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Found 1466 Enz. Inhib. hit(s) with Target = 'Protein Wnt-3a'
TargetProtein Wnt-3a(Homo sapiens (Human))
Momenta Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50017345(CHEMBL3288260)
Affinity DataKd:  1.80E+4nMAssay Description:Binding affinity to human recombinant WNT3A by surface plasmon resonance assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Wnt-3a(Homo sapiens (Human))
Momenta Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50017346(CHEMBL3288258)
Affinity DataKd:  2.50E+8nMAssay Description:Binding affinity to human recombinant WNT3A by surface plasmon resonance assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Wnt-3a(Homo sapiens (Human))
Momenta Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50017347(CHEMBL3288259)
Affinity DataKd:  2.50E+8nMAssay Description:Binding affinity to human recombinant WNT3A by surface plasmon resonance assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Wnt-3a(Mus musculus)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM89228(1-N-(oxolan-2-ylmethyl)-4-N-(pyridin-4-ylmethyl)be...)
Affinity DataIC50:  7.09E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetProtein Wnt-3a(Mus musculus)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM35354(4-N-(2-methylcyclohexyl)-1-N-(pyridin-4-ylmethyl)b...)
Affinity DataIC50:  1.43E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetProtein Wnt-3a(Mus musculus)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM36829(5-Phenyl-7-[4-(5-trifluoromethyl-pyridin-2-yl)-pip...)
Affinity DataIC50:  5.78E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetProtein Wnt-3a(Mus musculus)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM89229(8-(2-Methoxy-ethylamino)-1,3-dimethyl-7-(3-methyl-...)
Affinity DataIC50:  1.95E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetProtein Wnt-3a(Mus musculus)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM36857((2,4-Dimethoxy-benzyl)-(5-methyl-[1,2,4]triazolo[1...)
Affinity DataIC50:  4.21E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PCBioAssay
TargetProtein Wnt-3a(Mus musculus)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM89230(8-(2-methoxyethylamino)-1,3-dimethyl-7-[3-(trifluo...)
Affinity DataIC50:  5.24E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetProtein Wnt-3a(Mus musculus)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM39087(7-[(4-chlorophenyl)methyl]-1,3-dimethyl-8-prop-2-e...)
Affinity DataIC50:  1.88E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetProtein Wnt-3a(Mus musculus)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM39088(7-[(2,4-dichlorophenyl)methyl]-1,3-dimethyl-8-prop...)
Affinity DataIC50:  2.97E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetProtein Wnt-3a(Mus musculus)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM89231((3-ethyl-1-methyl-2-propyl-4-quinolylidene)amine;h...)
Affinity DataIC50:  1.13E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetProtein Wnt-3a(Mus musculus)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM36929(4-butoxy-8-fluoranyl-5H-pyrimido[5,4-b]indole | 4-...)
Affinity DataIC50:  1.56E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetProtein Wnt-3a(Mus musculus)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM36933(MLS000041708 | N-[2-(3,4-dimethoxyphenyl)ethyl]-4-...)
Affinity DataIC50:  1.07E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetProtein Wnt-3a(Mus musculus)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM89232((8-chloro-5H-pyrimid[5,4-b]indol-4-yl)-[(1-ethylpy...)
Affinity DataIC50: >5.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetProtein Wnt-3a(Mus musculus)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM89233(7-(2-methoxyethyl)-1,3-dimethyl-8-[[4-(phenylmethy...)
Affinity DataIC50:  2.11E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetProtein Wnt-3a(Mus musculus)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM89234(7-butyl-1,3-dimethyl-8-[[methyl-(phenylmethyl)amin...)
Affinity DataIC50:  4.51E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetProtein Wnt-3a(Mus musculus)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM89235(1-butyl-2-[(3,5-dimethyl-1,2-oxazol-4-yl)methylsul...)
Affinity DataIC50: >5.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetProtein Wnt-3a(Mus musculus)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM77990(4-(2-furanyl)-3-propan-2-yl-N-(3-pyridinyl)-2-thia...)
Affinity DataIC50:  1.05E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetProtein Wnt-3a(Mus musculus)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM89236(4-[2-[(4-chloranylphenoxy)methyl]-1-(oxolan-2-ylme...)
Affinity DataIC50:  4.10E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PCBioAssay
TargetProtein Wnt-3a(Mus musculus)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM67747(2-(1-ethyl-2-methyl-5-benzimidazolyl)-5-(5-methyl-...)
Affinity DataIC50:  2.59E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PCBioAssay
TargetProtein Wnt-3a(Mus musculus)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM38951(2,4-dimethyl-N-(3,4,5-trimethoxyphenyl)benzenesulf...)
Affinity DataIC50:  1.38E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetProtein Wnt-3a(Mus musculus)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM89237(4-[(E)-2-(2,3-dimethoxyphenyl)ethenyl]pyridine;hyd...)
Affinity DataIC50:  1.70E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetProtein Wnt-3a(Mus musculus)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM38994(MLS000089367 | N-(2-methoxyethyl)-2-[({5-methyl-2-...)
Affinity DataIC50: >5.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetProtein Wnt-3a(Mus musculus)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM37095(4-(6-methyl-5-imidazo[2,1-b]thiazolyl)-N-(phenylme...)
Affinity DataIC50: >5.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetProtein Wnt-3a(Mus musculus)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM71820(2-(2,5-dimethylphenoxy)-N-(2-hydroxy-5-methyl-phen...)
Affinity DataIC50: >5.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetProtein Wnt-3a(Mus musculus)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM77011(5-(4-methoxy-1-phthalazinyl)-2-(1-piperidinyl)anil...)
Affinity DataIC50:  2.58E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetProtein Wnt-3a(Mus musculus)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM39113(MLS000066583 | N-(3-chloranyl-4-morpholin-4-yl-phe...)
Affinity DataIC50:  5.24E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetProtein Wnt-3a(Mus musculus)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM89238(1-[4-[2-hydroxy-3-(2-methyl-1-benzimidazolyl)propo...)
Affinity DataIC50: >5.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetProtein Wnt-3a(Mus musculus)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM89239((4-cyclohexyl-1-piperazinyl)-(4-methyl-2-furo[3,2-...)
Affinity DataIC50: >5.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetProtein Wnt-3a(Mus musculus)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM41360(MLS000118109 | N-[2-(dipropylamino)ethyl]-1,5-dime...)
Affinity DataIC50: >5.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetProtein Wnt-3a(Mus musculus)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM37170(3-methyl-4-oxo-6-(3,4,5-trimethoxyphenyl)-1,5,6,7-...)
Affinity DataIC50:  1.89E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetProtein Wnt-3a(Mus musculus)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM75787(3-[[4-(2-methyl-2,3-dihydroindole-1-carbonyl)pheny...)
Affinity DataIC50:  1.64E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PCBioAssay
TargetProtein Wnt-3a(Mus musculus)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM89240(7-[(4-fluorophenyl)methyl]-1,3-dimethyl-8-(prop-2-...)
Affinity DataIC50:  5.06E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetProtein Wnt-3a(Mus musculus)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM37221(1-[4-[4-[5-(trifluoromethyl)-2-pyridinyl]-1-pipera...)
Affinity DataIC50:  2.43E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetProtein Wnt-3a(Mus musculus)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM37252((E)-[1-[4-(2-fluorobenzyl)oxyphenyl]-2,5-dimethyl-...)
Affinity DataIC50:  6.57E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetProtein Wnt-3a(Mus musculus)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM89242(MLS000111630 | N-[4-[(3,4-dimethoxyphenyl)sulfamoy...)
Affinity DataIC50:  1.20E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetProtein Wnt-3a(Mus musculus)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM89243(4-(2-Aza-spiro[5.5]undecane-2-sulfonyl)-N-sec-buty...)
Affinity DataIC50:  5.16E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetProtein Wnt-3a(Mus musculus)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM89244(10-(4-tert-Butyl-benzyl)-2,3,4,10-tetrahydro-benzo...)
Affinity DataIC50:  2.94E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetProtein Wnt-3a(Mus musculus)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM89245(1-[4-(5-Chloro-2-methyl-phenyl)-piperazin-1-yl]-2-...)
Affinity DataIC50:  4.43E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetProtein Wnt-3a(Mus musculus)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM89246(4-(4-Benzothiazol-2-yl-piperidine-1-sulfonyl)-N,N-...)
Affinity DataIC50:  3.97E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetProtein Wnt-3a(Mus musculus)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM89247(MLS000123919 | N-(2-Methoxy-benzyl)-4-methyl-N-(4-...)
Affinity DataIC50:  3.27E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetProtein Wnt-3a(Mus musculus)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM89248(2-(3-Methyl-4-oxo-3,4-dihydro-phthalazin-1-yl)-N-(...)
Affinity DataIC50:  1.09E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetProtein Wnt-3a(Mus musculus)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM89249((4-Benzothiazol-2-yl-piperazin-1-yl)-[4-(4-fluoro-...)
Affinity DataIC50:  5.49E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetProtein Wnt-3a(Mus musculus)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM89250((4-Benzothiazol-2-yl-piperazin-1-yl)-(4-benzyl-4H-...)
Affinity DataIC50:  2.68E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetProtein Wnt-3a(Mus musculus)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM89251(9b-(4-chlorophenyl)-1-(4-methylbenzoyl)-1,2,3,9b-t...)
Affinity DataIC50:  1.03E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetProtein Wnt-3a(Mus musculus)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM77198(5,6-dimethyl-4-[4-[2-(4-methylphenoxy)ethyl]-1-pip...)
Affinity DataIC50:  282nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetProtein Wnt-3a(Mus musculus)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM89252(7-(3-Methoxy-benzyl)-8-(2-methoxy-ethoxy)-1,3-dime...)
Affinity DataIC50:  6.29E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetProtein Wnt-3a(Mus musculus)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM89253(8-[2-(4-tert-Butyl-phenoxy)-ethylamino]-1,3,7-trim...)
Affinity DataIC50:  1.20E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetProtein Wnt-3a(Mus musculus)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM54188(1-(3-methylphenyl)-3-[(Z)-(2-oxidanylidene-1-prop-...)
Affinity DataIC50:  2.92E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
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