Found 141 Enz. Inhib. hit(s) with Target = 'Nuclear receptor subfamily 1 group I member 3' TargetNuclear receptor subfamily 1 group I member 3(Homo sapiens (Human))
Tes Pharma
Curated by ChEMBL
Tes Pharma
Curated by ChEMBL
Affinity DataEC50: 5nMAssay Description:Agonist activity at human CARMore data for this Ligand-Target Pair
3D Structure (crystal)TargetNuclear receptor subfamily 1 group I member 3(Homo sapiens (Human))
Tes Pharma
Curated by ChEMBL
Tes Pharma
Curated by ChEMBL
Affinity DataEC50: 20nMAssay Description:Agonist activity at CAR LBD (108 to 348 residues) expressed in human HepG2 cells assessed as receptor binding to PGC1alpha by lanthascreenTR-FRET coa...More data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Homo sapiens (Human))
Tes Pharma
Curated by ChEMBL
Tes Pharma
Curated by ChEMBL
Affinity DataEC50: 49nMAssay Description:Agonist activity at Polyhistidine-tagged human CAR LBD expressed in Escherichia coli by FRET-based assayMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Homo sapiens (Human))
Tes Pharma
Curated by ChEMBL
Tes Pharma
Curated by ChEMBL
Affinity DataEC50: 49nMAssay Description:Agonist activity at Polyhistidine-tagged human CAR LBD expressed in Escherichia coli by FRET-based assayMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Homo sapiens (Human))
Tes Pharma
Curated by ChEMBL
Tes Pharma
Curated by ChEMBL
Affinity DataEC50: 75nMAssay Description:Agonist activity at human CAR expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Homo sapiens (Human))
Tes Pharma
Curated by ChEMBL
Tes Pharma
Curated by ChEMBL
Affinity DataEC50: 150nMAssay Description:Agonist activity at human constitutive androstane receptor expressed in HepG2 cells co-expressing CYP2B6 incubated for 23 hrs by One-Glo luciferase r...More data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Homo sapiens (Human))
Tes Pharma
Curated by ChEMBL
Tes Pharma
Curated by ChEMBL
Affinity DataEC50: 190nMAssay Description:Agonist activity at human constitutive androstane receptor expressed in HepG2 cells co-expressing CYP2B6 incubated for 23 hrs by One-Glo luciferase r...More data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Homo sapiens (Human))
Tes Pharma
Curated by ChEMBL
Tes Pharma
Curated by ChEMBL
Affinity DataEC50: 240nMAssay Description:Agonist activity at human constitutive androstane receptor expressed in HepG2 cells co-expressing CYP2B6 incubated for 23 hrs by One-Glo luciferase r...More data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Homo sapiens (Human))
Tes Pharma
Curated by ChEMBL
Tes Pharma
Curated by ChEMBL
Affinity DataEC50: 370nMAssay Description:Agonist activity at human CAR transfected in human HepG2 cells cotransfected with CYP2B6 incubated for 23 hrs by luciferase reported gene assayMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Homo sapiens (Human))
Tes Pharma
Curated by ChEMBL
Tes Pharma
Curated by ChEMBL
Affinity DataEC50: 380nMAssay Description:Agonist activity at human CAR transfected in human HepG2 cells cotransfected with CYP2B6 incubated for 23 hrs by luciferase reported gene assayMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Homo sapiens (Human))
Tes Pharma
Curated by ChEMBL
Tes Pharma
Curated by ChEMBL
Affinity DataEC50: 400nMAssay Description:Agonist activity at human constitutive androstane receptor expressed in HepG2 cells co-expressing CYP2B6 incubated for 23 hrs by One-Glo luciferase r...More data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Homo sapiens (Human))
Tes Pharma
Curated by ChEMBL
Tes Pharma
Curated by ChEMBL
Affinity DataEC50: 410nMAssay Description:Agonist activity at human CAR transfected in human HepG2 cells cotransfected with CYP2B6 incubated for 23 hrs by luciferase reported gene assayMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Homo sapiens (Human))
Tes Pharma
Curated by ChEMBL
Tes Pharma
Curated by ChEMBL
Affinity DataEC50: 440nMAssay Description:Agonist activity at human constitutive androstane receptor expressed in HepG2 cells co-expressing CYP2B6 incubated for 23 hrs by One-Glo luciferase r...More data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Homo sapiens (Human))
Tes Pharma
Curated by ChEMBL
Tes Pharma
Curated by ChEMBL
Affinity DataEC50: 460nMAssay Description:Agonist activity at human constitutive androstane receptor expressed in HepG2 cells co-expressing CYP2B6 incubated for 23 hrs by One-Glo luciferase r...More data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Homo sapiens (Human))
Tes Pharma
Curated by ChEMBL
Tes Pharma
Curated by ChEMBL
Affinity DataEC50: 470nMAssay Description:Agonist activity at human CAR transfected in human HepG2 cells cotransfected with CYP2B6 incubated for 23 hrs by luciferase reported gene assayMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Homo sapiens (Human))
Tes Pharma
Curated by ChEMBL
Tes Pharma
Curated by ChEMBL
Affinity DataEC50: 480nMAssay Description:Agonist activity at human CAR transfected in human HepG2 cells cotransfected with CYP2B6 incubated for 23 hrs by luciferase reported gene assayMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Homo sapiens (Human))
Tes Pharma
Curated by ChEMBL
Tes Pharma
Curated by ChEMBL
Affinity DataEC50: 490nMAssay Description:Agonist activity at human CAR transfected in human HepG2 cells cotransfected with CYP2B6 incubated for 23 hrs by luciferase reported gene assayMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Homo sapiens (Human))
Tes Pharma
Curated by ChEMBL
Tes Pharma
Curated by ChEMBL
Affinity DataEC50: 490nMAssay Description:Agonist activity at human CAR transfected in human HepG2 cells cotransfected with CYP2B6 incubated for 23 hrs by luciferase reported gene assayMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Homo sapiens (Human))
Tes Pharma
Curated by ChEMBL
Tes Pharma
Curated by ChEMBL
Affinity DataEC50: 510nMAssay Description:Agonist activity at human CAR3 expressed in African green monkey COS-1 cells cotransfected with RXRalpha after 24 hrs by CYP2B6-luciferase reporter g...More data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Homo sapiens (Human))
Tes Pharma
Curated by ChEMBL
Tes Pharma
Curated by ChEMBL
Affinity DataEC50: 560nMAssay Description:Agonist activity at human constitutive androstane receptor expressed in HepG2 cells co-expressing CYP2B6 incubated for 23 hrs by One-Glo luciferase r...More data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Homo sapiens (Human))
Tes Pharma
Curated by ChEMBL
Tes Pharma
Curated by ChEMBL
Affinity DataEC50: 570nMAssay Description:Agonist activity at human constitutive androstane receptor expressed in HepG2 cells co-expressing CYP2B6 incubated for 23 hrs by One-Glo luciferase r...More data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Homo sapiens (Human))
Tes Pharma
Curated by ChEMBL
Tes Pharma
Curated by ChEMBL
Affinity DataEC50: 580nMAssay Description:Agonist activity at human CAR transfected in human HepG2 cells cotransfected with CYP2B6 incubated for 23 hrs by luciferase reported gene assayMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Homo sapiens (Human))
Tes Pharma
Curated by ChEMBL
Tes Pharma
Curated by ChEMBL
Affinity DataEC50: 590nMAssay Description:Agonist activity at human CAR transfected in human HepG2 cells cotransfected with CYP2B6 incubated for 23 hrs by luciferase reported gene assayMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Homo sapiens (Human))
Tes Pharma
Curated by ChEMBL
Tes Pharma
Curated by ChEMBL
Affinity DataEC50: 620nMAssay Description:Agonist activity at human CAR transfected in human HepG2 cells cotransfected with CYP2B6 incubated for 23 hrs by luciferase reported gene assayMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Homo sapiens (Human))
Tes Pharma
Curated by ChEMBL
Tes Pharma
Curated by ChEMBL
Affinity DataEC50: 650nMAssay Description:Agonist activity at human constitutive androstane receptor expressed in HepG2 cells co-expressing CYP2B6 incubated for 23 hrs by One-Glo luciferase r...More data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Homo sapiens (Human))
Tes Pharma
Curated by ChEMBL
Tes Pharma
Curated by ChEMBL
Affinity DataEC50: 660nMAssay Description:Agonist activity at human constitutive androstane receptor expressed in HepG2 cells co-expressing CYP2B6 incubated for 23 hrs by One-Glo luciferase r...More data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Homo sapiens (Human))
Tes Pharma
Curated by ChEMBL
Tes Pharma
Curated by ChEMBL
Affinity DataEC50: 670nMAssay Description:Agonist activity at human CAR transfected in human HepG2 cells cotransfected with CYP2B6 incubated for 23 hrs by luciferase reported gene assayMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Homo sapiens (Human))
Tes Pharma
Curated by ChEMBL
Tes Pharma
Curated by ChEMBL
Affinity DataEC50: 670nMAssay Description:Agonist activity at human constitutive androstane receptor expressed in HepG2 cells co-expressing CYP2B6 incubated for 23 hrs by One-Glo luciferase r...More data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Homo sapiens (Human))
Tes Pharma
Curated by ChEMBL
Tes Pharma
Curated by ChEMBL
Affinity DataEC50: 690nMAssay Description:Agonist activity at CAR LBD (108 to 348 residues) expressed in human HepG2 cells assessed as receptor binding to PGC1alpha by lanthascreenTR-FRET coa...More data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Homo sapiens (Human))
Tes Pharma
Curated by ChEMBL
Tes Pharma
Curated by ChEMBL
Affinity DataEC50: 740nMAssay Description:Agonist activity at human constitutive androstane receptor expressed in HepG2 cells co-expressing CYP2B6 incubated for 23 hrs by One-Glo luciferase r...More data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Homo sapiens (Human))
Tes Pharma
Curated by ChEMBL
Tes Pharma
Curated by ChEMBL
Affinity DataEC50: 840nMAssay Description:Agonist activity at human CAR transfected in human HepG2 cells cotransfected with CYP2B6 incubated for 23 hrs by luciferase reported gene assayMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Homo sapiens (Human))
Tes Pharma
Curated by ChEMBL
Tes Pharma
Curated by ChEMBL
Affinity DataEC50: 880nMAssay Description:Agonist activity at human CAR transfected in human HepG2 cells cotransfected with CYP2B6 incubated for 23 hrs by luciferase reported gene assayMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Homo sapiens (Human))
Tes Pharma
Curated by ChEMBL
Tes Pharma
Curated by ChEMBL
Affinity DataEC50: 920nMAssay Description:Agonist activity at human constitutive androstane receptor expressed in HepG2 cells co-expressing CYP2B6 incubated for 23 hrs by One-Glo luciferase r...More data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Homo sapiens (Human))
Tes Pharma
Curated by ChEMBL
Tes Pharma
Curated by ChEMBL
Affinity DataEC50: 930nMAssay Description:Agonist activity at human constitutive androstane receptor expressed in HepG2 cells co-expressing CYP2B6 incubated for 23 hrs by One-Glo luciferase r...More data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Homo sapiens (Human))
Tes Pharma
Curated by ChEMBL
Tes Pharma
Curated by ChEMBL
Affinity DataEC50: 940nMAssay Description:Agonist activity at human CAR transfected in human HepG2 cells cotransfected with CYP2B6 incubated for 23 hrs by luciferase reported gene assayMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Homo sapiens (Human))
Tes Pharma
Curated by ChEMBL
Tes Pharma
Curated by ChEMBL
Affinity DataEC50: 980nMAssay Description:Agonist activity at human CAR transfected in human HepG2 cells cotransfected with CYP2B6 incubated for 23 hrs by luciferase reported gene assayMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Homo sapiens (Human))
Tes Pharma
Curated by ChEMBL
Tes Pharma
Curated by ChEMBL
Affinity DataEC50: 990nMAssay Description:Agonist activity at human CAR transfected in human HepG2 cells cotransfected with CYP2B6 incubated for 23 hrs by luciferase reported gene assayMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Homo sapiens (Human))
Tes Pharma
Curated by ChEMBL
Tes Pharma
Curated by ChEMBL
Affinity DataEC50: 1.10E+3nMAssay Description:Agonist activity at human constitutive androstane receptor expressed in HepG2 cells co-expressing CYP2B6 incubated for 23 hrs by One-Glo luciferase r...More data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Homo sapiens (Human))
Tes Pharma
Curated by ChEMBL
Tes Pharma
Curated by ChEMBL
Affinity DataEC50: 1.10E+3nMAssay Description:Agonist activity at human constitutive androstane receptor expressed in HepG2 cells co-expressing CYP2B6 incubated for 23 hrs by One-Glo luciferase r...More data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Homo sapiens (Human))
Tes Pharma
Curated by ChEMBL
Tes Pharma
Curated by ChEMBL
Affinity DataEC50: 1.10E+3nMAssay Description:Agonist activity at human CAR transfected in human HepG2 cells cotransfected with CYP2B6 incubated for 23 hrs by luciferase reported gene assayMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Homo sapiens (Human))
Tes Pharma
Curated by ChEMBL
Tes Pharma
Curated by ChEMBL
Affinity DataEC50: 1.10E+3nMAssay Description:Agonist activity at human CAR transfected in human HepG2 cells cotransfected with CYP2B6 incubated for 23 hrs by luciferase reported gene assayMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Homo sapiens (Human))
Tes Pharma
Curated by ChEMBL
Tes Pharma
Curated by ChEMBL
Affinity DataEC50: 1.30E+3nMAssay Description:Agonist activity at human constitutive androstane receptor expressed in HepG2 cells co-expressing CYP2B6 incubated for 23 hrs by One-Glo luciferase r...More data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Homo sapiens (Human))
Tes Pharma
Curated by ChEMBL
Tes Pharma
Curated by ChEMBL
Affinity DataEC50: 1.50E+3nMAssay Description:Agonist activity at human constitutive androstane receptor expressed in HepG2 cells co-expressing CYP2B6 incubated for 23 hrs by One-Glo luciferase r...More data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Homo sapiens (Human))
Tes Pharma
Curated by ChEMBL
Tes Pharma
Curated by ChEMBL
Affinity DataEC50: 1.50E+3nMAssay Description:Agonist activity at human constitutive androstane receptor expressed in HepG2 cells co-expressing CYP2B6 incubated for 23 hrs by One-Glo luciferase r...More data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Homo sapiens (Human))
Tes Pharma
Curated by ChEMBL
Tes Pharma
Curated by ChEMBL
Affinity DataEC50: 1.50E+3nMAssay Description:Agonist activity at human CAR transfected in human HepG2 cells cotransfected with CYP2B6 incubated for 23 hrs by luciferase reported gene assayMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Homo sapiens (Human))
Tes Pharma
Curated by ChEMBL
Tes Pharma
Curated by ChEMBL
Affinity DataEC50: 1.60E+3nMAssay Description:Agonist activity at human constitutive androstane receptor expressed in HepG2 cells co-expressing CYP2B6 incubated for 23 hrs by One-Glo luciferase r...More data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Homo sapiens (Human))
Tes Pharma
Curated by ChEMBL
Tes Pharma
Curated by ChEMBL
Affinity DataEC50: 1.70E+3nMAssay Description:Agonist activity at human CAR transfected in human HepG2 cells cotransfected with CYP2B6 incubated for 23 hrs by luciferase reported gene assayMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Homo sapiens (Human))
Tes Pharma
Curated by ChEMBL
Tes Pharma
Curated by ChEMBL
Affinity DataEC50: 1.90E+3nMAssay Description:Agonist activity at human constitutive androstane receptor expressed in HepG2 cells co-expressing CYP2B6 incubated for 23 hrs by One-Glo luciferase r...More data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Homo sapiens (Human))
Tes Pharma
Curated by ChEMBL
Tes Pharma
Curated by ChEMBL
Affinity DataEC50: 2.07E+3nMAssay Description:Agonist activity at CAR LBD (108 to 348 residues) expressed in human HepG2 cells assessed as receptor binding to PGC1alpha by lanthascreenTR-FRET coa...More data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Homo sapiens (Human))
Tes Pharma
Curated by ChEMBL
Tes Pharma
Curated by ChEMBL
Affinity DataEC50: 2.10E+3nMAssay Description:Agonist activity at human constitutive androstane receptor expressed in HepG2 cells co-expressing CYP2B6 incubated for 23 hrs by One-Glo luciferase r...More data for this Ligand-Target Pair
