Compile Data Set for Download or QSAR
maximum 50k data
Found 25 of ki data for polymerid = 50002809
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50497543(CHEMBL3359693)
Affinity DataKi:  0.700nMAssay Description:Inhibition of Plasmodium falciparum M1 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50497544(CHEMBL3359688)
Affinity DataKi:  0.800nMAssay Description:Inhibition of Plasmodium falciparum M1 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50497553(CHEMBL3359696)
Affinity DataKi:  1.90nMAssay Description:Inhibition of Plasmodium falciparum M1 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50497545(CHEMBL3359697)
Affinity DataKi:  4nMAssay Description:Inhibition of Plasmodium falciparum M1 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50497556(CHEMBL3359699)
Affinity DataKi:  5.5nMAssay Description:Inhibition of Plasmodium falciparum M1 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50497551(CHEMBL3359700)
Affinity DataKi:  7.40nMAssay Description:Inhibition of Plasmodium falciparum M1 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50497552(CHEMBL3359698)
Affinity DataKi:  11nMAssay Description:Inhibition of Plasmodium falciparum M1 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50497557(CHEMBL3359692)
Affinity DataKi:  12nMAssay Description:Inhibition of Plasmodium falciparum M1 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50497547(CHEMBL3359694)
Affinity DataKi:  15nMAssay Description:Inhibition of Plasmodium falciparum M1 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50497546(CHEMBL3359695)
Affinity DataKi:  23nMAssay Description:Inhibition of Plasmodium falciparum M1 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50497548(CHEMBL3359691)
Affinity DataKi:  41nMAssay Description:Inhibition of Plasmodium falciparum M1 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50339789((S)-2-((2S,3R)-3-amino-2-hydroxy-4-(4-methoxypheny...)
Affinity DataKi:  43nMAssay Description:Inhibition of Plasmodium falciparum recombinant M1-aminopeptidase expressed in Escherichia coli after 40 mins uisng fluorigenic substrate L-Leucyl-7-...More data for this Ligand-Target Pair
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50497554(CHEMBL3359689)
Affinity DataKi:  75nMAssay Description:Inhibition of Plasmodium falciparum M1 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50497549(CHEMBL3359690)
Affinity DataKi:  113nMAssay Description:Inhibition of Plasmodium falciparum M1 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM23971((2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-phenylbutanami...)
Affinity DataKi:  190nMAssay Description:Inhibition of Plasmodium falciparum recombinant M1-aminopeptidase expressed in Escherichia coli after 40 mins uisng fluorigenic substrate L-Leucyl-7-...More data for this Ligand-Target Pair
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50339790((S)-2-((2S,3R)-3-amino-4-(4-(benzyloxy)phenyl)-2-h...)
Affinity DataKi:  490nMAssay Description:Inhibition of Plasmodium falciparum recombinant M1-aminopeptidase expressed in Escherichia coli after 40 mins uisng fluorigenic substrate L-Leucyl-7-...More data for this Ligand-Target Pair
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50497555(CHEMBL3359686)
Affinity DataKi: >500nMAssay Description:Inhibition of Plasmodium falciparum M1 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50497550(CHEMBL3359687)
Affinity DataKi: >500nMAssay Description:Inhibition of Plasmodium falciparum M1 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50339784((S)-2-((2S,3R)-3-amino-2-hydroxy-4-phenylbutanamid...)
Affinity DataKi:  900nMAssay Description:Inhibition of Plasmodium falciparum recombinant M1-aminopeptidase expressed in Escherichia coli after 40 mins uisng fluorigenic substrate L-Leucyl-7-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50339785((S)-2-((2S,3R)-3-amino-2-hydroxy-4-phenylbutanamid...)
Affinity DataKi:  1.45E+3nMAssay Description:Inhibition of Plasmodium falciparum recombinant M1-aminopeptidase expressed in Escherichia coli after 40 mins uisng fluorigenic substrate L-Leucyl-7-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50339791((S)-2-((2S,3R)-3-amino-2-hydroxy-4-(naphthalen-2-y...)
Affinity DataKi:  3.00E+3nMAssay Description:Inhibition of Plasmodium falciparum recombinant M1-aminopeptidase expressed in Escherichia coli after 40 mins uisng fluorigenic substrate L-Leucyl-7-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50339792((S)-2-((2S,3R)-3-amino-2-hydroxyheptanamido)-4-met...)
Affinity DataKi:  5.30E+3nMAssay Description:Inhibition of Plasmodium falciparum recombinant M1-aminopeptidase expressed in Escherichia coli after 40 mins uisng fluorigenic substrate L-Leucyl-7-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50339786((S)-2-((2S,3R)-3-amino-2-hydroxy-4-phenylbutanamid...)
Affinity DataKi: >1.50E+4nMAssay Description:Inhibition of Plasmodium falciparum recombinant M1-aminopeptidase expressed in Escherichia coli after 40 mins uisng fluorigenic substrate L-Leucyl-7-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50339787((S)-2-((2S,3R)-3-amino-2-hydroxy-4-phenylbutanamid...)
Affinity DataKi: >1.50E+4nMAssay Description:Inhibition of Plasmodium falciparum recombinant M1-aminopeptidase expressed in Escherichia coli after 40 mins uisng fluorigenic substrate L-Leucyl-7-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50339788((S)-2-((2S,3R)-3-amino-2-hydroxy-4-phenylbutanamid...)
Affinity DataKi: >1.50E+4nMAssay Description:Inhibition of Plasmodium falciparum recombinant M1-aminopeptidase expressed in Escherichia coli after 40 mins uisng fluorigenic substrate L-Leucyl-7-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed