Compile Data Set for Download or QSAR
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Found 4 Enz. Inhib. hit(s) with Target = 'Cyclin-dependent protein kinase PHO85'
LigandPNGBDBM50326018((1R,2R,3R,4R,5R,6S)-2,3,4,5,6-pentakis(phosphonoox...)
Affinity DataKi:  1.90E+4nMAssay Description:Competitive inhibition of Saccharomyces cerevisiae Pho80-Pho85-Pho81-MD catalyzed phosphorylation of Pho4 assessed as increase in substrate concentra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent protein kinase PHO85(Saccharomyces cerevisiae)
University Of California

Curated by ChEMBL
LigandPNGBDBM50113707(2,6,9-Trisubstitute purine, 2 | 2-(2-hydroxyethyla...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of yeast W303 Pho85 phosphorylation assessed as [32P] incorporation in histone H1 from [gamma32P]ATP by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50326018((1R,2R,3R,4R,5R,6S)-2,3,4,5,6-pentakis(phosphonoox...)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of Saccharomyces cerevisiae Pho80-Pho85-Pho81-MD catalyzed phosphorylation of Pho4-site 6 peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent protein kinase PHO85(Saccharomyces cerevisiae)
University Of California

Curated by ChEMBL
LigandPNGBDBM50267719(2-(6-((3-chlorophenyl)(methyl)amino)-9-isopropyl-9...)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibition of yeast W303 Pho85 phosphorylation assessed as [32P] incorporation in histone H1 from [gamma32P]ATP by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed