Compile Data Set for Download or QSAR
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Found 4 Enz. Inhib. hit(s) with Target = 'Secretin receptor'
TargetSecretin receptor(Homo sapiens (Human))
Mayo Clinic

Curated by ChEMBL
LigandPNGBDBM50327887(CHEMBL1255581 | HSDGTFTSELSRLQDSARLQRLLQGLV-NH2)
Affinity DataEC50:  0.0800nMAssay Description:Agonist activity at secretin receptor expressed in CHO cells assessed as increase of cAMP levelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSecretin receptor(Homo sapiens (Human))
Mayo Clinic

Curated by ChEMBL
LigandPNGBDBM50327888(CHEMBL1256314)
Affinity DataEC50:  0.100nMAssay Description:Agonist activity at secretin receptor expressed in CHO cells assessed as increase of cAMP levelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSecretin receptor(Homo sapiens (Human))
Mayo Clinic

Curated by ChEMBL
LigandPNGBDBM50327887(CHEMBL1255581 | HSDGTFTSELSRLQDSARLQRLLQGLV-NH2)
Affinity DataKi:  3.5nMAssay Description:Displacement of [125I]-secretin-27 from secretin receptor expressed in CHO cells by gamma-spectrometer analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSecretin receptor(Homo sapiens (Human))
Mayo Clinic

Curated by ChEMBL
LigandPNGBDBM50327888(CHEMBL1256314)
Affinity DataKi:  11nMAssay Description:Displacement of [125I]-secretin-27 from secretin receptor expressed in CHO cells by gamma-spectrometer analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed