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Found 607 Enz. Inhib. hit(s) with Target = 'Ras-related C3 botulinum toxin substrate 1'
LigandPNGBDBM41685(4-[3-(4-bromophenyl)-5-(4-fluorophenyl)-2-pyrazoli...)
Affinity DataEC50:  14nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela...More data for this Ligand-Target Pair
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LigandPNGBDBM42384(2-(2-phenylethylsulfanyl)pyridine-3-carboxylic aci...)
Affinity DataEC50:  20.2nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
LigandPNGBDBM42384(2-(2-phenylethylsulfanyl)pyridine-3-carboxylic aci...)
Affinity DataEC50:  25.4nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
LigandPNGBDBM54622(3-(3,4-dimethoxyphenyl)-2-(3-fluorophenyl)-5-(4-fl...)
Affinity DataEC50:  27nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela...More data for this Ligand-Target Pair
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LigandPNGBDBM54653(4-[3-(2-methylphenyl)-5-phenyl-3,4-dihydropyrazol-...)
Affinity DataEC50:  30nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela...More data for this Ligand-Target Pair
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LigandPNGBDBM41685(4-[3-(4-bromophenyl)-5-(4-fluorophenyl)-2-pyrazoli...)
Affinity DataEC50:  32nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela...More data for this Ligand-Target Pair
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LigandPNGBDBM54661(4-[3-(4-methoxyphenyl)-5-methyl-3,4-dihydropyrazol...)
Affinity DataEC50:  63nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela...More data for this Ligand-Target Pair
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LigandPNGBDBM43221(2-(benzoylcarbamothioylamino)-5,5-dimethyl-4,7-dih...)
Affinity DataEC50:  80.6nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela...More data for this Ligand-Target Pair
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LigandPNGBDBM43221(2-(benzoylcarbamothioylamino)-5,5-dimethyl-4,7-dih...)
Affinity DataEC50:  80.6nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela...More data for this Ligand-Target Pair
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LigandPNGBDBM46331(1-[(5-bromanylfuran-2-yl)carbonylamino]-3-[(4-chlo...)
Affinity DataEC50:  85.7nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela...More data for this Ligand-Target Pair
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LigandPNGBDBM54623(1-(2,5-dichlorophenyl)-3-(4-fluorophenyl)-5-(4-met...)
Affinity DataEC50:  89nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela...More data for this Ligand-Target Pair
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LigandPNGBDBM46328(MLS000393082 | N-[3-(1H-benzimidazol-2-yl)-4,5,6,7...)
Affinity DataEC50:  99.9nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela...More data for this Ligand-Target Pair
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LigandPNGBDBM43246(2-(2,5-dimethyl-3-furoyl)oxybenzoic acid | 2-(2,5-...)
Affinity DataEC50:  103nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela...More data for this Ligand-Target Pair
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LigandPNGBDBM54619(3-(4-chlorophenyl)-5-(3,4-dimethoxyphenyl)-1-pheny...)
Affinity DataEC50:  139nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela...More data for this Ligand-Target Pair
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LigandPNGBDBM43252(2-(2-bromobenzyl)oxybenzoic acid | 2-[(2-bromophen...)
Affinity DataEC50:  151nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela...More data for this Ligand-Target Pair
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LigandPNGBDBM44154((E)-3-[1-benzyl-3-(4-chlorophenyl)pyrazol-4-yl]acr...)
Affinity DataEC50:  164nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela...More data for this Ligand-Target Pair
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LigandPNGBDBM43241(1-[2-(2,5-dimethylphenoxy)ethyl]-3-indolecarboxyli...)
Affinity DataEC50:  222nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela...More data for this Ligand-Target Pair
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LigandPNGBDBM54709(1-[4-(4-bromophenyl)-1-piperazinyl]-3-[3-(4-methox...)
Affinity DataEC50:  257nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela...More data for this Ligand-Target Pair
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LigandPNGBDBM43265(9-(2,5-dimethoxyphenyl)-2,6,7-trihydroxy-3-xanthen...)
Affinity DataEC50:  280nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela...More data for this Ligand-Target Pair
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LigandPNGBDBM43270(MLS000591720 | N-(12-Cyano-indolizino[2,3-b]quinox...)
Affinity DataEC50:  292nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela...More data for this Ligand-Target Pair
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LigandPNGBDBM43266(7-(diethylamino)-3-[4-(4-methoxyphenyl)-1,3-thiazo...)
Affinity DataEC50:  372nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela...More data for this Ligand-Target Pair
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LigandPNGBDBM54638(4-[3-(2-bromophenyl)-5-(4-methoxyphenyl)-2-pyrazol...)
Affinity DataEC50:  449nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela...More data for this Ligand-Target Pair
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LigandPNGBDBM54570(3-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]-1-[4-...)
Affinity DataEC50:  527nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela...More data for this Ligand-Target Pair
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LigandPNGBDBM43266(7-(diethylamino)-3-[4-(4-methoxyphenyl)-1,3-thiazo...)
Affinity DataEC50:  554nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela...More data for this Ligand-Target Pair
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LigandPNGBDBM43256(7-(3,4-dihydro-1H-isoquinolin-2-ylcarbonyl)-3-(2-m...)
Affinity DataEC50:  605nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela...More data for this Ligand-Target Pair
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LigandPNGBDBM34905(1,6-dimethyl-3-propyl-pyrimido[5,4-e][1,2,4]triazi...)
Affinity DataEC50:  623nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela...More data for this Ligand-Target Pair
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LigandPNGBDBM43290(2-methyl-1-[2-(2-methylphenoxy)ethyl]-3-indolecarb...)
Affinity DataEC50:  625nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela...More data for this Ligand-Target Pair
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LigandPNGBDBM46322((4E)-2-methoxy-4-[(5H-[1,2,4]triazino[5,6-b]indol-...)
Affinity DataEC50:  634nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela...More data for this Ligand-Target Pair
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LigandPNGBDBM43278(1-[2-(2-isopropyl-5-methyl-phenoxy)ethyl]indole-3-...)
Affinity DataEC50:  635nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela...More data for this Ligand-Target Pair
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LigandPNGBDBM43246(2-(2,5-dimethyl-3-furoyl)oxybenzoic acid | 2-(2,5-...)
Affinity DataEC50:  665nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
LigandPNGBDBM54570(3-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]-1-[4-...)
Affinity DataEC50:  675nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
LigandPNGBDBM54594(3-(4-bromophenyl)-1-(2-chlorophenyl)-5-(4-methoxyp...)
Affinity DataEC50:  697nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
LigandPNGBDBM43241(1-[2-(2,5-dimethylphenoxy)ethyl]-3-indolecarboxyli...)
Affinity DataEC50:  802nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela...More data for this Ligand-Target Pair
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LigandPNGBDBM43277(1-(2-phenoxyethyl)-3-indolecarboxylic acid | 1-(2-...)
Affinity DataEC50:  857nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela...More data for this Ligand-Target Pair
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LigandPNGBDBM43270(MLS000591720 | N-(12-Cyano-indolizino[2,3-b]quinox...)
Affinity DataEC50:  889nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela...More data for this Ligand-Target Pair
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LigandPNGBDBM43261(3-ethyl-4-keto-phthalazine-1-carboxylic acid [2-[2...)
Affinity DataEC50:  892nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela...More data for this Ligand-Target Pair
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LigandPNGBDBM46335(2-[(2-chlorobenzyl)amino]benzoic acid | 2-[(2-chlo...)
Affinity DataEC50:  899nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
LigandPNGBDBM54571(1-[4-(4-fluorophenyl)-1-piperazinyl]-3-[3-(4-metho...)
Affinity DataEC50:  912nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela...More data for this Ligand-Target Pair
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LigandPNGBDBM46314(2-(4-fluoro-N-[2-[(8-methoxy-5H-[1,2,4]triazin[5,6...)
Affinity DataEC50:  923nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela...More data for this Ligand-Target Pair
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LigandPNGBDBM46326(2-(3,4-Dimethyl-phenyl)-4-[(2-methoxy-4-thiocyanat...)
Affinity DataEC50:  966nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela...More data for this Ligand-Target Pair
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LigandPNGBDBM46319(3-[(5Z)-5-[[5-(1,3-benzothiazol-2-yl)-2-furanyl]me...)
Affinity DataEC50:  976nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela...More data for this Ligand-Target Pair
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LigandPNGBDBM43230(2-(7,8-dihydro-6H-cyclopenta[2,3]thieno[2,4-d]pyri...)
Affinity DataEC50:  1.08E+3nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela...More data for this Ligand-Target Pair
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LigandPNGBDBM54578(1-[4-(2-fluorophenyl)-1-piperazinyl]-3-[3-(4-metho...)
Affinity DataEC50:  1.11E+3nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela...More data for this Ligand-Target Pair
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LigandPNGBDBM54554(3-[3-(2-chlorophenyl)-1,2,4-oxadiazol-5-yl]-1-[4-(...)
Affinity DataEC50:  1.19E+3nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela...More data for this Ligand-Target Pair
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LigandPNGBDBM54584(1-[4-(2,5-dimethylphenyl)-1-piperidinyl]-3-[3-(4-m...)
Affinity DataEC50:  1.22E+3nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela...More data for this Ligand-Target Pair
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LigandPNGBDBM54565(1-[4-(2,5-dimethylphenyl)-1-piperazinyl]-3-[3-(3-m...)
Affinity DataEC50:  1.22E+3nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela...More data for this Ligand-Target Pair
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LigandPNGBDBM43239(3-(4-acetylphenyl)-1-(4-nitrophenyl)-2-propyn-1-on...)
Affinity DataEC50:  1.22E+3nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela...More data for this Ligand-Target Pair
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LigandPNGBDBM43230(2-(7,8-dihydro-6H-cyclopenta[2,3]thieno[2,4-d]pyri...)
Affinity DataEC50:  1.22E+3nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela...More data for this Ligand-Target Pair
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LigandPNGBDBM54553(1-[4-(2,5-dimethylphenyl)-1-piperazinyl]-3-[3-(4-f...)
Affinity DataEC50:  1.27E+3nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela...More data for this Ligand-Target Pair
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LigandPNGBDBM54576(1-[4-(2,3-dimethylphenyl)-1-piperazinyl]-3-[3-(4-m...)
Affinity DataEC50:  1.31E+3nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela...More data for this Ligand-Target Pair
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