Found 161 Enz. Inhib. hit(s) with Target = 'Small conductance calcium-activated potassium channel protein 1'
TargetSmall conductance calcium-activated potassium channel protein 1(Homo sapiens (Human))
Neurosearch
Curated by ChEMBL
Neurosearch
Curated by ChEMBL
Affinity DataKd: 54nMAssay Description:Inhibition of human SK1 channel by inside-out patch clamp techniqueMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 1/2/3(Rattus norvegicus)
University Of Li£Ge
Curated by ChEMBL
University Of Li£Ge
Curated by ChEMBL
Affinity DataKi: 0.00400nMAssay Description:Displacement of [125I]apamin from Wistar rat cortical apamin-sensitive siteMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 1/2/3(Rattus norvegicus)
University Of Li£Ge
Curated by ChEMBL
University Of Li£Ge
Curated by ChEMBL
Affinity DataKi: 23nMAssay Description:Displacement of [125I]apamin from SK channel in Wistar rat cortexMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 1/2/3(Rattus norvegicus)
University Of Li£Ge
Curated by ChEMBL
University Of Li£Ge
Curated by ChEMBL
Affinity DataKi: 33nMAssay Description:Displacement of [125I]apamin from SK channel in Wistar rat cortexMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 1/2/3(Rattus norvegicus)
University Of Li£Ge
Curated by ChEMBL
University Of Li£Ge
Curated by ChEMBL
Affinity DataKi: 35nMAssay Description:Displacement of [125I]apamin from SK channel in Wistar rat cortexMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 1/2/3(Rattus norvegicus)
University Of Li£Ge
Curated by ChEMBL
University Of Li£Ge
Curated by ChEMBL
Affinity DataKi: 42nMAssay Description:Displacement of [125I]apamin from SK channel in Wistar rat cortexMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 1/2/3(Rattus norvegicus)
University Of Li£Ge
Curated by ChEMBL
University Of Li£Ge
Curated by ChEMBL
Affinity DataKi: 90nMAssay Description:Displacement of [125I]apamin from SK channel in Wistar rat cortexMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 1/2/3(Rattus norvegicus)
University Of Li£Ge
Curated by ChEMBL
University Of Li£Ge
Curated by ChEMBL
Affinity DataKi: 106nMAssay Description:Displacement of [125I]apamin from SK channel in Wistar rat cortexMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 1/2/3(Rattus norvegicus)
University Of Li£Ge
Curated by ChEMBL
University Of Li£Ge
Curated by ChEMBL
Affinity DataKi: 132nMAssay Description:Displacement of [125I]apamin from SK channel in Wistar rat cortexMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 1/2/3(Rattus norvegicus)
University Of Li£Ge
Curated by ChEMBL
University Of Li£Ge
Curated by ChEMBL
Affinity DataKi: 150nMAssay Description:Displacement of [125I]apamin from SK channel in Wistar rat cortexMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 1/2/3(Rattus norvegicus)
University Of Li£Ge
Curated by ChEMBL
University Of Li£Ge
Curated by ChEMBL
Affinity DataKi: 163nMAssay Description:Displacement of [125I]apamin from SK channel in Wistar rat cortexMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 1/2/3(Rattus norvegicus)
University Of Li£Ge
Curated by ChEMBL
University Of Li£Ge
Curated by ChEMBL
Affinity DataKi: 164nMAssay Description:Displacement of [125I]apamin from SK channel in Wistar rat cortexMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 1/2/3(Rattus norvegicus)
University Of Li£Ge
Curated by ChEMBL
University Of Li£Ge
Curated by ChEMBL
Affinity DataKi: 196nMAssay Description:Displacement of [125I]apamin from SK channel in Wistar rat cortexMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 1/2/3(Rattus norvegicus)
University Of Li£Ge
Curated by ChEMBL
University Of Li£Ge
Curated by ChEMBL
Affinity DataKi: 221nMAssay Description:Displacement of [125I]apamin from SK channel in Wistar rat cortexMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 1/2/3(Rattus norvegicus)
University Of Li£Ge
Curated by ChEMBL
University Of Li£Ge
Curated by ChEMBL
Affinity DataKi: 280nMAssay Description:Displacement of [125I]apamin from SK channel in Wistar rat cortexMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 1/2/3(Rattus norvegicus)
University Of Li£Ge
Curated by ChEMBL
University Of Li£Ge
Curated by ChEMBL
Affinity DataKi: 438nMAssay Description:Displacement of [125I]apamin from SK channel in Wistar rat cortexMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 1/2/3(Rattus norvegicus)
University Of Li£Ge
Curated by ChEMBL
University Of Li£Ge
Curated by ChEMBL
Affinity DataKi: 730nMAssay Description:Displacement of [125I]apamin from Wistar rat cortical apamin-sensitive siteMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 1/2/3(Rattus norvegicus)
University Of Li£Ge
Curated by ChEMBL
University Of Li£Ge
Curated by ChEMBL
Affinity DataKi: 910nMAssay Description:Displacement of [125I]apamin from Wistar rat cortical apamin-sensitive siteMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 1/2/3(Rattus norvegicus)
University Of Li£Ge
Curated by ChEMBL
University Of Li£Ge
Curated by ChEMBL
Affinity DataKi: 1.10E+3nMAssay Description:Displacement of [125I]apamin from SK channel in Wistar rat cortexMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 1/2/3(Rattus norvegicus)
University Of Li£Ge
Curated by ChEMBL
University Of Li£Ge
Curated by ChEMBL
Affinity DataKi: 1.30E+3nMAssay Description:Displacement of [125I]apamin from SK channel in Wistar rat cortexMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 1/2/3(Rattus norvegicus)
University Of Li£Ge
Curated by ChEMBL
University Of Li£Ge
Curated by ChEMBL
Affinity DataKi: 1.30E+3nMAssay Description:Displacement of [125I]apamin from Wistar rat cortical apamin-sensitive siteMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 1/2/3(Rattus norvegicus)
University Of Li£Ge
Curated by ChEMBL
University Of Li£Ge
Curated by ChEMBL
Affinity DataKi: 1.47E+3nMAssay Description:Displacement of [125I]apamin from SK channel in Wistar rat cortexMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 1/2/3(Rattus norvegicus)
University Of Li£Ge
Curated by ChEMBL
University Of Li£Ge
Curated by ChEMBL
Affinity DataKi: 1.60E+3nMAssay Description:Inhibition of [125I]apamin binding to calcium-activated potassium (SK) channel of rat cortexMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 1/2/3(Rattus norvegicus)
University Of Li£Ge
Curated by ChEMBL
University Of Li£Ge
Curated by ChEMBL
Affinity DataKi: 1.60E+3nMAssay Description:Inhibition of [125I]apamin binding to calcium-activated potassium (SK) channel of rat cortexMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 1/2/3(Rattus norvegicus)
University Of Li£Ge
Curated by ChEMBL
University Of Li£Ge
Curated by ChEMBL
Affinity DataKi: 1.69E+3nMAssay Description:Displacement of [125I]apamin from SK channel in Wistar rat cortexMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 1/2/3(Rattus norvegicus)
University Of Li£Ge
Curated by ChEMBL
University Of Li£Ge
Curated by ChEMBL
Affinity DataKi: 1.96E+3nMAssay Description:Displacement of [125I]apamin from SK channel in Wistar rat cortexMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 1/2/3(Rattus norvegicus)
University Of Li£Ge
Curated by ChEMBL
University Of Li£Ge
Curated by ChEMBL
Affinity DataKi: 2.20E+3nMAssay Description:Displacement of [125I]apamin from Wistar rat cortical apamin-sensitive siteMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 1/2/3(Rattus norvegicus)
University Of Li£Ge
Curated by ChEMBL
University Of Li£Ge
Curated by ChEMBL
Affinity DataKi: 2.60E+3nMAssay Description:Inhibition of [125I]apamin binding to calcium-activated potassium (SK) channel of rat cortexMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 1/2/3(Rattus norvegicus)
University Of Li£Ge
Curated by ChEMBL
University Of Li£Ge
Curated by ChEMBL
Affinity DataKi: 3.60E+3nMAssay Description:Inhibition of [125I]apamin binding to calcium-activated potassium (SK) channel of rat cortexMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 1/2/3(Rattus norvegicus)
University Of Li£Ge
Curated by ChEMBL
University Of Li£Ge
Curated by ChEMBL
Affinity DataKi: 3.60E+3nMAssay Description:Displacement of [125I]apamin from Wistar rat cortical apamin-sensitive siteMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 1/2/3(Rattus norvegicus)
University Of Li£Ge
Curated by ChEMBL
University Of Li£Ge
Curated by ChEMBL
Affinity DataKi: 3.80E+3nMAssay Description:Inhibition of [125I]apamin binding to calcium-activated potassium (SK) channel of rat cortexMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 1/2/3(Rattus norvegicus)
University Of Li£Ge
Curated by ChEMBL
University Of Li£Ge
Curated by ChEMBL
Affinity DataKi: 4.90E+3nMAssay Description:Inhibition of [125I]apamin binding to calcium-activated potassium (SK) channel of rat cortexMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 1/2/3(Rattus norvegicus)
University Of Li£Ge
Curated by ChEMBL
University Of Li£Ge
Curated by ChEMBL
Affinity DataKi: 5.40E+3nMAssay Description:Displacement of [125I]apamin from Wistar rat cortical apamin-sensitive siteMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 1/2/3(Rattus norvegicus)
University Of Li£Ge
Curated by ChEMBL
University Of Li£Ge
Curated by ChEMBL
Affinity DataKi: 5.50E+3nMAssay Description:Inhibition of [125I]apamin binding to calcium-activated potassium (SK) channel of rat cortexMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 1/2/3(Rattus norvegicus)
University Of Li£Ge
Curated by ChEMBL
University Of Li£Ge
Curated by ChEMBL
Affinity DataKi: 5.80E+3nMAssay Description:Displacement of [125I]apamin from Wistar rat cortical apamin-sensitive siteMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 1/2/3(Rattus norvegicus)
University Of Li£Ge
Curated by ChEMBL
University Of Li£Ge
Curated by ChEMBL
Affinity DataKi: 6.80E+3nMAssay Description:Inhibition of [125I]apamin binding to calcium-activated potassium (SK) channel of rat cortexMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 1/2/3(Rattus norvegicus)
University Of Li£Ge
Curated by ChEMBL
University Of Li£Ge
Curated by ChEMBL
Affinity DataKi: 7.60E+3nMAssay Description:Inhibition of [125I]apamin binding to calcium-activated potassium (SK) channel of rat cortexMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 1/2/3(Rattus norvegicus)
University Of Li£Ge
Curated by ChEMBL
University Of Li£Ge
Curated by ChEMBL
Affinity DataKi: 9.30E+3nMAssay Description:Inhibition of [125I]apamin binding to calcium-activated potassium (SK) channel of rat cortexMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 1(RAT)
Pudue Pharma Discovery Research
Curated by PDSP Ki Database
Pudue Pharma Discovery Research
Curated by PDSP Ki Database
TargetSmall conductance calcium-activated potassium channel protein 1(Homo sapiens (Human))
Neurosearch
Curated by ChEMBL
Neurosearch
Curated by ChEMBL
Affinity DataIC50: 1.19E+3nMAssay Description:Inhibition of Kca2.1 channel (unknown origin) expressed in HEK293 cells by thallium flux assayMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 1(Homo sapiens (Human))
Neurosearch
Curated by ChEMBL
Neurosearch
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Inhibition of Kca2.1 channel (unknown origin) expressed in HEK293 cells by thallium flux assayMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 1/2/3(Rattus norvegicus)
University Of Li£Ge
Curated by ChEMBL
University Of Li£Ge
Curated by ChEMBL
Affinity DataIC50: 0.0160nMAssay Description:Displacement of [125I]apamin from rat cerebral cortex small conductance calcium-activated potassium channelMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 1(RAT)
Pudue Pharma Discovery Research
Curated by PDSP Ki Database
Pudue Pharma Discovery Research
Curated by PDSP Ki Database
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [125I]apamin from SK+Ca channel in rat cerebral cortexMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 1(Homo sapiens (Human))
Neurosearch
Curated by ChEMBL
Neurosearch
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Inhibition of hSK1 calcium activated potassium channel (SKCa channel)More data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 1(Homo sapiens (Human))
Neurosearch
Curated by ChEMBL
Neurosearch
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibition of hSK1 calcium activated potassium channel (SKCa channel); Range is 1-2More data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 1(Homo sapiens (Human))
Neurosearch
Curated by ChEMBL
Neurosearch
Curated by ChEMBL
Affinity DataIC50: 3.80E+3nMAssay Description:Inhibition of SK1 expressed in CHO FlipIn cells by whole cell patch-clamp assayMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 1(Homo sapiens (Human))
Neurosearch
Curated by ChEMBL
Neurosearch
Curated by ChEMBL
Affinity DataIC50: 43nMAssay Description:Inhibition of Kca2.1 channel expressed in HEK293 cells by thallium flux assayMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 1(Homo sapiens (Human))
Neurosearch
Curated by ChEMBL
Neurosearch
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Inhibition of Kca2.1 channel expressed in HEK293 cells by thallium flux assayMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 1(RAT)
Pudue Pharma Discovery Research
Curated by PDSP Ki Database
Pudue Pharma Discovery Research
Curated by PDSP Ki Database
Affinity DataIC50: 0.0240nMAssay Description:Inhibition of rat SK Calcium channelMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 1(Homo sapiens (Human))
Neurosearch
Curated by ChEMBL
Neurosearch
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMpH: 7.35 T: 2°CAssay Description:All experiments were conducted at room temperature (22-24° C.) with an EPC-10 amplifier and Pulse software (HEKA, Lambrecht/Pfalz, Germany) in the wh...More data for this Ligand-Target Pair