Compile Data Set for Download or QSAR
maximum 50k data
Found 26 of kd data for polymerid = 49000976,49000978,49000979,49000981,49000983,49000985,50000466,50000724,50000725,50000731
TargetP2X purinoceptor 7(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50126720((S)-4-(2-(N-methylisoquinoline-5-sulfonamido)-3-ox...)
Affinity DataKd:  3.60nMAssay Description:Equilibrium constant for P2X purinoceptor 7 expressed in HEK 293 cells at 1 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50126720((S)-4-(2-(N-methylisoquinoline-5-sulfonamido)-3-ox...)
Affinity DataKd:  3.60nMAssay Description:Maximum binding affinity towards P2X purinoceptor 7 expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50409686(CHEMBL173068)
Affinity DataKd:  77.6nMAssay Description:pA2 value was evaluated against P2Y purinoceptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
University Park Nottingham

Curated by ChEMBL
LigandPNGBDBM50271557(CHEMBL4127889)
Affinity DataKd:  89nMAssay Description:Binding affinity to recombinant human N-terminal NLuc-tagged P2Y2R expressed in human 1321N1 cells incubated for 1 hr in presence of AR-C118925 by fu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50118229(CHEMBL129841 | MRS 2179)
Affinity DataKd:  109nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
University Park Nottingham

Curated by ChEMBL
LigandPNGBDBM50271587(CHEMBL4128532)
Affinity DataKd:  129nMAssay Description:Binding affinity to recombinant human N-terminal NLuc-tagged P2Y2R expressed in human 1321N1 cells incubated for 1 hr in presence of AR-C118925 by fu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50118229(CHEMBL129841 | MRS 2179)
Affinity DataKd:  282nMAssay Description:pA2 value was evaluated against P2Y purinoceptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
University Park Nottingham

Curated by ChEMBL
LigandPNGBDBM50271589(CHEMBL4128024)
Affinity DataKd:  295nMAssay Description:Binding affinity to recombinant human N-terminal NLuc-tagged P2Y2R expressed in human 1321N1 cells incubated for 1 hr in presence of AR-C118925 by fu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
University Park Nottingham

Curated by ChEMBL
LigandPNGBDBM50271588(CHEMBL4126655)
Affinity DataKd:  479nMAssay Description:Binding affinity to recombinant human N-terminal NLuc-tagged P2Y2R expressed in human 1321N1 cells incubated for 1 hr in presence of AR-C118925 by fu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50586608(CHEMBL5083184)
Affinity DataKd:  710nMAssay Description:Binding affinity to human wild type P2X7R assessed as dissociation constant by microscale thermophoresis analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
University Park Nottingham

Curated by ChEMBL
LigandPNGBDBM50271560(CHEMBL4125853)
Affinity DataKd:  759nMAssay Description:Binding affinity to recombinant human N-terminal NLuc-tagged P2Y2R expressed in human 1321N1 cells incubated for 1 hr in presence of AR-C118925 by fu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 1(RAT)
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50118237(CHEMBL130059 | Uniblue A)
Affinity DataKd:  800nMAssay Description:Dissociation constant at P2X purinoceptor 1 from guinea pig taenia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
University Park Nottingham

Curated by ChEMBL
LigandPNGBDBM50271561(CHEMBL4125987)
Affinity DataKd:  851nMAssay Description:Binding affinity to recombinant human N-terminal NLuc-tagged P2Y2R expressed in human 1321N1 cells incubated for 1 hr in presence of AR-C118925 by fu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
University Park Nottingham

Curated by ChEMBL
LigandPNGBDBM50271586(CHEMBL4125833)
Affinity DataKd:  891nMAssay Description:Binding affinity to recombinant human N-terminal NLuc-tagged P2Y2R expressed in human 1321N1 cells incubated for 1 hr in presence of AR-C118925 by fu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50118211(Acid Blue 129 | CHEMBL133576 | cid_23675739 | sodi...)
Affinity DataKd:  1.40E+3nMAssay Description:Dissociative constant at P2Y purinoceptor 1 (P2Y1) from guinea pig taenia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 1(RAT)
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50118231(CHEMBL134193 | Cibachron Blue 3GA)
Affinity DataKd:  1.60E+3nMAssay Description:Dissociation constant of the copound at P2X purinoceptor 1 (P2X1) from rat vas deferens was reportedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
University Park Nottingham

Curated by ChEMBL
LigandPNGBDBM50271545(CHEMBL4127230)
Affinity DataKd:  1.66E+3nMAssay Description:Binding affinity to recombinant human N-terminal NLuc-tagged P2Y2R expressed in human 1321N1 cells incubated for 1 hr in presence of AR-C118925 by fu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
University Park Nottingham

Curated by ChEMBL
LigandPNGBDBM50271569(CHEMBL4128318)
Affinity DataKd:  2.14E+3nMAssay Description:Binding affinity to recombinant human N-terminal NLuc-tagged P2Y2R expressed in human 1321N1 cells incubated for 1 hr in presence of AR-C118925 by fu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
University Park Nottingham

Curated by ChEMBL
LigandPNGBDBM50271559(CHEMBL4126826)
Affinity DataKd:  2.75E+3nMAssay Description:Binding affinity to recombinant human N-terminal NLuc-tagged P2Y2R expressed in human 1321N1 cells incubated for 1 hr in presence of AR-C118925 by fu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50118231(CHEMBL134193 | Cibachron Blue 3GA)
Affinity DataKd:  2.90E+3nMAssay Description:The compound was evaluated for antagonistic activity at P2Y purinoceptor 1 (P2Y1) from guinea pig taenia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50118234(CHEMBL129904 | MRS 2160)
Affinity DataKd:  2.90E+3nMAssay Description:The compound was evaluated for antagonistic activity at P2Y purinoceptor 1 (P2Y1) from guinea pig taenia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
University Park Nottingham

Curated by ChEMBL
LigandPNGBDBM50271585(CHEMBL4129129)
Affinity DataKd:  4.17E+3nMAssay Description:Binding affinity to recombinant human N-terminal NLuc-tagged P2Y2R expressed in human 1321N1 cells incubated for 1 hr in presence of AR-C118925 by fu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
University Park Nottingham

Curated by ChEMBL
LigandPNGBDBM50271568(CHEMBL4129299)
Affinity DataKd:  5.13E+3nMAssay Description:Binding affinity to recombinant human N-terminal NLuc-tagged P2Y2R expressed in human 1321N1 cells incubated for 1 hr in presence of AR-C118925 by fu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
University Park Nottingham

Curated by ChEMBL
LigandPNGBDBM50271546(CHEMBL4129692)
Affinity DataKd:  1.23E+4nMAssay Description:Binding affinity to recombinant human N-terminal NLuc-tagged P2Y2R expressed in human 1321N1 cells incubated for 1 hr in presence of AR-C118925 by fu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 1(RAT)
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50118211(Acid Blue 129 | CHEMBL133576 | cid_23675739 | sodi...)
Affinity DataKd: >1.00E+5nMAssay Description:The compound was evaluated for antagonist activity against P2X purinoceptor 1 (P2X1) like receptor from rat vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50118237(CHEMBL130059 | Uniblue A)
Affinity DataKd: >1.00E+5nMAssay Description:Dissociation constant at P2Y purinoceptor 1 (P2Y1) from guinea pig taenia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed