Compile Data Set for Download or QSAR
maximum 50k data
Found 61 of ki data for polymerid = 2433,4995,9427,9934
TargetMaltase-glucoamylase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291029((2R,3R,4R,5S)-2-Hydroxymethyl-1-((E)-3-trimethylsi...)
Affinity DataKi:  2.30nMAssay Description:In vitro inhibition constant against rat small intestinal glucoamylaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMaltase-glucoamylase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291026((2R,3R,4R,5S)-1-[(E)-3-(Dimethyl-phenyl-silanyl)-a...)
Affinity DataKi:  4nMAssay Description:In vitro inhibition constant against rat small intestinal glucoamylaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMaltase-glucoamylase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291020((2R,3R,4R,5S)-1-[3-(Dimethyl-phenyl-silanyl)-propy...)
Affinity DataKi:  10nMAssay Description:In vitro inhibition constant against rat small intestinal glucoamylaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMaltase-glucoamylase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50327503((1R,2R,3S,4S)-3,4-dihydroxy-2-(hydroxymethyl)-1-((...)
Affinity DataKi:  15nMAssay Description:Inhibition of human recombinant N-terminal domain of maltase-glucoamylase after 60 mins by glucose oxidase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMaltase-glucoamylase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50330961((2R,3S,4S)-1-((2S,3S,4R,5R,6S)-2,3,4,5,6,7-hexahyd...)
Affinity DataKi:  20nMAssay Description:Inhibition of human recombinant N-terminal subunit of maltase-glucoamylase after 60 mins by glucose oxidase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMaltase-glucoamylase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291027((2R,3R,4R,5S)-2-Hydroxymethyl-1-(4-trimethylsilany...)
Affinity DataKi:  28nMAssay Description:In vitro inhibition constant against rat small intestinal glucoamylaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMaltase-glucoamylase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50330954(CHEMBL1276973 | de-O-sulfonated kotalanol)
Affinity DataKi:  30nMAssay Description:Inhibition of human recombinant N-terminal subunit of maltase-glucoamylase after 60 mins by glucose oxidase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMaltase-glucoamylase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50327502((1R,2R,3S,4S)-3,4-dihydroxy-2-(hydroxymethyl)-1-((...)
Affinity DataKi:  43nMAssay Description:Inhibition of human recombinant N-terminal domain of maltase-glucoamylase after 60 mins by glucose oxidase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMaltase-glucoamylase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50327502((1R,2R,3S,4S)-3,4-dihydroxy-2-(hydroxymethyl)-1-((...)
Affinity DataKi:  43nMAssay Description:Inhibition of human N-terminal maltase-glucoamylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMaltase-glucoamylase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291031((2R,3R,4R,5S)-2-Hydroxymethyl-1-(3-trimethylsilany...)
Affinity DataKi:  50nMAssay Description:In vitro inhibition constant against rat small intestinal glucoamylaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMaltase-glucoamylase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50330960((2R,3R,4R)-1-((2R,3R,4S,5R,6S)-2,3,4,5,6,7-hexahyd...)
Affinity DataKi:  60nMAssay Description:Inhibition of human recombinant N-terminal subunit of maltase-glucoamylase after 60 mins by glucose oxidase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMaltase-glucoamylase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291034((2R,3R,4R,5S)-2-Hydroxymethyl-1-(5-trimethylsilany...)
Affinity DataKi:  70nMAssay Description:In vitro inhibition constant against rat small intestinal glucoamylaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMaltase-glucoamylase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50330959(CHEMBL1277153)
Affinity DataKi:  80nMAssay Description:Inhibition of human recombinant N-terminal subunit of maltase-glucoamylase after 60 mins by glucose oxidase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMaltase-glucoamylase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291023((2R,3R,4R,5S)-1-[(E)-3-(tert-Butyl-dimethyl-silany...)
Affinity DataKi:  87nMAssay Description:In vitro inhibition constant against rat small intestinal glucoamylaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMaltase-glucoamylase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50316180((1S,2R,3S,4S)-1-{(1S)-2-[(2R,3S,4S)-3,4-dihydroxy-...)
Affinity DataKi:  100nMAssay Description:Inhibition of recombinant human maltase glucoamylase N-terminal catalytic domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMaltase-glucoamylase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291021((2R,3R,4R,5S)-2-Hydroxymethyl-1-(4-trimethylsilany...)
Affinity DataKi:  120nMAssay Description:In vitro inhibition constant against rat small intestinal glucoamylaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMaltase-glucoamylase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50316181((1S,2R,3S,4R)-1-{(1S)-2-[(2R,3S,4S)-3,4-dihydroxy-...)
Affinity DataKi:  130nMAssay Description:Inhibition of recombinant human maltase glucoamylase N-terminal catalytic domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMaltase-glucoamylase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50327501(CHEMBL1258528 | ponkoranol)
Affinity DataKi:  170nMAssay Description:Inhibition of human recombinant N-terminal domain of maltase-glucoamylase after 60 mins by glucose oxidase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMaltase-glucoamylase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50316179((1S,2R,3R,4S)-1-{(1S)-2-[(2R,3S,4S)-3,4-dihydroxy-...)
Affinity DataKi:  190nMAssay Description:Inhibition of recombinant human maltase glucoamylase N-terminal catalytic domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMaltase-glucoamylase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50316179((1S,2R,3R,4S)-1-{(1S)-2-[(2R,3S,4S)-3,4-dihydroxy-...)
Affinity DataKi:  190nMAssay Description:Inhibition of human recombinant N-terminal subunit of maltase-glucoamylase after 60 mins by glucose oxidase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMaltase-glucoamylase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50330955((1S,2S)-3-[(2R,3S,4S)-3,4-dihydroxy-2-(hydroxymeth...)
Affinity DataKi:  190nMAssay Description:Inhibition of recombinant human maltase-glucoamylase using p-nitrophenyl-alpha-D-glucopyranoside as substrate incubated for 35 mins by microtiter pla...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMaltase-glucoamylase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50316178(1,4-Dideoxy-1,4-[[2S,3S,4R,5R,6R-2,4,5,6,7-pentahy...)
Affinity DataKi:  200nMAssay Description:Inhibition of recombinant human maltase glucoamylase N-terminal catalytic domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMaltase-glucoamylase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50408432(CHEMBL2115215)
Affinity DataKi:  450nMAssay Description:Compound was tested for binding affinity against alpha-glucosidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMaltase-glucoamylase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50327504(1,4-Dideoxy-1,4-[[2S,3S,4R,5S]-2,4,5,6-tetrahydrox...)
Affinity DataKi:  500nMAssay Description:Inhibition of human recombinant N-terminal maltase-glucoamylase by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMaltase-glucoamylase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50327504(1,4-Dideoxy-1,4-[[2S,3S,4R,5S]-2,4,5,6-tetrahydrox...)
Affinity DataKi:  500nMAssay Description:Inhibition of human N-terminal maltase-glucoamylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMaltase-glucoamylase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50327504(1,4-Dideoxy-1,4-[[2S,3S,4R,5S]-2,4,5,6-tetrahydrox...)
Affinity DataKi:  500nMAssay Description:Inhibition of human recombinant N-terminal domain of maltase-glucoamylase after 60 mins by glucose oxidase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMaltase-glucoamylase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291028((2R,3R,4R,5S)-1-(Dimethyl-propyl-silanylmethyl)-2-...)
Affinity DataKi:  900nMAssay Description:In vitro inhibition constant against rat small intestinal glucoamylaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMaltase-glucoamylase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50242271((2R,3R,4R,5S)-1-(2-hydroxyethyl)-2-(hydroxymethyl)...)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of human recombinant N-terminal subunit of maltase-glucoamylase after 60 mins by glucose oxidase assayMore data for this Ligand-Target Pair
TargetMaltase-glucoamylase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291032((2R,3R,4R,5S)-2-Hydroxymethyl-1-(3-trimethylsilany...)
Affinity DataKi:  1.00E+3nMAssay Description:In vitro inhibition constant against rat small intestinal glucoamylaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMaltase-glucoamylase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50330955((1S,2S)-3-[(2R,3S,4S)-3,4-dihydroxy-2-(hydroxymeth...)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of human recombinant N-terminal subunit of maltase-glucoamylase after 60 mins by glucose oxidase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMaltase-glucoamylase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50330957(7'-[(1,5-Dideoxy-1,5-imino-D-glucitol)-5-N-ammoniu...)
Affinity DataKi:  1.40E+3nMAssay Description:Inhibition of human recombinant N-terminal subunit of maltase-glucoamylase after 60 mins by glucose oxidase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMaltase-glucoamylase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50486898(Broussonol E | CHEBI:66727)
Affinity DataKi:  2.30E+3nMAssay Description:Mixed type inhibition of alpha-glucosidase (unknown origin) using p-nitrophenyl-alpha-D glucopyranoside as substrate incubated for 30 mins by Linewea...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMaltase-glucoamylase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50330956(7'-[(1,5-Dideoxy-1,5-imino-D-glucitol)-5-N-ammoniu...)
Affinity DataKi:  2.30E+3nMAssay Description:Inhibition of human recombinant N-terminal subunit of maltase-glucoamylase after 60 mins by glucose oxidase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMaltase-glucoamylase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291022((2R,3R,4R,5S)-2-Hydroxymethyl-1-trimethylsilanylme...)
Affinity DataKi:  2.50E+3nMAssay Description:In vitro inhibition constant against rat small intestinal glucoamylaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMaltase-glucoamylase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291033((2R,3R,4R,5S)-1-[(Dimethyl-phenyl-silanyl)-methyl]...)
Affinity DataKi:  2.60E+3nMAssay Description:In vitro inhibition constant against rat small intestinal glucoamylaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-glucosidase MAL12(Saccharomyces cerevisiae)
Gyeongsang National University

LigandPNGBDBM84968(Urea derivative, 12)
Affinity DataKi:  3.20E+3nM IC50:  8.40E+3nMAssay Description:All enzymatic activities were determined by using the appropriate substrate (p-nitrophenyl-alpha-D-glucopyranoside, p-nitrophenyl-beta-D-gulcopyranos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMaltase-glucoamylase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50550994(CHEMBL4760193)
Affinity DataKi:  4.20E+3nMAssay Description:Mixed type inhibition of alpha-glucosidase (unknown origin) using p-nitrophenyl-alpha-D glucopyranoside as substrate incubated for 30 mins by Linewea...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-glucosidase MAL12(Saccharomyces cerevisiae)
Gyeongsang National University

LigandPNGBDBM84969(Urea derivative, 13)
Affinity DataKi:  4.60E+3nM IC50:  1.43E+4nMAssay Description:All enzymatic activities were determined by using the appropriate substrate (p-nitrophenyl-alpha-D-glucopyranoside, p-nitrophenyl-beta-D-gulcopyranos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMaltase-glucoamylase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50121025((E)-1-[2,4-Dihydroxy-5-(3-methyl-but-2-enyl)-pheny...)
Affinity DataKi:  5.30E+3nMAssay Description:Non-competitive inhibition of alpha-glucosidase (unknown origin) using p-nitrophenyl-alpha-D glucopyranoside as substrate incubated for 30 mins by Li...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMaltase-glucoamylase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50549692(CHEMBL4749306)
Affinity DataKi:  6.00E+3nMAssay Description:Inhibition of recombinant human maltase-glucoamylase using p-nitrophenyl-alpha-D-glucopyranoside as substrate incubated for 35 mins by microtiter pla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMaltase-glucoamylase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50408431(CHEMBL2114210)
Affinity DataKi:  6.20E+3nMAssay Description:Compound was tested for binding affinity against alpha-glucosidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMaltase-glucoamylase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50065255((R)-2,6-Bis-hydroxymethyl-piperidine-3,4,5-triol |...)
Affinity DataKi:  6.90E+3nMAssay Description:Compound was tested for binding affinity against alpha-glucosidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-glucosidase MAL12(Saccharomyces cerevisiae)
Gyeongsang National University

LigandPNGBDBM84967(Urea derivative, 11)
Affinity DataKi:  7.20E+3nM IC50:  1.98E+4nMAssay Description:All enzymatic activities were determined by using the appropriate substrate (p-nitrophenyl-alpha-D-glucopyranoside, p-nitrophenyl-beta-D-gulcopyranos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-glucosidase MAL12(Saccharomyces cerevisiae)
Gyeongsang National University

LigandPNGBDBM84972(Urea derivative, 16)
Affinity DataKi:  9.40E+3nM IC50:  1.85E+4nMAssay Description:All enzymatic activities were determined by using the appropriate substrate (p-nitrophenyl-alpha-D-glucopyranoside, p-nitrophenyl-beta-D-gulcopyranos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMaltase-glucoamylase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291024((2R,3R,4R,5S)-2-Hydroxymethyl-1-(2-trimethylsilany...)
Affinity DataKi:  1.00E+4nMAssay Description:In vitro inhibition constant against rat small intestinal glucoamylaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMaltase-glucoamylase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM19459(5,7-dihydroxy-3-(4-hydroxyphenyl)-4H-chromen-4-one...)
Affinity DataKi:  1.04E+4nMAssay Description:Inhibition of yeast alpha-glucosidase by genisteinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-glucosidase MAL12(Saccharomyces cerevisiae)
Gyeongsang National University

LigandPNGBDBM84963(Urea derivative, 7)
Affinity DataKi:  1.05E+4nM IC50:  1.95E+4nMAssay Description:All enzymatic activities were determined by using the appropriate substrate (p-nitrophenyl-alpha-D-glucopyranoside, p-nitrophenyl-beta-D-gulcopyranos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-glucosidase MAL12(Saccharomyces cerevisiae)
Gyeongsang National University

LigandPNGBDBM84962(Urea derivative, 6)
Affinity DataKi:  1.06E+4nM IC50:  4.21E+4nMAssay Description:All enzymatic activities were determined by using the appropriate substrate (p-nitrophenyl-alpha-D-glucopyranoside, p-nitrophenyl-beta-D-gulcopyranos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-glucosidase MAL12(Saccharomyces cerevisiae)
Gyeongsang National University

LigandPNGBDBM84966(Urea derivative, 10)
Affinity DataKi:  1.21E+4nM IC50:  2.88E+4nMAssay Description:All enzymatic activities were determined by using the appropriate substrate (p-nitrophenyl-alpha-D-glucopyranoside, p-nitrophenyl-beta-D-gulcopyranos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-glucosidase MAL12(Saccharomyces cerevisiae)
Gyeongsang National University

LigandPNGBDBM243075(α-Gl inhibitor, C3)
Affinity DataKi:  1.40E+4nMpH: 7.0Assay Description:In this study, the inhibition assay of yeast enzyme was performed in 100 mM phosphate buffer pH 7.0 at 25°C with minor changes, according to the meth...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 61 total ) | Next | Last >>
Jump to: