Compile Data Set for Download or QSAR
maximum 50k data
Found 38 of kd data for polymerid = 2972
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM13174((2S,4S)-1-[(2S)-3,3-dimethyl-2-[(2S)-2-(methylamin...)
Affinity DataKd:  5nMpH: 7.4 T: 2°CAssay Description:A fluorescence polarization anisotropy (FPA) competition assay was used to determine the affinities of compounds to BIR3 protein. Fluorescence polari...More data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM13176((2S,4S)-1-[(2S)-2-cyclohexyl-2-[(2S)-2-(methylamin...)
Affinity DataKd:  6nMpH: 7.4 T: 2°CAssay Description:A fluorescence polarization anisotropy (FPA) competition assay was used to determine the affinities of compounds to BIR3 protein. Fluorescence polari...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM13166((2S)-1-[(2S)-3,3-dimethyl-2-[(2S)-2-(methylamino)p...)
Affinity DataKd:  12nMpH: 7.4 T: 2°CAssay Description:A fluorescence polarization anisotropy (FPA) competition assay was used to determine the affinities of compounds to BIR3 protein. Fluorescence polari...More data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM13175((2S)-1-[(2S)-2-cyclohexyl-2-[(2S)-2-(methylamino)p...)
Affinity DataKd:  16nMpH: 7.4 T: 2°CAssay Description:A fluorescence polarization anisotropy (FPA) competition assay was used to determine the affinities of compounds to BIR3 protein. Fluorescence polari...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM13168((2S)-N-[(1R)-2,3-dihydro-1H-inden-1-yl]-1-[(2S)-3,...)
Affinity DataKd:  29nMpH: 7.4 T: 2°CAssay Description:A fluorescence polarization anisotropy (FPA) competition assay was used to determine the affinities of compounds to BIR3 protein. Fluorescence polari...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM13172((2S)-1-[(2S)-3,3-dimethyl-2-[(2S)-2-(methylamino)p...)
Affinity DataKd:  47nMpH: 7.4 T: 2°CAssay Description:A fluorescence polarization anisotropy (FPA) competition assay was used to determine the affinities of compounds to BIR3 protein. Fluorescence polari...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM13173((2S)-1-[(2S)-3,3-dimethyl-2-[(2S)-2-(methylamino)p...)
Affinity DataKd:  167nMpH: 7.4 T: 2°CAssay Description:A fluorescence polarization anisotropy (FPA) competition assay was used to determine the affinities of compounds to BIR3 protein. Fluorescence polari...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM13170((2S)-1-[(2S)-3,3-dimethyl-2-[(2S)-2-(methylamino)p...)
Affinity DataKd: >500nMpH: 7.4 T: 2°CAssay Description:A fluorescence polarization anisotropy (FPA) competition assay was used to determine the affinities of compounds to BIR3 protein. Fluorescence polari...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM13167((2S)-1-[(2S)-3,3-dimethyl-2-[(2S)-2-(methylamino)p...)
Affinity DataKd:  706nMpH: 7.4 T: 2°CAssay Description:A fluorescence polarization anisotropy (FPA) competition assay was used to determine the affinities of compounds to BIR3 protein. Fluorescence polari...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM13190((2S)-2-amino-N-[4-(4-bromophenyl)-5-phenyl-1,3-thi...)
Affinity DataKd:  740nMAssay Description:A fluorescence polarization anisotropy (FPA) competition assay was used to determine the affinities of compounds to BIR3 protein. Fluorescence polari...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM13180((2S)-1-[(2S)-3,3-dimethyl-2-[(2R)-2-(methylamino)p...)
Affinity DataKd: >1.00E+3nMpH: 7.4 T: 2°CAssay Description:A fluorescence polarization anisotropy (FPA) competition assay was used to determine the affinities of compounds to BIR3 protein. Fluorescence polari...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM13179((2S)-1-[(2S)-2-cyclohexyl-2-[(2S)-2-(dimethylamino...)
Affinity DataKd: >1.00E+3nMpH: 7.4 T: 2°CAssay Description:A fluorescence polarization anisotropy (FPA) competition assay was used to determine the affinities of compounds to BIR3 protein. Fluorescence polari...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM13177((2S)-1-[(2S)-2-[(2S)-2-(dimethylamino)propanamido]...)
Affinity DataKd: >1.00E+3nMpH: 7.4 T: 2°CAssay Description:A fluorescence polarization anisotropy (FPA) competition assay was used to determine the affinities of compounds to BIR3 protein. Fluorescence polari...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM13171((2S)-1-[(2S)-3,3-dimethyl-2-[(2S)-2-(methylamino)p...)
Affinity DataKd: >1.00E+3nMpH: 7.4 T: 2°CAssay Description:A fluorescence polarization anisotropy (FPA) competition assay was used to determine the affinities of compounds to BIR3 protein. Fluorescence polari...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM13169((2S)-N-[(1S)-2,3-dihydro-1H-inden-1-yl]-1-[(2S)-3,...)
Affinity DataKd: >1.00E+3nMpH: 7.4 T: 2°CAssay Description:A fluorescence polarization anisotropy (FPA) competition assay was used to determine the affinities of compounds to BIR3 protein. Fluorescence polari...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM13178((2S,4S)-1-[(2S)-2-[(2S)-2-(dimethylamino)propanami...)
Affinity DataKd: >1.00E+3nMpH: 7.4 T: 2°CAssay Description:A fluorescence polarization anisotropy (FPA) competition assay was used to determine the affinities of compounds to BIR3 protein. Fluorescence polari...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM13189((2S)-2-amino-N-(4,5-diphenyl-1,3-thiazol-2-yl)prop...)
Affinity DataKd:  1.10E+3nMAssay Description:A fluorescence polarization anisotropy (FPA) competition assay was used to determine the affinities of compounds to BIR3 protein. Fluorescence polari...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM13191((2S)-2-amino-N-[4-(4-benzylphenyl)-5-phenyl-1,3-th...)
Affinity DataKd:  1.20E+3nMAssay Description:A fluorescence polarization anisotropy (FPA) competition assay was used to determine the affinities of compounds to BIR3 protein. Fluorescence polari...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM13185((2S)-2-amino-N-{5-methyl-4-[(2,4,6-trimethylphenyl...)
Affinity DataKd:  2.00E+3nMpH: 7.4 T: 2°CAssay Description:A fluorescence polarization anisotropy (FPA) competition assay was used to determine the affinities of compounds to BIR3 protein. Fluorescence polari...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM13193((2S)-2-amino-N-[5-benzyl-4-(phenoxymethyl)-1,3-thi...)
Affinity DataKd:  4.10E+3nMAssay Description:A fluorescence polarization anisotropy (FPA) competition assay was used to determine the affinities of compounds to BIR3 protein. Fluorescence polari...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM13194((2S)-2-amino-N-{5-benzyl-4-[(benzyloxy)methyl]-1,3...)
Affinity DataKd:  4.10E+3nMAssay Description:A fluorescence polarization anisotropy (FPA) competition assay was used to determine the affinities of compounds to BIR3 protein. Fluorescence polari...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM13187((2S)-2-amino-N-(5-tert-butyl-4-phenyl-1,3-thiazol-...)
Affinity DataKd:  4.80E+3nMAssay Description:A fluorescence polarization anisotropy (FPA) competition assay was used to determine the affinities of compounds to BIR3 protein. Fluorescence polari...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM13199((2S)-2-amino-N-{5-thia-3-azatricyclo[7.4.0.0^{2,6}...)
Affinity DataKd:  5.60E+3nMAssay Description:A fluorescence polarization anisotropy (FPA) competition assay was used to determine the affinities of compounds to BIR3 protein. Fluorescence polari...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM13198((2S)-2-amino-N-{5-thia-3-azatricyclo[7.4.0.0^{2,6}...)
Affinity DataKd:  7.10E+3nMAssay Description:A fluorescence polarization anisotropy (FPA) competition assay was used to determine the affinities of compounds to BIR3 protein. Fluorescence polari...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM17336((2S)-2-{[(2S)-1-({2-[(1S)-1-aminoethyl]-1,3-oxazol...)
Affinity DataKd:  1.10E+4nMpH: 7.0 T: 2°CAssay Description:AVPC-badan can be displaced from the binding pocket of the protein by test compounds. As the dye is displaced from the binding pocket, the emission i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM13196((2S)-2-amino-N-{5-benzyl-4-[(naphthalen-2-yloxy)me...)
Affinity DataKd:  1.40E+4nMAssay Description:A fluorescence polarization anisotropy (FPA) competition assay was used to determine the affinities of compounds to BIR3 protein. Fluorescence polari...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM13186((2S)-2-amino-N-(5-methyl-4-phenyl-1,3-thiazol-2-yl...)
Affinity DataKd:  1.50E+4nMpH: 7.4 T: 2°CAssay Description:A fluorescence polarization anisotropy (FPA) competition assay was used to determine the affinities of compounds to BIR3 protein. Fluorescence polari...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM13188((2S)-2-amino-N-(4-methyl-5-phenyl-1,3-thiazol-2-yl...)
Affinity DataKd:  1.50E+4nMAssay Description:A fluorescence polarization anisotropy (FPA) competition assay was used to determine the affinities of compounds to BIR3 protein. Fluorescence polari...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM13181((2S)-2-amino-N-(5,7-dimethyl-1,8-naphthyridin-2-yl...)
Affinity DataKd:  2.00E+4nMpH: 7.4 T: 2°CAssay Description:A fluorescence polarization anisotropy (FPA) competition assay was used to determine the affinities of compounds to BIR3 protein. Fluorescence polari...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM13195((2S)-2-amino-N-{5-benzyl-4-[(naphthalen-1-yloxy)me...)
Affinity DataKd:  2.10E+4nMAssay Description:A fluorescence polarization anisotropy (FPA) competition assay was used to determine the affinities of compounds to BIR3 protein. Fluorescence polari...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM13197((2S)-2-amino-N-{5-benzyl-4-[(2,3-dihydro-1H-inden-...)
Affinity DataKd:  2.20E+4nMAssay Description:A fluorescence polarization anisotropy (FPA) competition assay was used to determine the affinities of compounds to BIR3 protein. Fluorescence polari...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM13182((2S)-2-amino-N-[5-(4-butoxyphenyl)-1,3,4-thiadiazo...)
Affinity DataKd:  2.50E+4nMpH: 7.4 T: 2°CAssay Description:A fluorescence polarization anisotropy (FPA) competition assay was used to determine the affinities of compounds to BIR3 protein. Fluorescence polari...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM13183((2S)-2-amino-N-(5-benzoyl-1H-1,3-benzodiazol-2-yl)...)
Affinity DataKd:  3.00E+4nMpH: 7.4 T: 2°CAssay Description:A fluorescence polarization anisotropy (FPA) competition assay was used to determine the affinities of compounds to BIR3 protein. Fluorescence polari...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM13184((2S)-2-amino-N-[4-(4-chloro-3-methylphenyl)-1,3-th...)
Affinity DataKd:  3.00E+4nMpH: 7.4 T: 2°CAssay Description:A fluorescence polarization anisotropy (FPA) competition assay was used to determine the affinities of compounds to BIR3 protein. Fluorescence polari...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM17338((2S)-2-{[(2S)-1-({2-[(1S)-1-aminoethyl]-1,3-oxazol...)
Affinity DataKd:  3.00E+4nMpH: 7.0 T: 2°CAssay Description:AVPC-badan can be displaced from the binding pocket of the protein by test compounds. As the dye is displaced from the binding pocket, the emission i...More data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM13192((2S)-2-amino-N-[5-benzyl-4-(3-benzylphenyl)-1,3-th...)
Affinity DataKd: >1.00E+5nMAssay Description:A fluorescence polarization anisotropy (FPA) competition assay was used to determine the affinities of compounds to BIR3 protein. Fluorescence polari...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM17339((2S)-2-{[(2S)-1-({2-[(1S)-1-aminoethyl]-1,3-oxazol...)
Affinity DataKd:  1.20E+5nMpH: 7.0 T: 2°CAssay Description:AVPC-badan can be displaced from the binding pocket of the protein by test compounds. As the dye is displaced from the binding pocket, the emission i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM17340((2S,3R)-2-{[(2S)-1-({2-[(1S)-1-aminoethyl]-1,3-oxa...)
Affinity DataKd:  3.00E+5nMpH: 7.0 T: 2°CAssay Description:AVPC-badan can be displaced from the binding pocket of the protein by test compounds. As the dye is displaced from the binding pocket, the emission i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed