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Found 202 Enz. Inhib. hit(s) with Target = 'Putative P2Y purinoceptor 10'
TargetPutative P2Y purinoceptor 10(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50560840(CHEMBL4753103)
Affinity DataEC50:  0.977nMAssay Description:Agonist activity at mouse P2Y10 expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain shedding of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPutative P2Y purinoceptor 10(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50560840(CHEMBL4753103)
Affinity DataEC50:  1nMAssay Description:Agonist activity at mouse P2Y10 expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain shedding of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPutative P2Y purinoceptor 10(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096400(CHEMBL3577182)
Affinity DataEC50:  1.30nMAssay Description:Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative P2Y purinoceptor 10(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096400(CHEMBL3577182)
Affinity DataEC50:  1.30nMAssay Description:Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative P2Y purinoceptor 10(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096458(CHEMBL3577179)
Affinity DataEC50:  1.70nMAssay Description:Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative P2Y purinoceptor 10(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096458(CHEMBL3577179)
Affinity DataEC50:  1.70nMAssay Description:Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative P2Y purinoceptor 10(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096359(CHEMBL3577171)
Affinity DataEC50:  2nMAssay Description:Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative P2Y purinoceptor 10(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096359(CHEMBL3577171)
Affinity DataEC50:  2nMAssay Description:Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative P2Y purinoceptor 10(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096360(CHEMBL3577174)
Affinity DataEC50:  2.60nMAssay Description:Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative P2Y purinoceptor 10(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096360(CHEMBL3577174)
Affinity DataEC50:  2.70nMAssay Description:Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative P2Y purinoceptor 10(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096358(CHEMBL3577170)
Affinity DataEC50:  3.20nMAssay Description:Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative P2Y purinoceptor 10(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096358(CHEMBL3577170)
Affinity DataEC50:  3.20nMAssay Description:Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative P2Y purinoceptor 10(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096503(CHEMBL3577262)
Affinity DataEC50:  3.30nMAssay Description:Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative P2Y purinoceptor 10(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096503(CHEMBL3577262)
Affinity DataEC50:  3.30nMAssay Description:Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative P2Y purinoceptor 10(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096362(CHEMBL3577178)
Affinity DataEC50:  3.70nMAssay Description:Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative P2Y purinoceptor 10(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096362(CHEMBL3577178)
Affinity DataEC50:  3.70nMAssay Description:Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative P2Y purinoceptor 10(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50560837(CHEMBL4745025)
Affinity DataEC50:  5.70nMAssay Description:Agonist activity at mouse P2Y10 expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain shedding of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPutative P2Y purinoceptor 10(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50560837(CHEMBL4745025)
Affinity DataEC50:  5.80nMAssay Description:Agonist activity at mouse P2Y10 expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain shedding of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPutative P2Y purinoceptor 10(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50177139(CHEMBL3814492)
Affinity DataEC50:  6.60nMAssay Description:Agonist activity at mouse P2Y10 receptor expressed in HEK293A cells after 1.5 hrs by alkaline phosphatase tagged-TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative P2Y purinoceptor 10(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50177139(CHEMBL3814492)
Affinity DataEC50:  6.70nMAssay Description:Agonist activity at mouse P2Y10 receptor expressed in HEK293A cells after 1.5 hrs by alkaline phosphatase tagged-TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative P2Y purinoceptor 10(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096441(CHEMBL3577172)
Affinity DataEC50:  12nMAssay Description:Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative P2Y purinoceptor 10(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50560845(CHEMBL4755564)
Affinity DataEC50:  12nMAssay Description:Agonist activity at mouse P2Y10 expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain shedding of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPutative P2Y purinoceptor 10(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096441(CHEMBL3577172)
Affinity DataEC50:  12nMAssay Description:Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative P2Y purinoceptor 10(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50560845(CHEMBL4755564)
Affinity DataEC50:  12nMAssay Description:Agonist activity at mouse P2Y10 expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain shedding of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPutative P2Y purinoceptor 10(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096361(CHEMBL3577175)
Affinity DataEC50:  13nMAssay Description:Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative P2Y purinoceptor 10(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096361(CHEMBL3577175)
Affinity DataEC50:  13nMAssay Description:Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative P2Y purinoceptor 10(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50177150(CHEMBL3813843)
Affinity DataEC50:  17nMAssay Description:Agonist activity at mouse P2Y10 receptor expressed in HEK293A cells after 1.5 hrs by alkaline phosphatase tagged-TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative P2Y purinoceptor 10(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096422(CHEMBL3577137)
Affinity DataEC50:  19nMAssay Description:Agonist activity at mouse P2Y10 expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain shedding of ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative P2Y purinoceptor 10(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096349(CHEBI:52649 | CHEMBL1742484)
Affinity DataEC50:  19nMAssay Description:Agonist activity at mouse P2Y10 expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain shedding of ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative P2Y purinoceptor 10(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096422(CHEMBL3577137)
Affinity DataEC50:  20nMAssay Description:Agonist activity at mouse P2Y10 expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain shedding of ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative P2Y purinoceptor 10(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096349(CHEBI:52649 | CHEMBL1742484)
Affinity DataEC50:  20nMAssay Description:Agonist activity at mouse P2Y10 expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain shedding of ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative P2Y purinoceptor 10(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096426(CHEMBL3577150)
Affinity DataEC50:  21nMAssay Description:Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative P2Y purinoceptor 10(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096426(CHEMBL3577150)
Affinity DataEC50:  21nMAssay Description:Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative P2Y purinoceptor 10(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096422(CHEMBL3577137)
Affinity DataEC50:  25nMAssay Description:Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative P2Y purinoceptor 10(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096349(CHEBI:52649 | CHEMBL1742484)
Affinity DataEC50:  25nMAssay Description:Agonist activity at mouse P2Y10 receptor expressed in HEK293A cells after 1.5 hrs by alkaline phosphatase tagged-TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative P2Y purinoceptor 10(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096349(CHEBI:52649 | CHEMBL1742484)
Affinity DataEC50:  25nMAssay Description:Agonist activity at mouse P2Y10 receptor expressed in HEK293A cells after 1.5 hrs by alkaline phosphatase tagged-TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative P2Y purinoceptor 10(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096422(CHEMBL3577137)
Affinity DataEC50:  25nMAssay Description:Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative P2Y purinoceptor 10(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50560843(CHEMBL4759297)
Affinity DataEC50:  26nMAssay Description:Agonist activity at mouse P2Y10 expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain shedding of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPutative P2Y purinoceptor 10(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50560843(CHEMBL4759297)
Affinity DataEC50:  26nMAssay Description:Agonist activity at mouse P2Y10 expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain shedding of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPutative P2Y purinoceptor 10(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096353(CHEMBL3577145)
Affinity DataEC50:  26nMAssay Description:Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative P2Y purinoceptor 10(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096353(CHEMBL3577145)
Affinity DataEC50:  26nMAssay Description:Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative P2Y purinoceptor 10(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096349(CHEBI:52649 | CHEMBL1742484)
Affinity DataEC50:  28nMAssay Description:Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative P2Y purinoceptor 10(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096349(CHEBI:52649 | CHEMBL1742484)
Affinity DataEC50:  28nMAssay Description:Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative P2Y purinoceptor 10(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096478(CHEMBL3577180)
Affinity DataEC50:  32nMAssay Description:Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative P2Y purinoceptor 10(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096478(CHEMBL3577180)
Affinity DataEC50:  33nMAssay Description:Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative P2Y purinoceptor 10(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50560822(CHEMBL4764512)
Affinity DataEC50:  37nMAssay Description:Agonist activity at mouse P2Y10 expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain shedding of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPutative P2Y purinoceptor 10(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50560822(CHEMBL4764512)
Affinity DataEC50:  37nMAssay Description:Agonist activity at mouse P2Y10 expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain shedding of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPutative P2Y purinoceptor 10(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096350(CHEMBL3577138)
Affinity DataEC50:  39nMAssay Description:Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative P2Y purinoceptor 10(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096350(CHEMBL3577138)
Affinity DataEC50:  39nMAssay Description:Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative P2Y purinoceptor 10(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50177142(CHEMBL3813751)
Affinity DataEC50:  42nMAssay Description:Agonist activity at mouse P2Y10 receptor expressed in HEK293A cells after 1.5 hrs by alkaline phosphatase tagged-TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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