Affinity DataKd: 0.220nMAssay Description:Binding affinity to DNA-tagged recombinant human BIKE (34 to 329 residues) expressed in bacterial expression system by KINOMEscan assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKd: 2.20nMAssay Description:Binding constant for BIKE kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 3.70nMAssay Description:Average Binding Constant for BIKE; NA=Not Active at 10 uMMore data for this Ligand-Target Pair
Affinity DataKd: 3.80nMAssay Description:Binding affinity to BIKE (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKd: 5.5nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 5.5nMAssay Description:Binding constant for BIKE kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 5.5nMAssay Description:Binding affinity to BIKEMore data for this Ligand-Target Pair
Affinity DataKd: 5.5nMAssay Description:Binding constant for BIKE kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 5.60nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 5.60nMAssay Description:Binding constant for BIKE kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 5.60nMAssay Description:Binding constant for BIKE kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 7.5nMAssay Description:Binding affinity to DNA-tagged recombinant human BIKE (34 to 329 residues) expressed in bacterial expression system by KINOMEscan assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKd: 9.60nMAssay Description:Binding constant for BIKE kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 16nMAssay Description:Binding affinity to BIKEMore data for this Ligand-Target Pair
Affinity DataKd: 16nMAssay Description:Binding constant for BIKE kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 19nMAssay Description:Binding affinity to recombinant full-length N-terminal His-FLAG-GST-tagged BMP2K (unknown origin) expressed in baculovirus infected Sf9 insect cells ...More data for this Ligand-Target Pair
Affinity DataKd: 20nMAssay Description:Binding affinity to BIKE (unknown origin)More data for this Ligand-Target Pair
Affinity DataKd: 20nMAssay Description:Binding affinity to BIKE (unknown origin)More data for this Ligand-Target Pair
Affinity DataKd: 24nMAssay Description:Binding affinity to recombinant full-length N-terminal His-FLAG-GST-tagged BMP2K (unknown origin) expressed in baculovirus infected Sf9 insect cells ...More data for this Ligand-Target Pair
Affinity DataKd: 25nMAssay Description:Average Binding Constant for BIKE; NA=Not Active at 10 uMMore data for this Ligand-Target Pair
Affinity DataKd: 27nMAssay Description:Binding constant for BIKE kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 27nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 27nMAssay Description:Binding constant for BIKE kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 32nMAssay Description:Binding constant for BIKE kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 38nMAssay Description:Average Binding Constant for BIKE; NA=Not Active at 10 uMMore data for this Ligand-Target Pair
Affinity DataKd: 47nMAssay Description:Binding constant for BIKE kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 54nMAssay Description:Binding constant for BIKE kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 54nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 54nMAssay Description:Binding constant for BIKE kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 65nMAssay Description:Binding constant for BIKE kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 65nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 65nMAssay Description:Binding constant for BIKE kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 120nMAssay Description:Binding constant for BIKE kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 140nMAssay Description:Binding constant for BIKE kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 180nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 180nMAssay Description:Binding constant for BIKE kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 210nMAssay Description:Binding constant for BIKE kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 220nMAssay Description:Binding affinity to BIKEMore data for this Ligand-Target Pair
Affinity DataKd: 220nMAssay Description:Binding constant for BIKE kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 220nMAssay Description:Binding constant for BIKE kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 220nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 350nMAssay Description:Binding constant for BIKE kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 430nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 430nMAssay Description:Binding constant for BIKE kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 430nMAssay Description:Binding constant for BIKE kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 470nMAssay Description:Binding constant for BIKE kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 540nMAssay Description:Average Binding Constant for BIKE; NA=Not Active at 10 uMMore data for this Ligand-Target Pair
Affinity DataKd: 640nMAssay Description:Binding constant for BIKE kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 740nMAssay Description:Binding constant for BIKE kinase domainMore data for this Ligand-Target Pair