Compile Data Set for Download or QSAR
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Found 143 Enz. Inhib. hit(s) with Target = 'Galectin-9'
TargetGalectin-9(Homo sapiens (Human))
The Hashemite University

Curated by ChEMBL
LigandPNGBDBM50326594(CHEMBL1253743 | Di-(3-deoxy-3-(4-((benzylamino)car...)
Affinity DataKd:  530nMAssay Description:Binding affinity to human galectin 9 N-terminal domain at 20 degC by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-9(Homo sapiens (Human))
The Hashemite University

Curated by ChEMBL
LigandPNGBDBM50273581(CHEMBL444662 | N-[(2S,3R,4S,5R,6R)-2-{[(2S,3R,4S,5...)
Affinity DataKd:  730nMAssay Description:Binding affinity to galectin 9N terminal domain at 0 degC by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-9(Homo sapiens (Human))
The Hashemite University

Curated by ChEMBL
LigandPNGBDBM50273581(CHEMBL444662 | N-[(2S,3R,4S,5R,6R)-2-{[(2S,3R,4S,5...)
Affinity DataKd:  730nMAssay Description:Competitive binding affinity to recombinant human galectin-9 N-terminal after 5 mins in presence of fluorescent probe 2-(fluorescein-5-yl-carbonylami...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-9(Homo sapiens (Human))
The Hashemite University

Curated by ChEMBL
LigandPNGBDBM50326596(CHEMBL1253187 | Di-(3-deoxy-3-(4-((allylamino)carb...)
Affinity DataKd:  740nMAssay Description:Binding affinity to human galectin 9 N-terminal domain at 20 degC by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-9(Homo sapiens (Human))
The Hashemite University

Curated by ChEMBL
LigandPNGBDBM50326592(CHEMBL1253923 | Di-(3-deoxy-3-(4-((methylamino)car...)
Affinity DataKd:  910nMAssay Description:Binding affinity to human galectin 9 N-terminal domain at 20 degC by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-9(Homo sapiens (Human))
The Hashemite University

Curated by ChEMBL
LigandPNGBDBM50326595(CHEMBL1253726 | Di-(3-deoxy-3-(4-((2-phenylethylam...)
Affinity DataKd:  1.10E+3nMAssay Description:Binding affinity to human galectin 9 N-terminal domain at 20 degC by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-9(Homo sapiens (Human))
The Hashemite University

Curated by ChEMBL
LigandPNGBDBM50326593(CHEMBL1253742 | Di-(3-deoxy-3-(4-((butylamino)carb...)
Affinity DataKd:  1.10E+3nMAssay Description:Binding affinity to human galectin 9 N-terminal domain at 20 degC by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-9(Homo sapiens (Human))
The Hashemite University

Curated by ChEMBL
LigandPNGBDBM50273431(Bis-[3-O-(3-methoxybenzoyl)-beta-D-galactopyranosy...)
Affinity DataKd:  1.40E+3nMAssay Description:Binding affinity to galectin 9N terminal domain at 0 degC by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-9(Homo sapiens (Human))
The Hashemite University

Curated by ChEMBL
LigandPNGBDBM50273583((2R,3R,4S,5S,6R)-4-hydroxy-6-(hydroxymethyl)-2-met...)
Affinity DataKd:  1.60E+3nMAssay Description:Binding affinity to galectin 9N terminal domain at 0 degC by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-9(Homo sapiens (Human))
The Hashemite University

Curated by ChEMBL
LigandPNGBDBM50533580(CHEMBL4446622)
Affinity DataKd:  1.60E+3nMAssay Description:Competitive binding affinity to recombinant human galectin-9 N-terminal after 5 mins in presence of fluorescent probe 2-(fluorescein-5-yl-carbonylami...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGalectin-9(Homo sapiens (Human))
The Hashemite University

Curated by ChEMBL
LigandPNGBDBM50591132(CHEMBL5182222)
Affinity DataKd:  1.61E+3nMAssay Description:Binding affinity to human N-terminal domain of Galectin-9 assessed as dissociation constant by fluorescence polarizationMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGalectin-9(Homo sapiens (Human))
The Hashemite University

Curated by ChEMBL
LigandPNGBDBM50273580(CHEMBL503116 | N-[(2S,3R,4S,5R,6R)-2-{[(2S,3R,4S,5...)
Affinity DataKd:  1.80E+3nMAssay Description:Binding affinity to galectin 9N terminal domain at 0 degC by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-9(Homo sapiens (Human))
The Hashemite University

Curated by ChEMBL
LigandPNGBDBM50326600(CHEMBL1253217 | Di-(3,5-dimethoxybenzamido)-thiodi...)
Affinity DataKd:  1.82E+3nMAssay Description:Binding affinity to human galectin 9 N-terminal domain at 20 degC by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-9(Homo sapiens (Human))
The Hashemite University

Curated by ChEMBL
LigandPNGBDBM50591132(CHEMBL5182222)
Affinity DataKd:  1.94E+3nMAssay Description:Binding affinity to human C-terminal domain of Galectin-9 assessed as dissociation constant by fluorescence polarizationMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGalectin-9(Homo sapiens (Human))
The Hashemite University

Curated by ChEMBL
LigandPNGBDBM50326597(CHEMBL1253744 | Di-(3-deoxy-3-(4-((2-hydroxypropyl...)
Affinity DataKd:  2.10E+3nMAssay Description:Binding affinity to human galectin 9 N-terminal domain at 20 degC by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-9(Homo sapiens (Human))
The Hashemite University

Curated by ChEMBL
LigandPNGBDBM50273430(Bis-(3-O-benzoyl-beta-D-galactopyranosyl)sulfane |...)
Affinity DataKd:  2.20E+3nMAssay Description:Binding affinity to galectin 9N terminal domain at 0 degC by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-9(Homo sapiens (Human))
The Hashemite University

Curated by ChEMBL
LigandPNGBDBM50326598(CHEMBL1253745 | Di-(3-deoxy-3-(4-((2-methoxyethyla...)
Affinity DataKd:  2.30E+3nMAssay Description:Binding affinity to human galectin 9 N-terminal domain at 20 degC by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-9(Homo sapiens (Human))
The Hashemite University

Curated by ChEMBL
LigandPNGBDBM50533580(CHEMBL4446622)
Affinity DataKd:  2.40E+3nMAssay Description:Competitive binding affinity to recombinant human galectin-9 C-terminal after 5 mins in presence of fluorescent probe 3,3'-dideoxy-3-[4-(fluorescein-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGalectin-9(Homo sapiens (Human))
The Hashemite University

Curated by ChEMBL
LigandPNGBDBM50591130(CHEMBL5181579)
Affinity DataKd:  2.40E+3nMAssay Description:Binding affinity to human C-terminal domain of Galectin-9 assessed as dissociation constant by fluorescence polarizationMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGalectin-9(Homo sapiens (Human))
The Hashemite University

Curated by ChEMBL
LigandPNGBDBM50591130(CHEMBL5181579)
Affinity DataKd:  2.70E+3nMAssay Description:Binding affinity to human N-terminal domain of Galectin-9 assessed as dissociation constant by fluorescence polarizationMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGalectin-9(Homo sapiens (Human))
The Hashemite University

Curated by ChEMBL
LigandPNGBDBM50273434(Bis-(3-O-2-naphthoyl-beta-D-galactopyranosyl)sulfa...)
Affinity DataKd:  2.80E+3nMAssay Description:Binding affinity to galectin 9N terminal domain at 0 degC by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-9(Homo sapiens (Human))
The Hashemite University

Curated by ChEMBL
LigandPNGBDBM50509524(CHEMBL4438703)
Affinity DataKd:  2.80E+3nMAssay Description:Binding affinity at recombinant human C-terminal Galectin 9 expressed in Escherichia coli BL21 incubated for 5 mins by fluorescence anisotropy assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGalectin-9(Homo sapiens (Human))
The Hashemite University

Curated by ChEMBL
LigandPNGBDBM50591131(CHEMBL5193805)
Affinity DataKd:  3.19E+3nMAssay Description:Binding affinity to human N-terminal domain of Galectin-9 assessed as dissociation constant by fluorescence polarizationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGalectin-9(Homo sapiens (Human))
The Hashemite University

Curated by ChEMBL
LigandPNGBDBM50591131(CHEMBL5193805)
Affinity DataKd:  4.28E+3nMAssay Description:Binding affinity to human C-terminal domain of Galectin-9 assessed as dissociation constant by fluorescence polarizationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGalectin-9(Homo sapiens (Human))
The Hashemite University

Curated by ChEMBL
LigandPNGBDBM50509532(CHEMBL4465115)
Affinity DataKd:  4.60E+3nMAssay Description:Binding affinity at recombinant human C-terminal Galectin 9 expressed in Escherichia coli BL21 incubated for 5 mins by fluorescence anisotropy assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGalectin-9(Homo sapiens (Human))
The Hashemite University

Curated by ChEMBL
LigandPNGBDBM50509531(CHEMBL4446731)
Affinity DataKd:  5.80E+3nMAssay Description:Binding affinity at recombinant human C-terminal Galectin 9 expressed in Escherichia coli BL21 incubated for 5 mins by fluorescence anisotropy assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGalectin-9(Homo sapiens (Human))
The Hashemite University

Curated by ChEMBL
LigandPNGBDBM50509524(CHEMBL4438703)
Affinity DataKd:  6.10E+3nMAssay Description:Binding affinity at recombinant human N-terminal Galectin 9 expressed in Escherichia coli BL21 incubated for 5 mins by fluorescence anisotropy assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGalectin-9(Homo sapiens (Human))
The Hashemite University

Curated by ChEMBL
LigandPNGBDBM50273579(CHEMBL457221 | N-[(2S,3R,4S,5R,6R)-2-{[(2S,3R,4S,5...)
Affinity DataKd:  7.00E+3nMAssay Description:Binding affinity to galectin 9N terminal domain at 0 degC by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-9(Homo sapiens (Human))
The Hashemite University

Curated by ChEMBL
LigandPNGBDBM50273433(Bis-(3-O-1-naphthoyl-beta-D-galactopyranosyl)sulfa...)
Affinity DataKd:  8.30E+3nMAssay Description:Binding affinity to galectin 9N terminal domain at 0 degC by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-9(Homo sapiens (Human))
The Hashemite University

Curated by ChEMBL
LigandPNGBDBM50533579(CHEMBL4519227)
Affinity DataKd:  8.30E+3nMAssay Description:Competitive binding affinity to recombinant human galectin-9 N-terminal after 5 mins in presence of fluorescent probe 2-(fluorescein-5-yl-carbonylami...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGalectin-9(Homo sapiens (Human))
The Hashemite University

Curated by ChEMBL
LigandPNGBDBM50326590(CHEMBL1253740 | methyl 3-(4-benzylamino carbonyl-1...)
Affinity DataKd:  1.20E+4nMAssay Description:Binding affinity to human galectin 9 N-terminal domain at 20 degC by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-9(Homo sapiens (Human))
The Hashemite University

Curated by ChEMBL
LigandPNGBDBM50509531(CHEMBL4446731)
Affinity DataKd:  1.20E+4nMAssay Description:Binding affinity at recombinant human N-terminal Galectin 9 expressed in Escherichia coli BL21 incubated for 5 mins by fluorescence anisotropy assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGalectin-9(Homo sapiens (Human))
The Hashemite University

Curated by ChEMBL
LigandPNGBDBM50574702(CHEMBL4872829)
Affinity DataKd:  1.30E+4nMAssay Description:Binding affinity to human galactin-9 N terminal domain assessed as dissociation constant by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGalectin-9(Homo sapiens (Human))
The Hashemite University

Curated by ChEMBL
LigandPNGBDBM50326591(CHEMBL1253741 | methyl 3-deoxy-3-(4-(1-napthyl)-1H...)
Affinity DataKd:  1.30E+4nMAssay Description:Binding affinity to human galectin 9 N-terminal domain at 20 degC by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-9(Homo sapiens (Human))
The Hashemite University

Curated by ChEMBL
LigandPNGBDBM50509533(CHEMBL4557916)
Affinity DataKd:  1.40E+4nMAssay Description:Binding affinity at recombinant human N-terminal Galectin 9 expressed in Escherichia coli BL21 incubated for 5 mins by fluorescence anisotropy assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGalectin-9(Homo sapiens (Human))
The Hashemite University

Curated by ChEMBL
LigandPNGBDBM50509532(CHEMBL4465115)
Affinity DataKd:  1.40E+4nMAssay Description:Binding affinity at recombinant human N-terminal Galectin 9 expressed in Escherichia coli BL21 incubated for 5 mins by fluorescence anisotropy assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGalectin-9(Homo sapiens (Human))
The Hashemite University

Curated by ChEMBL
LigandPNGBDBM50273432(Bis-[3-O-(4-methylbenzoyl)-beta-D-galactopyranosyl...)
Affinity DataKd:  1.50E+4nMAssay Description:Binding affinity to galectin 9N terminal domain at 0 degC by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-9(Homo sapiens (Human))
The Hashemite University

Curated by ChEMBL
LigandPNGBDBM50509533(CHEMBL4557916)
Affinity DataKd:  1.50E+4nMAssay Description:Binding affinity at recombinant human C-terminal Galectin 9 expressed in Escherichia coli BL21 incubated for 5 mins by fluorescence anisotropy assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGalectin-9(Homo sapiens (Human))
The Hashemite University

Curated by ChEMBL
LigandPNGBDBM50574701(CHEMBL4858277)
Affinity DataKd:  1.60E+4nMAssay Description:Binding affinity to human galactin-9 N terminal domain assessed as dissociation constant by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-9(Homo sapiens (Human))
The Hashemite University

Curated by ChEMBL
LigandPNGBDBM50574702(CHEMBL4872829)
Affinity DataKd:  1.80E+4nMAssay Description:Binding affinity to human galactin-9 C terminal domain assessed as dissociation constant by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGalectin-9(Homo sapiens (Human))
The Hashemite University

Curated by ChEMBL
LigandPNGBDBM50048093(CHEBI:610092 | CHEMBL503075 | Lactoside | Methyl B...)
Affinity DataKd:  2.30E+4nMAssay Description:Antagonist activity against human galectin 9 N-terminal domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-9(Homo sapiens (Human))
The Hashemite University

Curated by ChEMBL
LigandPNGBDBM50370453(LACTOSE | Lactose, anhydrous)
Affinity DataKd:  2.30E+4nMAssay Description:Binding affinity to galectin 9N terminal domain at 0 degC by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-9(Homo sapiens (Human))
The Hashemite University

Curated by ChEMBL
LigandPNGBDBM50048095(CHEMBL3311523)
Affinity DataKd:  3.60E+4nMAssay Description:Antagonist activity against human galectin 9 N-terminal domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-9(Homo sapiens (Human))
The Hashemite University

Curated by ChEMBL
LigandPNGBDBM50077225((2R,3R,4S,5R,6S)-2-(hydroxymethyl)-6-{[(2S,3R,4S,5...)
Affinity DataKd:  3.80E+4nMAssay Description:Binding affinity to human galectin 9 N-terminal domain at 20 degC by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-9(Homo sapiens (Human))
The Hashemite University

Curated by ChEMBL
LigandPNGBDBM50077225((2R,3R,4S,5R,6S)-2-(hydroxymethyl)-6-{[(2S,3R,4S,5...)
Affinity DataKd:  3.80E+4nMAssay Description:Binding affinity to galectin 9N terminal domain at 0 degC by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-9(Homo sapiens (Human))
The Hashemite University

Curated by ChEMBL
LigandPNGBDBM50077225((2R,3R,4S,5R,6S)-2-(hydroxymethyl)-6-{[(2S,3R,4S,5...)
Affinity DataKd:  3.80E+4nMAssay Description:Competitive binding affinity to human galectin-9 N-terminal after 5 mins in presence of fluorescent probe by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-9(Homo sapiens (Human))
The Hashemite University

Curated by ChEMBL
LigandPNGBDBM50509526(CHEMBL4578860)
Affinity DataKd:  4.00E+4nMAssay Description:Binding affinity at recombinant human N-terminal Galectin 9 expressed in Escherichia coli BL21 incubated for 5 mins by fluorescence anisotropy assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGalectin-9(Homo sapiens (Human))
The Hashemite University

Curated by ChEMBL
LigandPNGBDBM50077225((2R,3R,4S,5R,6S)-2-(hydroxymethyl)-6-{[(2S,3R,4S,5...)
Affinity DataKd:  4.20E+4nMAssay Description:Competitive binding affinity to recombinant human galectin-9 C-terminal after 5 mins in presence of fluorescent probe 3,3'-dideoxy-3-[4-(fluorescein-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-9(Homo sapiens (Human))
The Hashemite University

Curated by ChEMBL
LigandPNGBDBM50574701(CHEMBL4858277)
Affinity DataKd:  4.50E+4nMAssay Description:Binding affinity to human galactin-9 C terminal domain assessed as dissociation constant by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalectin-9(Homo sapiens (Human))
The Hashemite University

Curated by ChEMBL
LigandPNGBDBM50048097(CHEMBL3311525)
Affinity DataKd:  4.50E+4nMAssay Description:Antagonist activity against human galectin 9 N-terminal domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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