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Found 851 Enz. Inhib. hit(s) with Target = 'Phenylethanolamine N-methyltransferase'
TargetPhenylethanolamine N-methyltransferase(Homo sapiens (Human))
Astex Therapeutics

Curated by ChEMBL
LigandPNGBDBM13014(7,8-Dichloro-1,2,3,4-tetrahydro-isoquinoline; hydr...)
Affinity DataIC50:  3nMAssay Description:Inhibition of PNMTMore data for this Ligand-Target Pair
TargetPhenylethanolamine N-methyltransferase(Homo sapiens (Human))
Astex Therapeutics

Curated by ChEMBL
LigandPNGBDBM13014(7,8-Dichloro-1,2,3,4-tetrahydro-isoquinoline; hydr...)
Affinity DataIC50:  10nMAssay Description:Inhibition of rabbit adrenal phenylethanolamine N-methyl-transferaseMore data for this Ligand-Target Pair
TargetPhenylethanolamine N-methyltransferase(Homo sapiens (Human))
Astex Therapeutics

Curated by ChEMBL
LigandPNGBDBM13014(7,8-Dichloro-1,2,3,4-tetrahydro-isoquinoline; hydr...)
Affinity DataIC50:  10nMAssay Description:Dissociation constant(Ki) of compound was determined to measure PNMT-inhibitory potencyMore data for this Ligand-Target Pair
TargetPhenylethanolamine N-methyltransferase(Homo sapiens (Human))
Astex Therapeutics

Curated by ChEMBL
LigandPNGBDBM50240934(3-(hydroxymethyl)-N-(3,3,3-trifluoropropyl)-1,2,3,...)
Affinity DataIC50:  28nMAssay Description:Inhibition of PNMTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhenylethanolamine N-methyltransferase(Homo sapiens (Human))
Astex Therapeutics

Curated by ChEMBL
LigandPNGBDBM50028902(7,8-dichloro-2-[2-(7,8-dichloro-1,2,3,4-tetrahydro...)
Affinity DataIC50:  80nMAssay Description:Inhibition of rabbit adrenal phenylethanolamine N-methyl-transferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhenylethanolamine N-methyltransferase(Homo sapiens (Human))
Astex Therapeutics

Curated by ChEMBL
LigandPNGBDBM50029108(6,7,8-Trichloro-1,2,3,4-tetrahydro-isoquinoline | ...)
Affinity DataIC50:  100nMAssay Description:In vitro inhibitory potency of the compound was measured against phenylethanolamine N-methyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhenylethanolamine N-methyltransferase(Homo sapiens (Human))
Astex Therapeutics

Curated by ChEMBL
LigandPNGBDBM50028908(7,8-dichloro-2-[4-(7,8-dichloro-1,2,3,4-tetrahydro...)
Affinity DataIC50:  100nMAssay Description:Inhibition of rabbit adrenal phenylethanolamine N-methyl-transferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhenylethanolamine N-methyltransferase(Homo sapiens (Human))
Astex Therapeutics

Curated by ChEMBL
LigandPNGBDBM50029102(7-Chloro-1,2,3,4-tetrahydro-isoquinoline | CHEMBL1...)
Affinity DataIC50:  200nMAssay Description:Dissociation constant(Ki) of compound was determined to measure Phenylethanolamine N-methyltransferase inhibitory potencyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhenylethanolamine N-methyltransferase(Homo sapiens (Human))
Astex Therapeutics

Curated by ChEMBL
LigandPNGBDBM50029101(5,6,7,8-Tetrachloro-1,2,3,4-tetrahydro-isoquinolin...)
Affinity DataIC50:  200nMAssay Description:In vitro inhibitory potency of the compound was measured against phenylethanolamine N-methyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhenylethanolamine N-methyltransferase(Homo sapiens (Human))
Astex Therapeutics

Curated by ChEMBL
LigandPNGBDBM50029107(8-Chloro-1,2,3,4-tetrahydro-isoquinoline | CHEMBL1...)
Affinity DataIC50:  200nMAssay Description:In vitro inhibitory potency of the compound was measured against phenylethanolamine N-methyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhenylethanolamine N-methyltransferase(Homo sapiens (Human))
Astex Therapeutics

Curated by ChEMBL
LigandPNGBDBM50029099(5,7,8-Trichloro-1,2,3,4-tetrahydro-isoquinoline | ...)
Affinity DataIC50:  300nMAssay Description:Dissociation constant(Ki) of compound was determined to measure Phenylethanolamine N-methyltransferase inhibitory potencyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhenylethanolamine N-methyltransferase(Homo sapiens (Human))
Astex Therapeutics

Curated by ChEMBL
LigandPNGBDBM50028903(7,8-dichloro-2-[3-(7,8-dichloro-1,2,3,4-tetrahydro...)
Affinity DataIC50:  300nMAssay Description:Inhibition of rabbit adrenal phenylethanolamine N-methyl-transferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhenylethanolamine N-methyltransferase(Homo sapiens (Human))
Astex Therapeutics

Curated by ChEMBL
LigandPNGBDBM50029106(2,3-Dichloro-benzylamine | CHEMBL13165)
Affinity DataIC50:  600nMAssay Description:Invitro inhibitory potency of the compound was measured against phenylethanolamine N-methyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhenylethanolamine N-methyltransferase(Homo sapiens (Human))
Astex Therapeutics

Curated by ChEMBL
LigandPNGBDBM50028910(7,8-dichloro-2-[6-(7,8-dichloro-1,2,3,4-tetrahydro...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of rabbit adrenal phenylethanolamine N-methyl-transferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhenylethanolamine N-methyltransferase(Homo sapiens (Human))
Astex Therapeutics

Curated by ChEMBL
LigandPNGBDBM50028901(7,8-Dichloro-2-ethyl-1,2,3,4-tetrahydro-isoquinoli...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of rabbit adrenal phenylethanolamine N-methyl-transferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhenylethanolamine N-methyltransferase(Homo sapiens (Human))
Astex Therapeutics

Curated by ChEMBL
LigandPNGBDBM50028914(7,8-dichloro-2-[7-(7,8-dichloro-1,2,3,4-tetrahydro...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of rabbit adrenal phenylethanolamine N-methyl-transferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhenylethanolamine N-methyltransferase(Homo sapiens (Human))
Astex Therapeutics

Curated by ChEMBL
LigandPNGBDBM50028911(7,8-dichloro-2-[8-(7,8-dichloro-1,2,3,4-tetrahydro...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of rabbit adrenal phenylethanolamine N-methyl-transferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhenylethanolamine N-methyltransferase(Homo sapiens (Human))
Astex Therapeutics

Curated by ChEMBL
LigandPNGBDBM50028909(2-(7,8-Dichloro-3,4-dihydro-1H-isoquinolin-2-yl)-e...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of rabbit adrenal phenylethanolamine N-methyl-transferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhenylethanolamine N-methyltransferase(Homo sapiens (Human))
Astex Therapeutics

Curated by ChEMBL
LigandPNGBDBM50028913(7,8-Dichloro-2-propyl-1,2,3,4-tetrahydro-isoquinol...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of rabbit adrenal phenylethanolamine N-methyl-transferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhenylethanolamine N-methyltransferase(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50028801(CHEMBL18486 | Cyclononanecarbaldehyde)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibitory activity against phenylethanolamine N-methyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhenylethanolamine N-methyltransferase(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50028808(CHEMBL18718 | Cyclononyl-trimethylsilanyloxy-aceto...)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibitory activity against phenylethanolamine N-methyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhenylethanolamine N-methyltransferase(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50028814(2-Amino-1-cyclononyl-ethanol | CHEMBL278978)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibitory activity against phenylethanolamine N-methyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhenylethanolamine N-methyltransferase(Homo sapiens (Human))
Astex Therapeutics

Curated by ChEMBL
LigandPNGBDBM50028912(2-Benzyl-7,8-dichloro-1,2,3,4-tetrahydro-isoquinol...)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibition of rabbit adrenal phenylethanolamine N-methyl-transferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhenylethanolamine N-methyltransferase(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50028783(2-Amino-1-cyclooctyl-ethanol | CHEMBL1204148 | CHE...)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibitory activity against phenylethanolamine N-methyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhenylethanolamine N-methyltransferase(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50028783(2-Amino-1-cyclooctyl-ethanol | CHEMBL1204148 | CHE...)
Affinity DataIC50:  8.00E+3nMAssay Description:The compound was measured for the 50% inhibition of phenylethanolamine N-methyl-transferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhenylethanolamine N-methyltransferase(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50028651(1-Aminomethyl-cycloundecanol | CHEMBL18707)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibitory activity against phenylethanolamine N-methyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhenylethanolamine N-methyltransferase(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50028802(CHEMBL275870 | Cycloheptyl-trimethylsilanyloxy-ace...)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibitory activity against phenylethanolamine N-methyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhenylethanolamine N-methyltransferase(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50028805(2-Amino-1-cycloheptyl-ethanol | CHEMBL280477)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibitory activity against phenylethanolamine N-methyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhenylethanolamine N-methyltransferase(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50028809(1-Trimethylsilanyloxy-cycloundecanecarbonitrile | ...)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibitory activity against phenylethanolamine N-methyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhenylethanolamine N-methyltransferase(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50028812(Aldehydes, 6 | CHEMBL277996 | Cycloheptanecarbalde...)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibitory activity against phenylethanolamine N-methyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhenylethanolamine N-methyltransferase(Homo sapiens (Human))
Astex Therapeutics

Curated by ChEMBL
LigandPNGBDBM12584((3-chlorophenyl)methanamine | 1-(3-CHLOROPHENYL)ME...)
Affinity DataIC50:  9.00E+3nMAssay Description:Invitro inhibitory potency of the compound was measured against phenylethanolamine N-methyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhenylethanolamine N-methyltransferase(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50028794(2-Amino-1-cycloundecyl-ethanol | CHEMBL19170)
Affinity DataIC50:  9.00E+3nMAssay Description:Inhibitory activity against phenylethanolamine N-methyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhenylethanolamine N-methyltransferase(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50028846(CHEMBL279363 | Cycloundecanecarbaldehyde)
Affinity DataIC50:  9.00E+3nMAssay Description:Inhibitory activity against phenylethanolamine N-methyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhenylethanolamine N-methyltransferase(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50028835(CHEMBL18302 | Cycloundecyl-trimethylsilanyloxy-ace...)
Affinity DataIC50:  9.00E+3nMAssay Description:Inhibitory activity against phenylethanolamine N-methyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhenylethanolamine N-methyltransferase(Homo sapiens (Human))
Astex Therapeutics

Curated by ChEMBL
LigandPNGBDBM50028906(7,8-dichloro-2-[5-(7,8-dichloro-1,2,3,4-tetrahydro...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of rabbit adrenal phenylethanolamine N-methyl-transferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhenylethanolamine N-methyltransferase(Homo sapiens (Human))
Astex Therapeutics

Curated by ChEMBL
LigandPNGBDBM13014(7,8-Dichloro-1,2,3,4-tetrahydro-isoquinoline; hydr...)
Affinity DataIC50:  1.00E+4nMAssay Description:In vitro inhibitory activity against human phenylethanolamine N-methyl-transferaseMore data for this Ligand-Target Pair
TargetPhenylethanolamine N-methyltransferase(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50028785(2-Amino-1-cyclohexyl-ethanol | CHEMBL1204147 | CHE...)
Affinity DataIC50:  1.40E+4nMAssay Description:Inhibitory activity against phenylethanolamine N-methyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhenylethanolamine N-methyltransferase(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50028785(2-Amino-1-cyclohexyl-ethanol | CHEMBL1204147 | CHE...)
Affinity DataIC50:  1.40E+4nMAssay Description:The compound was measured for the 50% inhibition of phenylethanolamine N-methyl-transferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhenylethanolamine N-methyltransferase(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50028800(1-Aminomethyl-cyclononanol | CHEMBL278410)
Affinity DataIC50:  1.70E+4nMAssay Description:Inhibitory activity against phenylethanolamine N-methyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhenylethanolamine N-methyltransferase(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50028851(CHEMBL276087 | Cyclononanone)
Affinity DataIC50:  1.70E+4nMAssay Description:Inhibitory activity against phenylethanolamine N-methyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhenylethanolamine N-methyltransferase(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50028838(1-Trimethylsilanyloxy-cyclononanecarbonitrile | CH...)
Affinity DataIC50:  1.70E+4nMAssay Description:Inhibitory activity against phenylethanolamine N-methyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhenylethanolamine N-methyltransferase(Homo sapiens (Human))
Astex Therapeutics

Curated by ChEMBL
LigandPNGBDBM50029104(2-Chloro-benzylamine | CHEMBL12712)
Affinity DataIC50:  2.00E+4nMAssay Description:Invitro inhibitory potency of the compound was measured against phenylethanolamine N-methyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhenylethanolamine N-methyltransferase(Homo sapiens (Human))
Astex Therapeutics

Curated by ChEMBL
LigandPNGBDBM50029105(2-(3,4,-dichlorophenyl)ethylamine | 2-(3,4-Dichlor...)
Affinity DataIC50:  2.00E+4nMAssay Description:In vitro inhibitory potency of the compound was measured against phenylethanolamine N-methyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhenylethanolamine N-methyltransferase(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50028836(2-Amino-1-cyclooct-1-enyl-ethanol | CHEMBL18481)
Affinity DataIC50:  3.80E+4nMAssay Description:Inhibitory activity against phenylethanolamine N-methyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhenylethanolamine N-methyltransferase(Homo sapiens (Human))
Astex Therapeutics

Curated by ChEMBL
LigandPNGBDBM50028905(7,8-Dichloro-2-(6-phenyl-hexyl)-1,2,3,4-tetrahydro...)
Affinity DataIC50:  5.00E+4nMAssay Description:Inhibition of rabbit adrenal phenylethanolamine N-methyl-transferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhenylethanolamine N-methyltransferase(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50028828(2-Amino-1-cyclohex-3-enyl-ethanol | CHEMBL18594)
Affinity DataIC50:  5.20E+4nMAssay Description:Inhibitory activity against phenylethanolamine N-methyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhenylethanolamine N-methyltransferase(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50028816(2-Amino-1-cycloocta-1,7-dienyl-ethanol | CHEMBL278...)
Affinity DataIC50:  5.70E+4nMAssay Description:Inhibitory activity against phenylethanolamine N-methyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhenylethanolamine N-methyltransferase(Homo sapiens (Human))
Astex Therapeutics

Curated by ChEMBL
LigandPNGBDBM50029103(2-(3-Chloro-phenyl)-1-methyl-ethylamine | CHEMBL14...)
Affinity DataIC50:  6.00E+4nMAssay Description:In vitro inhibitory potency of the compound was measured against phenylethanolamine N-methyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhenylethanolamine N-methyltransferase(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50028798(1-Trimethylsilanyloxy-cyclooctanecarbonitrile | CH...)
Affinity DataIC50:  7.20E+4nMAssay Description:Inhibitory activity against phenylethanolamine N-methyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhenylethanolamine N-methyltransferase(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50028793(CHEMBL18737 | Cyclooctanone)
Affinity DataIC50:  7.20E+4nMAssay Description:Inhibitory activity against phenylethanolamine N-methyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 851 total ) | Next | Last >>
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