Found 440 Enz. Inhib. hit(s) with Target = 'Motilin receptor' 
Affinity DataIC50: 1.10nMAssay Description:Displacement of [125I]motilin from MTL receptor in rabbit duodenum homogenateMore data for this Ligand-Target Pair
Affinity DataIC50: 1.80nMAssay Description:In vitro binding affinity towards motilin receptor was determined after treatment with hydrochloric acid in rabbit small intestinal smooth muscle tis...More data for this Ligand-Target Pair
Affinity DataIC50: 1.90nMAssay Description:In vitro binding affinity towards motilin receptor was determined in rabbit small intestinal smooth muscle tissue homogenateMore data for this Ligand-Target Pair
Affinity DataIC50: 1.90nMAssay Description:Displacement of [125I]motilin from MTL receptor in rabbit duodenum homogenateMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Antagonist activity against human motilin receptor in aequoscreen cells assessed as inhibition of motilin induced calcium release by aequorin assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.30nMAssay Description:In vitro binding affinity towards motilin receptor was determined in rabbit small intestinal smooth muscle tissue homogenateMore data for this Ligand-Target Pair
Affinity DataIC50: 2.5nMAssay Description:In vitro binding affinity towards motilin receptor was determined in rabbit small intestinal smooth muscle tissue homogenateMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Antagonist activity against human motilin receptor in aequoscreen cells assessed as inhibition of motilin induced calcium release by aequorin assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.20nMAssay Description:Concentration required for in vitro motilin receptor binding, expressed as negative logarithm of IC50More data for this Ligand-Target Pair
Affinity DataIC50: 3.20nMAssay Description:In vitro binding affinity towards motilin receptor was determined in rabbit small intestinal smooth muscle tissue homogenateMore data for this Ligand-Target Pair
Affinity DataIC50: 3.20nMAssay Description:Compound was tested for in vitro motilin receptor binding affinityMore data for this Ligand-Target Pair
Affinity DataIC50: 3.40nMAssay Description:Compound was tested for in vitro motilin receptor binding affinity after treatment with hydrochloric acid solution (pH 2.5)More data for this Ligand-Target Pair
Affinity DataIC50: 3.5nMAssay Description:In vitro binding affinity towards motilin receptor was determined in rabbit small intestinal smooth muscle tissue homogenateMore data for this Ligand-Target Pair
Affinity DataIC50: 3.80nMAssay Description:Concentration required for in vitro motilin receptor binding, expressed as negative logarithm of IC50More data for this Ligand-Target Pair
Affinity DataIC50: 3.80nMAssay Description:In vitro binding affinity towards motilin receptor was determined after treatment with hydrochloric acid in rabbit small intestinal smooth muscle tis...More data for this Ligand-Target Pair
Affinity DataIC50: 3.80nMAssay Description:In vitro binding affinity towards motilin receptor was determined after treatment with hydrochloric acid in rabbit small intestinal smooth muscle tis...More data for this Ligand-Target Pair
Affinity DataIC50: 3.90nMAssay Description:In vitro binding affinity towards motilin receptor was determined after treatment with hydrochloric acid in rabbit small intestinal smooth muscle tis...More data for this Ligand-Target Pair
Affinity DataIC50: 4.30nMAssay Description:Displacement of [125I]motilin from MTL receptor in rabbit duodenum homogenateMore data for this Ligand-Target Pair
Affinity DataIC50: 4.70nMAssay Description:Compound was tested for in vitro motilin receptor binding affinityMore data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Displacement of [125I]motilin from MTL receptor in rabbit duodenum homogenateMore data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:In vitro binding affinity towards motilin receptor was determined in rabbit small intestinal smooth muscle tissue homogenateMore data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Concentration required for in vitro motilin receptor binding, expressed as negative logarithm of IC50More data for this Ligand-Target Pair
Affinity DataIC50: 6.5nMpH: 2.5 T: 2°CAssay Description:Concentration required for in vitro acid stability with hydrochloric acid solution (pH 2.5 ) at room temperature for 2 hr by assaying the solution fo...More data for this Ligand-Target Pair
Affinity DataIC50: 6.5nMAssay Description:In vitro binding affinity towards motilin receptor was determined after treatment with hydrochloric acid in rabbit small intestinal smooth muscle tis...More data for this Ligand-Target Pair
Affinity DataIC50: 6.90nMAssay Description:Compound was tested for in vitro motilin receptor binding affinityMore data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Inhibition of the motilin receptor (MTL-R)More data for this Ligand-Target Pair
Affinity DataIC50: 7.60nMAssay Description:Compound was tested for in vitro motilin receptor binding affinityMore data for this Ligand-Target Pair
Affinity DataIC50: 7.90nMAssay Description:In vitro binding affinity towards motilin receptor was determined after treatment with hydrochloric acid in rabbit small intestinal smooth muscle tis...More data for this Ligand-Target Pair
Affinity DataIC50: 7.90nMpH: 2.5 T: 2°CAssay Description:Concentration required for in vitro acid stability with hydrochloric acid solution (pH 2.5 ) at room temperature for 2 hr by assaying the solution fo...More data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Antagonist activity against human motilin receptor in aequoscreen cells assessed as inhibition of motilin induced calcium release by aequorin assayMore data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Activity at rabbit duodenum motilin receptor by tissue contractility assayMore data for this Ligand-Target Pair
Affinity DataIC50: 8.30nMpH: 2.5Assay Description:Compound was tested for in vitro motilin receptor binding affinity after treatment with hydrochloric acid solution (pH 2.5)More data for this Ligand-Target Pair
Affinity DataIC50: 8.90nMpH: 2.5 T: 2°CAssay Description:Concentration required for in vitro acid stability with hydrochloric acid solution (pH 2.5 ) at room temperature for 2 hr by assaying the solution fo...More data for this Ligand-Target Pair
Affinity DataIC50: 8.90nMAssay Description:In vitro binding affinity towards motilin receptor was determined after treatment with hydrochloric acid in rabbit small intestinal smooth muscle tis...More data for this Ligand-Target Pair
Affinity DataIC50: 8.90nMpH: 2.5 T: 2°CAssay Description:Concentration required for in vitro acid stability with hydrochloric acid solution (pH 2.5 ) at room temperature for 2 hr by assaying the solution fo...More data for this Ligand-Target Pair
Affinity DataIC50: 9.10nMAssay Description:In vitro binding affinity towards motilin receptor was determined in rabbit small intestinal smooth muscle tissue homogenateMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of [125]I-motilin binding to rabbit motilin receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of the motilin receptor (MTL-R)More data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of [125]I-motilin binding to rabbit motilin receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Displacement of [125I]motilin from MTL receptor in rabbit duodenum homogenateMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Displacement of [125I]motilin from MTL receptor in rabbit duodenum homogenateMore data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Inhibition of [125]I-motilin binding to rabbit motilin receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 15nMpH: 2.5Assay Description:Compound was tested for in vitro motilin receptor binding affinity after treatment with hydrochloric acid solution (pH 2.5)More data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Inhibition of the motilin receptor (MTL-R)More data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibition of [125]I-motilin binding to rabbit motilin receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 21nMAssay Description:Activity at rabbit duodenum motilin receptor by tissue contractility assayMore data for this Ligand-Target Pair
Affinity DataIC50: 21nMAssay Description:Inhibition of [125]I-motilin binding to rabbit motilin receptor at 1 uMMore data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:Activity at human MOTR expressed in CHO cells assessed as inhibition of motilin-induced calcium releaseMore data for this Ligand-Target Pair
Affinity DataIC50: 24nMAssay Description:Displacement of [125I]motilin from MTL receptor in rabbit duodenum homogenateMore data for this Ligand-Target Pair
Affinity DataIC50: 24nMAssay Description:Activity at rabbit duodenum motilin receptor by tissue contractility assayMore data for this Ligand-Target Pair
