Displacement of 2-[2-(4-amino-3-[125I]iodophenyl)ethylamino]adenosine from human recombinant adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
University Of Virginia School Of Medicine
Curated by ChEMBL
University Of Virginia School Of Medicine
Curated by ChEMBL
Affinity DataKd: 0.800nMAssay Description:Binding affinity towards adenosine A1 receptor in rat brain membrane(KD)More data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
University Of Virginia School Of Medicine
Curated by ChEMBL
University Of Virginia School Of Medicine
Curated by ChEMBL
Affinity DataKd: 0.800nMAssay Description:Binding affinity towards adenosine A1 receptor in rat brain membrane(KD)More data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
National And Kapodistrian University Of Athens
Curated by ChEMBL
National And Kapodistrian University Of Athens
Curated by ChEMBL
Affinity DataKd: 0.820nMAssay Description:Binding affinity against human Adenosine A3 receptor in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKd: 1.10nMAssay Description:Binding affinity to human wild type adenosine A2B receptor expressed in Expi293F cells assessed as affinity on-rate by surface plasmon resonance assa...More data for this Ligand-Target Pair
Affinity DataKd: 1.13nMAssay Description:Binding affinity to human adenosine A2B receptorMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
University Of Virginia School Of Medicine
Curated by ChEMBL
University Of Virginia School Of Medicine
Curated by ChEMBL
Affinity DataKd: 1.20nMAssay Description:Binding affinity towards adenosine A1 receptor in rat brain membrane(KD)More data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
University Of Virginia School Of Medicine
Curated by ChEMBL
University Of Virginia School Of Medicine
Curated by ChEMBL
Affinity DataKd: 1.30nMAssay Description:Displacement of [3H] CGS 21680 from rat hippocampus adenosine A1 receptorMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
University Of Virginia School Of Medicine
Curated by ChEMBL
University Of Virginia School Of Medicine
Curated by ChEMBL
Affinity DataKd: 1.40nMAssay Description:Kd value for adenosine A1 receptor binding at 14.5 uMMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
National And Kapodistrian University Of Athens
Curated by ChEMBL
National And Kapodistrian University Of Athens
Curated by ChEMBL
Affinity DataKd: 1.42nMpH: 7.4 T: 2°CAssay Description:.(R)- and (S)-(4-Fluorophenyl)(4-((5-methyl-1H-pyrazol-3-yl)amino)quinazolin-2-yl)methanol was tested in a radioligand binding assay, according to th...More data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
National And Kapodistrian University Of Athens
Curated by ChEMBL
National And Kapodistrian University Of Athens
Curated by ChEMBL
Affinity DataKd: 1.5nMAssay Description:Antagonist activity at human adenosine A3 receptor expressed in forskolin-stimulated CHO cells assessed as inhibition of NECA-induced CRE-SPAP gene t...More data for this Ligand-Target Pair
Affinity DataKd: 1.5nMAssay Description:Binding affinity to human wild type adenosine A2B receptor expressed in Expi293F cells assessed as affinity off-rate by surface plasmon resonance ass...More data for this Ligand-Target Pair
Affinity DataKd: 1.5nMAssay Description:Binding affinity to human wild type adenosine A2B receptor expressed in Expi293F cells assessed as affinity on-rate by surface plasmon resonance assa...More data for this Ligand-Target Pair
Affinity DataKd: 1.65nMAssay Description:Binding affinity to human adenosine A2B receptorMore data for this Ligand-Target Pair
Affinity DataKd: 1.70nMAssay Description:Binding affinity of [3H]-MRE 2029-F20 towards human adenosine A2b receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKd: 1.80nMAssay Description:Displacement of [3H] ZM241385 from human A2AAR S227A mutant expressed in CHO cells assessed as dissociation constant incubated for 60 mins by radioli...More data for this Ligand-Target Pair
Affinity DataKd: 2nMAssay Description:Displacement of [3H] ZM241385 from wild type human A2AAR expressed in CHO cells assessed as dissociation constant incubated for 60 mins by radioligan...More data for this Ligand-Target Pair
Affinity DataKd: 2.20nMAssay Description:Displacement of [3H]4-[2-[7-amino-2-(2-furyl)-1,2,4-triazolo[1,5-a][1,3,5]triazin-5-yl-amino]ethylphenol from wild type human adenosine A2a receptor ...More data for this Ligand-Target Pair
Affinity DataKd: 2.70nMAssay Description:Displacement of [3H] ZM241385 from human A2AAR S277A/H278A double mutant expressed in CHO cells assessed as dissociation constant incubated for 60 mi...More data for this Ligand-Target Pair
Affinity DataKd: 2.90nMAssay Description:Displacement of [3H] ZM241385 from human A2AAR H278A mutant expressed in CHO cells assessed as dissociation constant incubated for 60 mins by radioli...More data for this Ligand-Target Pair
Affinity DataKd: 3.20nMAssay Description:Displacement of [3H]4-[2-[7-amino-2-(2-furyl)-1,2,4-triazolo[1,5-a][1,3,5]triazin-5-yl-amino]ethylphenol from wild type human adenosine A2a receptor ...More data for this Ligand-Target Pair
Affinity DataKd: 3.20nMAssay Description:Displacement of [3H]4-[2-[7-amino-2-(2-furyl)-1,2,4-triazolo[1,5-a][1,3,5]triazin-5-yl-amino]ethylphenol from wild type human adenosine A2a receptor ...More data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
National And Kapodistrian University Of Athens
Curated by ChEMBL
National And Kapodistrian University Of Athens
Curated by ChEMBL
Affinity DataKd: 3.40nMAssay Description:Antagonist activity at human adenosine A3 receptor expressed in forskolin-stimulated CHO cells assessed as inhibition of NECA-induced CRE-SPAP gene t...More data for this Ligand-Target Pair
Affinity DataKd: 4.30nMpH: 5.5Assay Description:Saturation binding of mutant human Adenosine A2A receptor (H250N) at pH 5.5More data for this Ligand-Target Pair
Affinity DataKd: 4.40nMAssay Description:Displacement of [3H]4-[2-[7-amino-2-(2-furyl)-1,2,4-triazolo[1,5-a][1,3,5]triazin-5-yl-amino]ethylphenol from wild type human adenosine A2a receptor ...More data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
National And Kapodistrian University Of Athens
Curated by ChEMBL
National And Kapodistrian University Of Athens
Curated by ChEMBL
Affinity DataKd: 4.90nMAssay Description:Binding affinity to human recombinant A3 adenosine receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKd: 5nMAssay Description:Displacement of [3H]4-[2-[7-amino-2-(2-furyl)-1,2,4-triazolo[1,5-a][1,3,5]triazin-5-yl-amino]ethylphenol from wild type human adenosine A2a receptor ...More data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
National And Kapodistrian University Of Athens
Curated by ChEMBL
National And Kapodistrian University Of Athens
Curated by ChEMBL
Affinity DataKd: 5.01nMAssay Description:Antagonist activity at human adenosine A3 receptor expressed in CHO cells assessed as inhibition of Cl-IB-MECA-mediated cyclic AMP productionMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
National And Kapodistrian University Of Athens
Curated by ChEMBL
National And Kapodistrian University Of Athens
Curated by ChEMBL
Affinity DataKd: 5.60nMAssay Description:Antagonist activity at human adenosine A3 receptor expressed in forskolin-stimulated CHO cells assessed as inhibition of NECA-induced CRE-SPAP gene t...More data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
National And Kapodistrian University Of Athens
Curated by ChEMBL
National And Kapodistrian University Of Athens
Curated by ChEMBL
Affinity DataKd: 6.20nMAssay Description:Antagonist activity at N-terminal NLuc tagged human A3 adenosine receptorMore data for this Ligand-Target Pair
Affinity DataKd: 7.60nMAssay Description:Kd in saturation experiments using [3H]CGS-21680 at H250N mutant receptor in COS-7 cellsMore data for this Ligand-Target Pair
Affinity DataKd: 7.60nMpH: 6.8Assay Description:Saturation binding of human Adenosine A2A receptor (H250N) at pH 6.8More data for this Ligand-Target Pair
Affinity DataKd: 7.80nMAssay Description:Binding affinity to NLuc human A2B adenosine receptor expressed in HEK293-A cells in presence of 1 uM PSB603 by NanoBRET binding assayMore data for this Ligand-Target Pair
Affinity DataKd: 9.10nMAssay Description:Binding affinity to human wild type adenosine A2A receptor expressed in Expi293F cells assessed as dissociation constant by surface plasmon resonance...More data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
National And Kapodistrian University Of Athens
Curated by ChEMBL
National And Kapodistrian University Of Athens
Curated by ChEMBL
Affinity DataKd: 9.10nMAssay Description:Binding affinity to N-terminal Nano-luc tagged human adenosine A3R expressed in HEK293 cells membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
National And Kapodistrian University Of Athens
Curated by ChEMBL
National And Kapodistrian University Of Athens
Curated by ChEMBL
Affinity DataKd: 10nMAssay Description:Binding affinity to Nluc-A3R (unknown origin) expressed in HEK293 cells by nanoBRET assayMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
University Of Virginia School Of Medicine
Curated by ChEMBL
University Of Virginia School Of Medicine
Curated by ChEMBL
Affinity DataKd: 11nMAssay Description:Kd value for adenosine A1 receptor binding at 145 uMMore data for this Ligand-Target Pair
