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Found 21 Enz. Inhib. hit(s) with Target = 'Heme ligase'
TargetHeme ligase(Plasmodium falciparum (isolate 3D7))
International Centre For Genetic Engineering And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50250134(CHEMBL4068384)
Affinity DataKd:  2.96E+3nMAssay Description:Binding affinity to Plasmodium falciparum 3D7 HDP assessed as equilibrium dissociation constant by SPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeme ligase(Plasmodium falciparum (isolate 3D7))
International Centre For Genetic Engineering And Biotechnology

Curated by ChEMBL
LigandPNGBDBM558642(US11365202, Compound 3a)
Affinity DataKi:  2.49E+3nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHeme ligase(Plasmodium falciparum (isolate 3D7))
International Centre For Genetic Engineering And Biotechnology

Curated by ChEMBL
LigandPNGBDBM558644(US11365202, Compound 5a)
Affinity DataKi:  2.60E+3nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHeme ligase(Plasmodium falciparum (isolate 3D7))
International Centre For Genetic Engineering And Biotechnology

Curated by ChEMBL
LigandPNGBDBM558642(US11365202, Compound 3a)
Affinity DataKi:  2.78E+3nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHeme ligase(Plasmodium falciparum (isolate 3D7))
International Centre For Genetic Engineering And Biotechnology

Curated by ChEMBL
LigandPNGBDBM558638(US11365202, Compound 3)
Affinity DataKi:  3.32E+3nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHeme ligase(Plasmodium falciparum (isolate 3D7))
International Centre For Genetic Engineering And Biotechnology

Curated by ChEMBL
LigandPNGBDBM558637(US11365202, Compound 2)
Affinity DataKi:  3.49E+3nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHeme ligase(Plasmodium falciparum (isolate 3D7))
International Centre For Genetic Engineering And Biotechnology

Curated by ChEMBL
LigandPNGBDBM558640(US11365202, Compound 5)
Affinity DataKi:  4.54E+3nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHeme ligase(Plasmodium falciparum (isolate 3D7))
International Centre For Genetic Engineering And Biotechnology

Curated by ChEMBL
LigandPNGBDBM558643(US11365202, Compound 3b)
Affinity DataKi:  6.91E+3nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHeme ligase(Plasmodium falciparum (isolate 3D7))
International Centre For Genetic Engineering And Biotechnology

Curated by ChEMBL
LigandPNGBDBM558643(US11365202, Compound 3b)
Affinity DataKi:  9.92E+3nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHeme ligase(Plasmodium falciparum (isolate 3D7))
International Centre For Genetic Engineering And Biotechnology

Curated by ChEMBL
LigandPNGBDBM558643(US11365202, Compound 3b)
Affinity DataIC50:  9.38E+3nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHeme ligase(Plasmodium falciparum (isolate 3D7))
International Centre For Genetic Engineering And Biotechnology

Curated by ChEMBL
LigandPNGBDBM558644(US11365202, Compound 5a)
Affinity DataIC50:  3.53E+3nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHeme ligase(Plasmodium falciparum (isolate 3D7))
International Centre For Genetic Engineering And Biotechnology

Curated by ChEMBL
LigandPNGBDBM558642(US11365202, Compound 3a)
Affinity DataIC50:  3.38E+3nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHeme ligase(Plasmodium falciparum (isolate 3D7))
International Centre For Genetic Engineering And Biotechnology

Curated by ChEMBL
LigandPNGBDBM558643(US11365202, Compound 3b)
Affinity DataIC50:  1.35E+4nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHeme ligase(Plasmodium falciparum (isolate 3D7))
International Centre For Genetic Engineering And Biotechnology

Curated by ChEMBL
LigandPNGBDBM558642(US11365202, Compound 3a)
Affinity DataIC50:  3.78E+3nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHeme ligase(Plasmodium falciparum (isolate 3D7))
International Centre For Genetic Engineering And Biotechnology

Curated by ChEMBL
LigandPNGBDBM558641(US11365202, Compound 6)
Affinity DataIC50: >1.00E+5nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHeme ligase(Plasmodium falciparum (isolate 3D7))
International Centre For Genetic Engineering And Biotechnology

Curated by ChEMBL
LigandPNGBDBM558640(US11365202, Compound 5)
Affinity DataIC50:  7.67E+3nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHeme ligase(Plasmodium falciparum (isolate 3D7))
International Centre For Genetic Engineering And Biotechnology

Curated by ChEMBL
LigandPNGBDBM558639(US11365202, Compound 4)
Affinity DataIC50: >1.00E+5nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHeme ligase(Plasmodium falciparum (isolate 3D7))
International Centre For Genetic Engineering And Biotechnology

Curated by ChEMBL
LigandPNGBDBM558638(US11365202, Compound 3)
Affinity DataIC50:  5.62E+3nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHeme ligase(Plasmodium falciparum (isolate 3D7))
International Centre For Genetic Engineering And Biotechnology

Curated by ChEMBL
LigandPNGBDBM558637(US11365202, Compound 2)
Affinity DataIC50:  5.90E+3nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHeme ligase(Plasmodium falciparum (isolate 3D7))
International Centre For Genetic Engineering And Biotechnology

Curated by ChEMBL
LigandPNGBDBM558645(US11365202, Compound 5b)
Affinity DataIC50: >1.00E+4nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHeme ligase(Plasmodium falciparum (isolate 3D7))
International Centre For Genetic Engineering And Biotechnology

Curated by ChEMBL
LigandPNGBDBM558636(US11365202, Compound 1)
Affinity DataIC50: >1.00E+5nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent