Affinity DataKd: 0.190nMAssay Description:Binding constant for MET kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 0.200nMAssay Description:Binding affinity to MET (unknown origin)More data for this Ligand-Target Pair
Affinity DataKd: 0.210nMpH: 7.0 T: 2°CAssay Description:Met (h) is incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 .mu.M KKKSPGEYVNIEFG, 10 mM MgAcetate and [.gamma.-.sup.33P-ATP] (specific activity appr...More data for this Ligand-Target Pair
Affinity DataKd: 0.270nMAssay Description:Binding constant for MET kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 0.5nMpH: 7.0 T: 2°CAssay Description:Met (h) is incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 .mu.M KKKSPGEYVNIEFG, 10 mM MgAcetate and [.gamma.-.sup.33P-ATP] (specific activity appr...More data for this Ligand-Target Pair
Affinity DataKd: 0.550nMAssay Description:Binding constant for MET(M1250T) kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 0.600nMAssay Description:Binding affinity to MET (unknown origin) by isothermal titration calorimetryMore data for this Ligand-Target Pair
Affinity DataKd: 0.600nMAssay Description:Binding affinity to MET (unknown origin) by isothermal titration calorimetryMore data for this Ligand-Target Pair
Affinity DataKd: 0.640nMAssay Description:Binding constant for MET(M1250T) kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 0.820nMAssay Description:Binding constant for MET(M1250T) kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 0.820nMAssay Description:Binding constant for MET(Y1235D) kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 0.830nMAssay Description:Binding constant for MET(Y1235D) kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 0.900nMAssay Description:Binding affinity to MET (unknown origin) by isothermal titration calorimetryMore data for this Ligand-Target Pair
Affinity DataKd: 0.900nMAssay Description:Binding affinity to MET (unknown origin) by isothermal titration calorimetryMore data for this Ligand-Target Pair
Affinity DataKd: 1nMAssay Description:Binding constant for MET(M1250T) kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 1.40nMAssay Description:Binding constant for MET kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 1.5nMAssay Description:Binding constant for MET(Y1235D) kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 2nMAssay Description:Binding affinity to MET (unknown origin) by isothermal titration calorimetryMore data for this Ligand-Target Pair
Affinity DataKd: 2nMAssay Description:Binding affinity to MET (unknown origin) by isothermal titration calorimetryMore data for this Ligand-Target Pair
Affinity DataKd: 2.10nMAssay Description:Binding constant for MET kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 2.40nMpH: 7.0 T: 2°CAssay Description:Met (h) is incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 .mu.M KKKSPGEYVNIEFG, 10 mM MgAcetate and [.gamma.-.sup.33P-ATP] (specific activity appr...More data for this Ligand-Target Pair
Affinity DataKd: 3.20nMAssay Description:Binding affinity to phosphorylated c-MET kinase domain (unknown origin)More data for this Ligand-Target Pair
Affinity DataKd: 3.90nMAssay Description:Binding constant for MET(M1250T) kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 4nMAssay Description:Binding affinity to human recombinant His6-tagged phosphorylated c-Met cytosolic domainMore data for this Ligand-Target Pair
Affinity DataKd: 4.40nMAssay Description:Binding affinity to human phosphorylated c-METMore data for this Ligand-Target Pair
Affinity DataKd: 8.70nMAssay Description:Binding affinity to MET (unknown origin) by isothermal titration calorimetryMore data for this Ligand-Target Pair
Affinity DataKd: 8.70nMAssay Description:Binding affinity to MET (unknown origin) by isothermal titration calorimetryMore data for this Ligand-Target Pair
Affinity DataKd: 10nMAssay Description:Binding affinity to unphosphorylated c-MET kinase domain (unknown origin)More data for this Ligand-Target Pair
Affinity DataKd: 12nMAssay Description:Binding affinity to MET (unknown origin) by isothermal titration calorimetryMore data for this Ligand-Target Pair
Affinity DataKd: 12nMAssay Description:Binding affinity to MET (unknown origin) by isothermal titration calorimetryMore data for this Ligand-Target Pair
Affinity DataKd: 25nMAssay Description:Binding affinity to human recombinant His6-tagged unphosphorylated c-Met cytosolic domainMore data for this Ligand-Target Pair
Affinity DataKd: 27.2nMAssay Description:Binding affinity to human unphosphorylated c-METMore data for this Ligand-Target Pair
Affinity DataKd: 38nMAssay Description:Binding affinity to MET (unknown origin)More data for this Ligand-Target Pair
Affinity DataKd: 41nMAssay Description:Binding constant for MET(Y1235D) kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 64nMAssay Description:Binding constant for MET(M1250T) kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 65nMAssay Description:Binding affinity to MET (unknown origin) after 1 hrMore data for this Ligand-Target Pair
Affinity DataKd: 79nMAssay Description:Binding affinity to human METMore data for this Ligand-Target Pair
Affinity DataKd: 79nMAssay Description:Binding affinity to human METMore data for this Ligand-Target Pair
Affinity DataKd: 93nMAssay Description:Binding constant for MET(M1250T) kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 130nMAssay Description:Binding constant for MET(M1250T) kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 140nMAssay Description:Binding constant for MET(Y1235D) kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 150nMAssay Description:Binding affinity to MET (unknown origin) after 1 hrMore data for this Ligand-Target Pair
Affinity DataKd: 170nMAssay Description:Binding constant for MET kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 170nMAssay Description:Binding constant for MET kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 180nMAssay Description:Binding constant for MET(Y1235D) kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 190nMAssay Description:Binding constant for MET kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 190nMAssay Description:Binding constant for MET kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 190nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 200nMpH: 7.0 T: 2°CAssay Description:Met (h) is incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 .mu.M KKKSPGEYVNIEFG, 10 mM MgAcetate and [.gamma.-.sup.33P-ATP] (specific activity appr...More data for this Ligand-Target Pair
Affinity DataKd: 200nMAssay Description:Binding constant for MET kinase domainMore data for this Ligand-Target Pair