Affinity DataKd: 1.30nMAssay Description:Compound was evaluated for Kd value against [3H]-SR- 48968 on the Tyr206Phe mutated human NK-2 receptorMore data for this Ligand-Target Pair
Affinity DataKd: 1.90nMAssay Description:Compound was evaluated for Kd value against [3H]-SR- 48968 on the Tyr206Phe mutated human NK-2 receptorMore data for this Ligand-Target Pair
Affinity DataKd: 2.10nMAssay Description:Compound was evaluated for Kd value against [125I]NKA on the Wild-type tachykinin receptor 2More data for this Ligand-Target Pair
Affinity DataKd: 2.70nMAssay Description:Compound was evaluated for Kd value against [125I]NKA on the Wild-type tachykinin receptor 2More data for this Ligand-Target Pair
Affinity DataKd: 3.10nMAssay Description:Compound was evaluated for Kd value against [125I]-NKA on the Tyr206Phe mutated human NK-2 receptorMore data for this Ligand-Target Pair
Affinity DataKd: 3.60nMAssay Description:Compound was evaluated for Kd value against [125I]NKA on the Tyr206Phe mutated human NK-2 receptorMore data for this Ligand-Target Pair
Affinity DataKd: 4.40nMAssay Description:Compound was evaluated for Kd value against [3H]-SR- 48968 on the Wild-type tachykinin receptor 2More data for this Ligand-Target Pair
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Affinity DataKd: 7.94nMAssay Description:Inhibition of eledoisin binding to NK-2 receptor in rat vas deferensMore data for this Ligand-Target Pair
Affinity DataKd: 10nMAssay Description:Compound was evaluated for Kd value against [3H]-SR- 48968 on the Wild-type tachykinin receptor 2More data for this Ligand-Target Pair
Affinity DataKd: 26nMAssay Description:Compound was evaluated for Kd value against [125I]NKA on the Tyr266Phe mutated human NK-2 receptorMore data for this Ligand-Target Pair
Affinity DataKd: 34nMAssay Description:Compound was evaluated for Kd value against [125I]NKA on the Tyr266Phe mutated human NK-2 receptorMore data for this Ligand-Target Pair
Affinity DataKd: 48nMAssay Description:Compound was evaluated for Kd value against [3H]-SR- 48968 on the Tyr266Phe mutated human NK-2 receptorMore data for this Ligand-Target Pair
Affinity DataKd: 48nMAssay Description:Compound was evaluated for Kd value against [3H]-SR- 48968 on the Tyr266Phe mutated human NK-2 receptorMore data for this Ligand-Target Pair
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Affinity DataKd: 200nMAssay Description:Inhibition of eledoisin binding to NK-2 receptor in rat vas deferensMore data for this Ligand-Target Pair
Affinity DataKd: 208nMAssay Description:Compound was evaluated for Kd value against [3H]-SR- 48968 on the Phe270Ala mutated human NK-2 receptorMore data for this Ligand-Target Pair
Affinity DataKd: 291nMAssay Description:Compound was evaluated for Kd value against [3H]-SR- 48968 on the Phe270Ala mutated human NK-2 receptorMore data for this Ligand-Target Pair
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Affinity DataKd: 398nMAssay Description:Inhibition of eledoisin binding to NK-2 receptor in rat vas deferensMore data for this Ligand-Target Pair
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Affinity DataKd: 631nMAssay Description:Inhibition of eledoisin binding to NK-2 receptor in rat vas deferensMore data for this Ligand-Target Pair
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Affinity DataKd: 1.00E+3nMAssay Description:Inhibition of eledoisin binding to NK-2 receptor in rat vas deferensMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+3nMAssay Description:Compound was evaluated for Kd value against [3H]-SR- 48968 on the Tyr206Ala mutated human NK-2 receptorMore data for this Ligand-Target Pair
Affinity DataKd: 1.96E+3nMAssay Description:Compound was evaluated for Kd value against [3H]-SR- 48968 on the Tyr206Ala mutated human NK-2 receptorMore data for this Ligand-Target Pair
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Affinity DataKd: 2.51E+3nMAssay Description:Inhibition of eledoisin binding to NK-2 receptor in rat vas deferensMore data for this Ligand-Target Pair
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Affinity DataKd: 7.94E+3nMAssay Description:Inhibition of eledoisin binding to NK-2 receptor in rat vas deferensMore data for this Ligand-Target Pair
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Affinity DataKd: 1.00E+4nMAssay Description:Inhibition of eledoisin binding to NK-2 receptor in rat vas deferensMore data for this Ligand-Target Pair
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Affinity DataKd: 1.00E+4nMAssay Description:Inhibition of eledoisin binding to NK-2 receptor in rat vas deferensMore data for this Ligand-Target Pair
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Affinity DataKd: 1.00E+4nMAssay Description:Inhibition of eledoisin binding to NK-2 receptor in rat vas deferensMore data for this Ligand-Target Pair
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Affinity DataKd: 1.26E+4nMAssay Description:Inhibition of eledoisin binding to NK-2 receptor in rat vas deferensMore data for this Ligand-Target Pair
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Affinity DataKd: 1.58E+4nMAssay Description:Inhibition of eledoisin binding to NK-2 receptor in rat vas deferensMore data for this Ligand-Target Pair
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Affinity DataKd: 1.58E+4nMAssay Description:Inhibition of eledoisin binding to NK-2 receptor in rat vas deferensMore data for this Ligand-Target Pair
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Affinity DataKd: 2.00E+4nMAssay Description:Inhibition of eledoisin binding to NK-2 receptor in rat vas deferensMore data for this Ligand-Target Pair
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Affinity DataKd: 2.51E+4nMAssay Description:Inhibition of eledoisin binding to NK-2 receptor in rat vas deferensMore data for this Ligand-Target Pair