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Found 8 Enz. Inhib. hit(s) with Target = 'Dual specificity protein kinase CLK1/CLK4'
TargetDual specificity protein kinase CLK1/CLK4(Homo sapiens (Human))
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50239787(CHEMBL4094143)
Affinity DataIC50: >1.50E+4nMAssay Description:Inhibition of CLK1/4 in human T24 cells assessed as down regulation of EGFR expression after 3 days by Western blot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK1/CLK4(Homo sapiens (Human))
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50239787(CHEMBL4094143)
Affinity DataIC50: >1.50E+4nMAssay Description:Inhibition of CLK1/4 in human T24 cells assessed as down regulation of HDAC1 expression after 3 days by Western blot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK1/CLK4(Homo sapiens (Human))
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50239782(CHEMBL4082113)
Affinity DataIC50:  9.50E+3nMAssay Description:Inhibition of CLK1/4 in human T24 cells assessed as down regulation of HDAC1 expression after 3 days by Western blot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK1/CLK4(Homo sapiens (Human))
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50239782(CHEMBL4082113)
Affinity DataIC50:  4.20E+3nMAssay Description:Inhibition of CLK1/4 in human MDA-MB-231 cells assessed as down regulation of EGFR expression after 3 days by Western blot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK1/CLK4(Homo sapiens (Human))
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50239787(CHEMBL4094143)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of CLK1/4 in human MDA-MB-231 cells assessed as down regulation of S6 kinase expression after 3 days by Western blot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK1/CLK4(Homo sapiens (Human))
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50239782(CHEMBL4082113)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of CLK1/4 in human MDA-MB-231 cells assessed as down regulation of S6 kinase expression after 3 days by Western blot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK1/CLK4(Homo sapiens (Human))
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50239782(CHEMBL4082113)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of CLK1/4 in human T24 cells assessed as down regulation of EGFR expression after 3 days by Western blot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK1/CLK4(Homo sapiens (Human))
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50239787(CHEMBL4094143)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of CLK1/4 in human MDA-MB-231 cells assessed as down regulation of EGFR expression after 3 days by Western blot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed