Affinity DataKd: 0.0400nMAssay Description:Tested for dissociation constant at V1a receptor of rat liver membraneMore data for this Ligand-Target Pair
Affinity DataKd: 0.0540nMAssay Description:Tested for dissociation constant at V1a receptor of rat liver membraneMore data for this Ligand-Target Pair
Affinity DataKd: 0.150nMAssay Description:Tested for dissociation constant at V1a receptor of rat liver membraneMore data for this Ligand-Target Pair
Affinity DataKd: 0.180nMAssay Description:Binding potency against Vasopressin V1 receptor in rat liver cells.More data for this Ligand-Target Pair
Affinity DataKd: 0.180nMAssay Description:Binding potency against Vasopressin V1 receptor in rat liver cells.More data for this Ligand-Target Pair
Affinity DataKd: 0.182nMAssay Description:Binding potency against Vasopressin V1 receptor in rat liver cells.More data for this Ligand-Target Pair
Affinity DataKd: 0.182nMAssay Description:Negative log of Kd for Vasopressin V1 receptorMore data for this Ligand-Target Pair
Affinity DataKd: 0.190nMAssay Description:Tested for dissociation constant at V1a receptor of rat liver membraneMore data for this Ligand-Target Pair
Affinity DataKd: 0.320nMAssay Description:Binding affinity to human V1A receptor expressed in CHO cells after 4 hrs by RP-LC-ICPMS analysisMore data for this Ligand-Target Pair
Affinity DataKd: 0.330nMAssay Description:Binding potency against Vasopressin V1 receptor in rat liver cells.More data for this Ligand-Target Pair
Affinity DataKd: 0.330nMAssay Description:Binding potency against Vasopressin V1 receptor in rat liver cells.More data for this Ligand-Target Pair
Affinity DataKd: 0.331nMAssay Description:Binding potency against Vasopressin V1 receptor in rat liver cells.More data for this Ligand-Target Pair
Affinity DataKd: 0.331nMAssay Description:Negative log of Kd for Vasopressin V1 receptorMore data for this Ligand-Target Pair
Affinity DataKd: 0.450nMAssay Description:Binding affinity to human V1A receptor expressed in CHO cells after 4 hrs by RP-LC-ICPMS analysisMore data for this Ligand-Target Pair
Affinity DataKd: 0.480nMAssay Description:Inhibition of the 3 nM VP stimulation of phospholipase-C in cultured WRK cells was used as a V1-mediated assayMore data for this Ligand-Target Pair
Affinity DataKd: 0.600nMAssay Description:Binding affinity to human V1A receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKd: 0.600nMAssay Description:Binding potency against Vasopressin V1 receptor in rat liver cells.More data for this Ligand-Target Pair
Affinity DataKd: 0.603nMAssay Description:Negative log of Kd for Vasopressin V1 receptorMore data for this Ligand-Target Pair
Affinity DataKd: 0.640nMAssay Description:Binding potency against V1 receptor in rat liver cellsMore data for this Ligand-Target Pair
Affinity DataKd: 0.646nMAssay Description:Negative log of Kd for Vasopressin V1 receptorMore data for this Ligand-Target Pair
Affinity DataKd: 0.990nMAssay Description:Binding affinity to human V1A receptor expressed in CHO cells after 4 hrs by RP-LC-ICPMS analysisMore data for this Ligand-Target Pair
Affinity DataKd: 1.70nMAssay Description:Negative log of Kd for Vasopressin V1 receptorMore data for this Ligand-Target Pair
Affinity DataKd: 1.80nMAssay Description:Negative log of Kd for Vasopressin V1 receptorMore data for this Ligand-Target Pair
Affinity DataKd: 1.80nMAssay Description:Binding potency against V1 receptor in rat liver cellsMore data for this Ligand-Target Pair
Affinity DataKd: 1.80nMAssay Description:Negative log of Kd for Vasopressin V1 receptorMore data for this Ligand-Target Pair
Affinity DataKd: 2.40nMAssay Description:Compound was evaluated for the anti-vasopressor activity at V1a receptor. .More data for this Ligand-Target Pair
Affinity DataKd: 2.60nMAssay Description:Negative log of Kd for Vasopressin V1 receptorMore data for this Ligand-Target Pair
Affinity DataKd: 2.60nMAssay Description:Binding potency against Vasopressin V1 receptor in rat liver cells.More data for this Ligand-Target Pair
Affinity DataKd: 2.60nMAssay Description:Negative log of Kd for Vasopressin V1 receptorMore data for this Ligand-Target Pair
Affinity DataKd: 2.60nMAssay Description:Negative log of Kd for Vasopressin V1 receptorMore data for this Ligand-Target Pair
Affinity DataKd: 2.63nMAssay Description:Negative log of Kd for Vasopressin V1 receptorMore data for this Ligand-Target Pair
Affinity DataKd: 2.64nMAssay Description:Binding potency against Vasopressin V1 receptor in rat liver cells.More data for this Ligand-Target Pair
Affinity DataKd: 3.20nMAssay Description:Binding potency against Vasopressin V1 receptor in rat liver cells.More data for this Ligand-Target Pair
Affinity DataKd: 3.20nMAssay Description:Negative log of Kd for Vasopressin V1 receptorMore data for this Ligand-Target Pair
Affinity DataKd: 4.90nMAssay Description:Binding potency against Vasopressin V1 receptor in rat liver cells.More data for this Ligand-Target Pair
Affinity DataKd: 5nMAssay Description:Binding potency against Vasopressin V1 receptor in rat liver cells.More data for this Ligand-Target Pair
Affinity DataKd: 6.03nMAssay Description:Anti-vasopressor activity at V1a receptor More data for this Ligand-Target Pair
Affinity DataKd: 6.92nMAssay Description:Anti-vasopressor activity at V1a receptor More data for this Ligand-Target Pair
Affinity DataKd: 8.71nMAssay Description:Anti-vasopressor activity at V1a receptor More data for this Ligand-Target Pair
Affinity DataKd: 11.0nMAssay Description:Anti-vasopressor activity at V1a receptorMore data for this Ligand-Target Pair
Affinity DataKd: 13.5nMAssay Description:Anti-vasopressor activity at V1a receptor More data for this Ligand-Target Pair
Affinity DataKd: 16nMAssay Description:Binding potency against Vasopressin V1 receptor in rat liver cells.More data for this Ligand-Target Pair
Affinity DataKd: 16nMAssay Description:Negative log of Kd for Vasopressin V1 receptorMore data for this Ligand-Target Pair
Affinity DataKd: 20nMAssay Description:Binding affinity to V1aR (unknown origin) expressed in HEK293 cells by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKd: 27nMAssay Description:Binding potency against Vasopressin V1 receptor in rat liver cells.More data for this Ligand-Target Pair
Affinity DataKd: 27.5nMAssay Description:Anti-vasopressor activity at V1a receptor More data for this Ligand-Target Pair
Affinity DataKd: 27.5nMAssay Description:Anti-vasopressor activity at V1a receptorMore data for this Ligand-Target Pair
Affinity DataKd: 29.5nMAssay Description:Anti-vasopressor activity at V1a receptorMore data for this Ligand-Target Pair