Affinity DataKd: >0.00100nMAssay Description:Inhibition of [3H]-RA binding to retinoic acid receptor RAR alphaMore data for this Ligand-Target Pair
Affinity DataKd: >0.00100nMAssay Description:Inhibition of [3H]-RA binding to retinoic acid receptor RAR alphaMore data for this Ligand-Target Pair
Affinity DataKd: 0.300nMpH: 7.9 T: 2°CAssay Description:Recombinant RAR protein expressed in E. coli was used in the direct binding assay. The apparent dissociation constants (Kd) were determined by the ch...More data for this Ligand-Target Pair
Affinity DataKd: 0.400nMpH: 7.9 T: 2°CAssay Description:Recombinant RAR protein expressed in E. coli was used in the direct binding assay. The apparent dissociation constants (Kd) were determined by the ch...More data for this Ligand-Target Pair
Affinity DataKd: 0.400nMpH: 7.9 T: 2°CAssay Description:Recombinant RAR protein expressed in E. coli was used in the direct binding assay. The apparent dissociation constants (Kd) were determined by the ch...More data for this Ligand-Target Pair
Affinity DataKd: 1.5nMAssay Description:Inhibition of [3H]ATRA binding to baculovirus expressed RAR alpha receptorMore data for this Ligand-Target Pair
Affinity DataKd: 2nMAssay Description:Binding affinity fo retinoic acid receptor RAR alphaMore data for this Ligand-Target Pair
Affinity DataKd: 2nMAssay Description:Binding constant for baculovirus-expressed Retinoic acid receptor RAR alphaMore data for this Ligand-Target Pair
Affinity DataKd: 2.30nMAssay Description:Apparent binding constant against Retinoic acid receptor alpha in HeLa cell GAl-4 transactivation assayMore data for this Ligand-Target Pair
Affinity DataKd: 2.80nMAssay Description:Inhibition of [3H]ATRA binding to baculovirus expressed RAR alpha receptorMore data for this Ligand-Target Pair
Affinity DataKd: 3nMAssay Description:Effective concentration for retinoic acid receptor RAR alpha transcriptional activationMore data for this Ligand-Target Pair
Affinity DataKd: 3nMAssay Description:Binding affinity fo retinoic acid receptor RAR alphaMore data for this Ligand-Target Pair
Affinity DataKd: 4nMAssay Description:Binding affinity fo retinoic acid receptor RAR alphaMore data for this Ligand-Target Pair
Affinity DataKd: 4.40nMAssay Description:Binding affinity for baculovirus-expressed Retinoic acid receptor RAR alphaMore data for this Ligand-Target Pair
Affinity DataKd: 5.5nMAssay Description:Binding affinity of [3H]- RA to baculovirus expressed human RAR alphaMore data for this Ligand-Target Pair
Affinity DataKd: 5.70nMAssay Description:Inhibition of [3H]ATRA binding to baculovirus expressed RAR alpha receptorMore data for this Ligand-Target Pair
Affinity DataKd: 7nMAssay Description:Binding affinity for retinoic acid receptor RAR betaMore data for this Ligand-Target Pair
Affinity DataKd: 8.40nMAssay Description:Binding affinity for baculovirus-expressed Retinoic acid receptor RAR alphaMore data for this Ligand-Target Pair
Affinity DataKd: 11nMAssay Description:Compound was tested for binding affinity against retinoic acid receptor using 5 nM of [3H]-RA as a radioligand in baculovirus expressed receptorMore data for this Ligand-Target Pair
Affinity DataKd: 13nMAssay Description:Binding affinity of [3H]- RA to baculovirus expressed human RAR alphaMore data for this Ligand-Target Pair
Affinity DataKd: 13nMAssay Description:Antagonistic activity against RAR alpha in transcriptional activation assay with 32 nM TTNPBMore data for this Ligand-Target Pair
Affinity DataKd: 14nMAssay Description:Binding affinity fo retinoic acid receptor RAR alphaMore data for this Ligand-Target Pair
Affinity DataKd: 14nMAssay Description:Ability to inhibit TTNPB-induced transactivation at retinoic acid receptor betaMore data for this Ligand-Target Pair
Affinity DataKd: 14nMAssay Description:Binding affinity of [3H]- RA to baculovirus expressed human RAR alphaMore data for this Ligand-Target Pair
Affinity DataKd: 15nMAssay Description:Inhibition of [3H]-ATRA binding to human Retinoic acid receptor RAR alphaMore data for this Ligand-Target Pair
Affinity DataKd: 15nMAssay Description:Binding affinity for baculovirus-expressed Retinoic acid receptor RAR alphaMore data for this Ligand-Target Pair
Affinity DataKd: 15nMAssay Description:Inhibition of [3H]ATRA binding to baculovirus expressed RAR alpha receptorMore data for this Ligand-Target Pair
Affinity DataKd: 15nMAssay Description:Binding affinity of [3H]- RA to baculovirus expressed human RAR alphaMore data for this Ligand-Target Pair
Affinity DataKd: 15nMAssay Description:Inhibition of [3H]-RA binding to retinoic acid receptor RAR alphaMore data for this Ligand-Target Pair
Affinity DataKd: 15nMAssay Description:Ability to displace 3[H]-(all-E)-retinoic acid (5 nM) from alpha retinoic acid receptor (alpha RAR) using transactivation assayMore data for this Ligand-Target Pair
Affinity DataKd: 15nMAssay Description:Compound was tested for binding affinity against retinoic acid receptor using 5 nM of [3H]-RA as a radioligand in baculovirus expressed receptorMore data for this Ligand-Target Pair
Affinity DataKd: 15nMAssay Description:Inhibition of [3H]-ATRA binding to baculovirus expressed Retinoic acid receptor RAR alphaMore data for this Ligand-Target Pair
Affinity DataKd: 15nMAssay Description:Binding affinity for Retinoic acid receptor gammaMore data for this Ligand-Target Pair
Affinity DataKd: 16nMAssay Description:In vitro binding affinity for Retinoic acid receptor RAR alphaMore data for this Ligand-Target Pair
Affinity DataKd: 16nMAssay Description:Ability to displace 3[H]-(all-E)-retinoic acid (5 nM) from alpha retinoic acid receptor (alpha RAR) using transactivation assayMore data for this Ligand-Target Pair
Affinity DataKd: 17nMAssay Description:Binding affinity of [3H]- RA to baculovirus expressed human RAR alphaMore data for this Ligand-Target Pair
Affinity DataKd: 17nMAssay Description:Binding affinity towards retinoic acid receptor alpha was determined using [3H]-ATRA (5 nM) as radioligandMore data for this Ligand-Target Pair
Affinity DataKd: 27nMAssay Description:Inhibition of [3H]ATRA binding to baculovirus expressed RAR alpha receptorMore data for this Ligand-Target Pair
Affinity DataKd: >30nMAssay Description:Inhibition of [3H]-ATRA binding to baculovirus expressed retinoic acid receptor RAR-alphaMore data for this Ligand-Target Pair
Affinity DataKd: 32nMAssay Description:Inhibition of [3H]ATRA binding to baculovirus expressed RAR alpha receptorMore data for this Ligand-Target Pair
Affinity DataKd: 36nMAssay Description:Binding affinity towards retinoic acid receptor alpha was determined using [3H]-ATRA (5 nM) as radioligandMore data for this Ligand-Target Pair
Affinity DataKd: 36nMAssay Description:Binding affinity for Retinoic acid receptor gammaMore data for this Ligand-Target Pair
Affinity DataKd: 36nMAssay Description:Binding affinity fo retinoic acid receptor RAR alphaMore data for this Ligand-Target Pair
Affinity DataKd: 36nMAssay Description:Binding affinity for baculovirus-expressed Retinoic acid receptor RAR alphaMore data for this Ligand-Target Pair
Affinity DataKd: 38nMAssay Description:Ability to displace 3[H]-(all-E)-retinoic acid (5 nM) from alpha retinoic acid receptor (alpha RAR) using transactivation assayMore data for this Ligand-Target Pair
Affinity DataKd: 40nMAssay Description:Ability to displace 3[H]-(all-E)-retinoic acid (5 nM) from alpha retinoic acid receptor (alpha RAR) using transactivation assayMore data for this Ligand-Target Pair
Affinity DataKd: 44nMAssay Description:Ability to displace 3[H]-(all-E)-retinoic acid (5 nM) from alpha retinoic acid receptor (alpha RAR) using transactivation assayMore data for this Ligand-Target Pair
Affinity DataKd: 52nMAssay Description:Binding affinity of the compound was determined for Retinoic acid receptor alphaMore data for this Ligand-Target Pair
Affinity DataKd: 58nMAssay Description:Ability to displace 3[H]-(all-E)-retinoic acid (5 nM) from alpha retinoic acid receptor (alpha RAR) using transactivation assayMore data for this Ligand-Target Pair
Affinity DataKd: 58nMAssay Description:Binding affinity of the compound was determined for Retinoic acid receptor alphaMore data for this Ligand-Target Pair