TargetTranslocator protein(Rattus norvegicus (rat))
Brain And Mind Research Institute
Curated by ChEMBL
Brain And Mind Research Institute
Curated by ChEMBL
Affinity DataKd: 0.600nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat cortexMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Brain And Mind Research Institute
Curated by ChEMBL
Brain And Mind Research Institute
Curated by ChEMBL
Affinity DataKd: 1.10nMAssay Description:Displacement of [3H]Ro5-4864 from TSPO in rat kainate lesioned striatumMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Brain And Mind Research Institute
Curated by ChEMBL
Brain And Mind Research Institute
Curated by ChEMBL
Affinity DataKd: 2nMAssay Description:Binding affinity constant for peripheral (mitochondrial) Benzodiazepine receptorMore data for this Ligand-Target Pair
Affinity DataKd: 2nMAssay Description:Binding affinity to human PBRMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Brain And Mind Research Institute
Curated by ChEMBL
Brain And Mind Research Institute
Curated by ChEMBL
Affinity DataKd: 3nMAssay Description:Displacement of [3H]SSR180575 from TSPO in rat cortexMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Brain And Mind Research Institute
Curated by ChEMBL
Brain And Mind Research Institute
Curated by ChEMBL
Affinity DataKd: 3.17nMAssay Description:Irreversible binding affinity to TSPO in rat kidney mitochondrial membraneMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Brain And Mind Research Institute
Curated by ChEMBL
Brain And Mind Research Institute
Curated by ChEMBL
Affinity DataKd: 3.5nMAssay Description:Binding affinity constant for Benzodiazepine receptor in rat RG-2 glioma cellsMore data for this Ligand-Target Pair
Affinity DataKd: 3.5nMAssay Description:Binding affinity to human PBRMore data for this Ligand-Target Pair
Affinity DataKd: 4nMAssay Description:Binding affinity to human PBRMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Brain And Mind Research Institute
Curated by ChEMBL
Brain And Mind Research Institute
Curated by ChEMBL
Affinity DataKd: 5.07nMAssay Description:Irreversible binding affinity to TSPO in rat kidney mitochondrial membraneMore data for this Ligand-Target Pair
Affinity DataKd: 6nMAssay Description:Binding affinity to human PBRMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Brain And Mind Research Institute
Curated by ChEMBL
Brain And Mind Research Institute
Curated by ChEMBL
Affinity DataKd: 8.31nMAssay Description:Irreversible binding affinity to TSPO in rat kidney mitochondrial membraneMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Brain And Mind Research Institute
Curated by ChEMBL
Brain And Mind Research Institute
Curated by ChEMBL
Affinity DataKd: >10nMAssay Description:Binding affinity constant for peripheral (mitochondrial) Benzodiazepine receptorMore data for this Ligand-Target Pair
Affinity DataKd: 11nMAssay Description:Inhibition concentration against human adenosine kinaseMore data for this Ligand-Target Pair
Affinity DataKd: 11nMAssay Description:Binding affinity to recombinant human TSPO by SPR assayMore data for this Ligand-Target Pair
Affinity DataKd: 40nMAssay Description:Binding affinity to C-terminal DDK-tagged human recombinant full-length TSPO expressed in HEK293 cells by SPR assayMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Brain And Mind Research Institute
Curated by ChEMBL
Brain And Mind Research Institute
Curated by ChEMBL
Affinity DataKd: 58nMAssay Description:Binding affinity constant for peripheral (mitochondrial) Benzodiazepine receptorMore data for this Ligand-Target Pair
Affinity DataKd: 61nMAssay Description:Binding affinity to C-terminal DDK-tagged human recombinant full-length TSPO expressed in HEK293 cells by SPR assayMore data for this Ligand-Target Pair
Affinity DataKd: 108nMAssay Description:Binding affinity to recombinant human TSPO by SPR assayMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Brain And Mind Research Institute
Curated by ChEMBL
Brain And Mind Research Institute
Curated by ChEMBL
Affinity DataKd: 213nMAssay Description:Binding affinity constant for peripheral (mitochondrial) Benzodiazepine receptorMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Brain And Mind Research Institute
Curated by ChEMBL
Brain And Mind Research Institute
Curated by ChEMBL
Affinity DataKd: 1.30E+3nMAssay Description:Binding affinity constant for Benzodiazepine receptor in normal rat brain homogenateMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Brain And Mind Research Institute
Curated by ChEMBL
Brain And Mind Research Institute
Curated by ChEMBL
Affinity DataKd: 4.00E+3nMAssay Description:Binding affinity constant for Benzodiazepine receptor in rat C6 glioma cellsMore data for this Ligand-Target Pair