Affinity DataKd: 0.0200nMAssay Description:Displacement of [TyrA14-125I]-human insulin from human insulin receptor isoform A expressed in baby hamster kidney cells after 2 days by gamma counti...More data for this Ligand-Target Pair
Affinity DataKd: 1.70nMAssay Description:Binding constant for INSR kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 2.40nMAssay Description:Binding constant for INSR kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 12nMAssay Description:Binding affinity to human InsR expressed in mouse IGF1R knockout MEF cells assessed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKd: 24nMAssay Description:Binding constant for INSR kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 72nMAssay Description:Binding affinity to human INSR by Ambit titration assayMore data for this Ligand-Target Pair
Affinity DataKd: 73nMAssay Description:Average Binding Constant for INSR; NA=Not Active at 10 uMMore data for this Ligand-Target Pair
Affinity DataKd: 110nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 110nMAssay Description:Binding constant for INSR kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 110nMAssay Description:Binding constant for INSR kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 180nMAssay Description:Average Binding Constant for INSR; NA=Not Active at 10 uMMore data for this Ligand-Target Pair
Affinity DataKd: 190nMAssay Description:Binding affinity to human INSR (997 to 1318 residues) expressed in mammalian expression system by kinome scan-based assayMore data for this Ligand-Target Pair
Affinity DataKd: 210nMAssay Description:Binding constant for INSR kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 330nMAssay Description:Binding constant for INSR kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 340nMAssay Description:Binding constant for INSR kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 400nMAssay Description:Binding constant for INSR kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 500nMAssay Description:Binding constant for INSR kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 500nMAssay Description:Binding affinity to INSRMore data for this Ligand-Target Pair
Affinity DataKd: 500nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 500nMAssay Description:Binding constant for INSR kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 506nMAssay Description:Binding affinity to human INSRMore data for this Ligand-Target Pair
Affinity DataKd: 630nMAssay Description:Binding constant for INSR kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 630nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 630nMAssay Description:Binding constant for INSR kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 850nMAssay Description:Binding constant for INSR kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 1.10E+3nMAssay Description:Binding constant for INSR kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 1.10E+3nMAssay Description:Binding affinity to INSRMore data for this Ligand-Target Pair
Affinity DataKd: 1.10E+3nMAssay Description:Binding constant for INSR kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 1.20E+3nMAssay Description:Binding constant for INSR kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 1.20E+3nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 1.20E+3nMAssay Description:Binding constant for INSR kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 1.69E+3nMAssay Description:Binding affinity to recombinant full-length N-terminal His-FLAG-GST-tagged INSR (unknown origin) (1005 to 1310 residues) expressed in baculovirus inf...More data for this Ligand-Target Pair
Affinity DataKd: 1.86E+3nMAssay Description:Binding affinity to recombinant full-length N-terminal His-FLAG-GST-tagged INSR (unknown origin) (1005 to 1310 residues) expressed in baculovirus inf...More data for this Ligand-Target Pair
Affinity DataKd: 2.20E+3nMAssay Description:Binding constant for INSR kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 2.30E+3nMAssay Description:Binding constant for INSR kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 3.00E+3nMAssay Description:Binding constant for INSR kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to INSRMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to INSRMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to INSRMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to INSRMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to INSRMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for INSR kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for INSR kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for INSR kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for INSR kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for INSR kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for INSR kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for INSR kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for INSR kinase domainMore data for this Ligand-Target Pair