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Found 290 Enz. Inhib. hit(s) with Target = 'Dopamine beta-hydroxylase'
TargetDopamine beta-hydroxylase(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50014978(1-(3,5-Difluoro-4-hydroxy-benzyl)-1,3-dihydro-imid...)
Affinity DataKi:  5.70nMpH: 4.5Assay Description:Binding affinity towards Dopamine beta hydroxylase using tyramine substrate at pH 4.5 in the absence of fumarateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDopamine beta-hydroxylase(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50014983(1-(3,5-Difluoro-benzyl)-1,3-dihydro-imidazole-2-th...)
Affinity DataKi:  41nMpH: 4.5Assay Description:Binding affinity towards Dopamine beta hydroxylase using tyramine substrate at pH 4.5 in the absence of fumarateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDopamine beta-hydroxylase(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50014968(1-(4-Hydroxy-benzyl)-1,3-dihydro-imidazole-2-thion...)
Affinity DataKi:  55nMpH: 4.5Assay Description:Binding affinity towards Dopamine beta hydroxylase using tyramine substrate at pH 4.5 in the absence of fumarateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDopamine beta-hydroxylase(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50014968(1-(4-Hydroxy-benzyl)-1,3-dihydro-imidazole-2-thion...)
Affinity DataKi:  55nMpH: 4.5Assay Description:Compound was evaluated for the inhibition of Dopamine beta hydroxylase at pH 4.5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDopamine beta-hydroxylase(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50000439(5-Butyl-pyridine-2-carboxylic acid | 5-Butyl-pyrid...)
Affinity DataKi:  149nMAssay Description:Compound was evaluated for the inhibition of Dopamine beta hydroxylase at pH 4.5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDopamine beta-hydroxylase(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50000439(5-Butyl-pyridine-2-carboxylic acid | 5-Butyl-pyrid...)
Affinity DataKi:  149nMpH: 4.5Assay Description:Binding affinity towards Dopamine beta hydroxylase using tyramine substrate at pH 4.5 in the absence of fumarateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDopamine beta-hydroxylase(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50014968(1-(4-Hydroxy-benzyl)-1,3-dihydro-imidazole-2-thion...)
Affinity DataKi:  344nMpH: 6.6Assay Description:Compound was evaluated for the inhibition of Dopamine beta hydroxylase at pH 6.6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDopamine beta-hydroxylase(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50017831(2-[1,3]Dithiolan-2-ylidene-ethylamine | CHEMBL1635...)
Affinity DataKi:  5.00E+3nMAssay Description:Compound was evaluated for the ability to bind to dopamine beta-hydroxylase of bovineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDopamine beta-hydroxylase(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50026182(3-Phenyl-prop-2-ynylamine | CHEMBL110611 | US91619...)
Affinity DataKi:  2.10E+4nMAssay Description:Compound was determined for the kinetic constant against Dopamine beta hydroxylase purified from beef adrenals, inhibitory constant (Ki)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDopamine beta-hydroxylase(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50023370(2-Thiophen-2-yl-allylamine | CHEMBL110604)
Affinity DataKi:  3.50E+4nMAssay Description:Compound was determined for the kinetic constant against Dopamine beta hydroxylase purified from beef adrenals, inhibitory constant (Ki)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDopamine beta-hydroxylase(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50023370(2-Thiophen-2-yl-allylamine | CHEMBL110604)
Affinity DataKi:  3.50E+4nMAssay Description:KI value was determined from plots of 1/kinact(observed) vs 1/[inhibitor]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDopamine beta-hydroxylase(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50017830(Benzofuran-6-ol | CHEMBL351630)
Affinity DataKi:  4.00E+4nMAssay Description:Compound was evaluated for the ability to bind to dopamine beta-hydroxylase of bovineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDopamine beta-hydroxylase(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50241361(CHEMBL1515 | METHIMAZOLE | US9138393, Methimazole ...)
Affinity DataKi:  4.50E+4nMpH: 4.5Assay Description:Compound was evaluated for the inhibition of Dopamine beta hydroxylase at pH 6.6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDopamine beta-hydroxylase(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50017834(4-(1-Aminomethyl-prop-2-ynyl)-phenol | CHEMBL16312...)
Affinity DataKi:  5.70E+4nMAssay Description:KI value was determined from plots of 1/kinact(observed) vs 1/[inhibitor]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDopamine beta-hydroxylase(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50017834(4-(1-Aminomethyl-prop-2-ynyl)-phenol | CHEMBL16312...)
Affinity DataKi:  5.70E+4nMAssay Description:Compound was evaluated for the ability to bind to dopamine beta-hydroxylase of bovineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDopamine beta-hydroxylase(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50017834(4-(1-Aminomethyl-prop-2-ynyl)-phenol | CHEMBL16312...)
Affinity DataKi:  5.70E+4nMAssay Description:KI value was determined from plots of 1/kinact(observed) vs 1/[inhibitor]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDopamine beta-hydroxylase(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50286807(1,1a,6,6a-Tetrahydro-cyclopropa[a]indene-3,4-diol ...)
Affinity DataKi:  1.09E+5nMAssay Description:Kinetic constant for inhibition (KI) of Dopamine beta-Hydroxylase(DBH) from bovine adrenal medullaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetDopamine beta-hydroxylase(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50286815(1,1a,6,6a-Tetrahydro-cyclopropa[a]inden-3-ol | CHE...)
Affinity DataKi:  1.50E+5nMAssay Description:Kinetic constant for inhibition (KI) of Dopamine beta-Hydroxylase(DBH) from bovine adrenal medullaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetDopamine beta-hydroxylase(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50286808(1,1a,7,7a-Tetrahydro-3,5-dioxa-cyclopropa[a]-s-ind...)
Affinity DataKi:  1.60E+5nMAssay Description:Kinetic constant for inhibition (KI) of Dopamine beta-Hydroxylase(DBH) from bovine adrenal medullaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetDopamine beta-hydroxylase(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50026184(2-Furan-3-yl-allylamine | CHEMBL108927)
Affinity DataKi:  2.30E+5nMAssay Description:Compound was determined for the kinetic constant against Dopamine beta hydroxylase purified from beef adrenals, inhibitory constant (Ki)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDopamine beta-hydroxylase(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50286814(1-Cyclopropylmethyl-4-methoxy-benzene | CHEMBL1766...)
Affinity DataKi:  2.40E+5nMAssay Description:Kinetic constant for inhibition (KI) of Dopamine beta-Hydroxylase(DBH) from bovine adrenal medullaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetDopamine beta-hydroxylase(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50026189(1-Methyl-2-thiophen-2-yl-allylamine | CHEMBL325080)
Affinity DataKi:  3.60E+5nMAssay Description:Compound was determined for the kinetic constant against Dopamine beta hydroxylase purified from beef adrenals, inhibitory constant (Ki)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDopamine beta-hydroxylase(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50286813(3-Methoxy-1,1a,6,6a-tetrahydro-1-aza-cyclopropa[a]...)
Affinity DataKi:  4.00E+5nMAssay Description:Kinetic constant for inhibition (KI) of Dopamine beta-Hydroxylase(DBH) from bovine adrenal medullaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetDopamine beta-hydroxylase(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50026187(2-Furan-2-yl-allylamine | CHEMBL106238)
Affinity DataKi:  4.10E+5nMAssay Description:Compound was determined for the kinetic constant against Dopamine beta hydroxylase purified from beef adrenals, inhibitory constant (Ki)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDopamine beta-hydroxylase(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50017827(4-(1-Aminomethyl-vinyl)-phenol | CHEMBL330118)
Affinity DataKi:  5.20E+5nMpH: 5.0Assay Description:KI value was determined from plots of 1/kinact(observed) vs 1/[inhibitor]; Apparent values at pH 5.0, 0.24 mM O2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDopamine beta-hydroxylase(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50017827(4-(1-Aminomethyl-vinyl)-phenol | CHEMBL330118)
Affinity DataKi:  5.20E+5nMAssay Description:Compound was evaluated for the ability to bind to dopamine beta-hydroxylase of bovineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDopamine beta-hydroxylase(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50026183(2-Thiophen-3-yl-allylamine | CHEMBL108921)
Affinity DataKi:  5.70E+5nMAssay Description:Compound was determined for the kinetic constant against Dopamine beta hydroxylase purified from beef adrenals, inhibitory constant (Ki)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDopamine beta-hydroxylase(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50286811(3-Methoxy-6,6a-dihydro-1aH-1-oxa-cyclopropa[a]inde...)
Affinity DataKi:  6.50E+5nMAssay Description:Kinetic constant for inhibition (KI) of Dopamine beta-Hydroxylase(DBH) from bovine adrenal medullaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetDopamine beta-hydroxylase(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50017833(4-Hydroxystyrene | 4-Vinylphenol | 4-ethenylphenol...)
Affinity DataKi:  7.00E+5nMAssay Description:Compound was evaluated for the ability to bind to dopamine beta-hydroxylase of bovineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDopamine beta-hydroxylase(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50241361(CHEMBL1515 | METHIMAZOLE | US9138393, Methimazole ...)
Affinity DataKi:  7.16E+5nMpH: 6.6Assay Description:Compound was evaluated for the inhibition of Dopamine beta hydroxylase at pH 4.5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDopamine beta-hydroxylase(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50286809(7,7a-Dihydro-1aH-1,3,5-trioxa-cyclopropa[a]-s-inda...)
Affinity DataKi:  1.01E+6nMAssay Description:Kinetic constant for inhibition (KI) of Dopamine beta-Hydroxylase(DBH) from bovine adrenal medullaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetDopamine beta-hydroxylase(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50286812(6,6a-Dihydro-1aH-1-oxa-cyclopropa[a]indene | CHEMB...)
Affinity DataKi:  1.06E+6nMAssay Description:Kinetic constant for inhibition (KI) of Dopamine beta-Hydroxylase(DBH) from bovine adrenal medullaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetDopamine beta-hydroxylase(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50286810(3-Methoxy-1,1a,6,6a-tetrahydro-cyclopropa[a]indene...)
Affinity DataKi:  1.12E+6nMAssay Description:Kinetic constant for inhibition (KI) of Dopamine beta-Hydroxylase(DBH) from bovine adrenal medullaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetDopamine beta-hydroxylase(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50023371(4-Cyclopropylmethyl-phenol | CHEMBL162030)
Affinity DataKi:  1.20E+6nMAssay Description:KI value was determined from plots of 1/kinact(observed) vs 1/[inhibitor]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDopamine beta-hydroxylase(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50017829(Benzofuran-5-ol | CHEMBL349283)
Affinity DataKi:  1.90E+6nMAssay Description:Compound was evaluated for the ability to bind to dopamine beta-hydroxylase of bovineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDopamine beta-hydroxylase(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50026186(CHEMBL106130 | Methyl-(2-thiophen-2-yl-allyl)-amin...)
Affinity DataKi:  2.15E+6nMAssay Description:Compound was determined for the kinetic constant against Dopamine beta hydroxylase purified from beef adrenals, inhibitory constant (Ki)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDopamine beta-hydroxylase(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50286806(1,1a,6,6a-Tetrahydro-cyclopropa[a]indene | CHEMBL1...)
Affinity DataKi:  3.03E+6nMAssay Description:Kinetic constant for inhibition (KI) of Dopamine beta-Hydroxylase(DBH) from bovine adrenal medullaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetDopamine beta-hydroxylase(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50017828(Benzofuran-7-ol | CHEMBL351411)
Affinity DataKi:  3.20E+6nMAssay Description:Compound was evaluated for the ability to bind to dopamine beta-hydroxylase of bovineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDopamine beta-hydroxylase(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50023371(4-Cyclopropylmethyl-phenol | CHEMBL162030)
Affinity DataKi:  1.20E+7nMAssay Description:Kinetic constant for inhibition (KI) of Dopamine beta-Hydroxylase(DBH) from bovine adrenal medullaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetDopamine beta-hydroxylase(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50026188(2-Phenyl-allylamine | CHEMBL89394)
Affinity DataKi:  1.30E+7nMAssay Description:Compound was determined for the kinetic constant against Dopamine beta hydroxylase purified from beef adrenals, inhibitory constant (Ki)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDopamine beta-hydroxylase(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50026185(CHEMBL105998 | Prop-1-ynyl-benzene)
Affinity DataKi:  2.00E+7nMAssay Description:Compound was determined for the kinetic constant against Dopamine beta hydroxylase purified from beef adrenals, inhibitory constant (Ki)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDopamine beta-hydroxylase(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50017832(4-Propenyl-phenol | CHEMBL163297)
Affinity DataKi: >2.00E+7nMAssay Description:Compound was evaluated for the ability to bind to dopamine beta-hydroxylase of bovineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDopamine beta-hydroxylase(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50014970(4-(3,5-Difluoro-4-hydroxy-benzyl)-2,4-dihydro-[1,2...)
Affinity DataIC50:  35nMAssay Description:Inhibitory activity was determined against bovine dopamine beta-hydroxylase(DBH)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDopamine beta-hydroxylase(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50548688(CHEMBL4764135)
Affinity DataIC50:  39nMAssay Description:Inhibition of bovine adrenal medulla DBH incubated for 25 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDopamine beta-hydroxylase(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50000439(5-Butyl-pyridine-2-carboxylic acid | 5-Butyl-pyrid...)
Affinity DataIC50:  50nMAssay Description:Inhibition of bovine adrenal medulla DBH incubated for 25 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDopamine beta-hydroxylase(Rattus norvegicus)
University Of Illinois

Curated by ChEMBL
LigandPNGBDBM50014978(1-(3,5-Difluoro-4-hydroxy-benzyl)-1,3-dihydro-imid...)
Affinity DataIC50:  74nMAssay Description:Inhibition of dopamine beta-hydroxylase (DbetaH) in hypertensive rats when administered orally (or) intraperitoneallyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDopamine beta-hydroxylase(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50014978(1-(3,5-Difluoro-4-hydroxy-benzyl)-1,3-dihydro-imid...)
Affinity DataIC50:  74nMAssay Description:Inhibitory activity was determined against bovine dopamine beta-hydroxylase(DBH)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDopamine beta-hydroxylase(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50014978(1-(3,5-Difluoro-4-hydroxy-benzyl)-1,3-dihydro-imid...)
Affinity DataIC50:  74nMAssay Description:Inhibitory Concentration against bovine Dopamine beta hydroxylase (DBH); Range is between (0.060-0.0877).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDopamine beta-hydroxylase(Homo sapiens (Human))
Harvard University

Curated by ChEMBL
LigandPNGBDBM50014978(1-(3,5-Difluoro-4-hydroxy-benzyl)-1,3-dihydro-imid...)
Affinity DataIC50:  74.1nMAssay Description:Inhibition of dopamine beta-hydroxylase (DbetaH) enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDopamine beta-hydroxylase(Homo sapiens (Human))
Harvard University

Curated by ChEMBL
LigandPNGBDBM50014978(1-(3,5-Difluoro-4-hydroxy-benzyl)-1,3-dihydro-imid...)
Affinity DataIC50:  74.1nMAssay Description:Inhibition of dopamine beta hydroxylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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