TargetTranslocator protein(Rattus norvegicus (rat))
Brain And Mind Research Institute
Curated by ChEMBL
Brain And Mind Research Institute
Curated by ChEMBL
Affinity DataKd: 0.600nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat cortexMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Brain And Mind Research Institute
Curated by ChEMBL
Brain And Mind Research Institute
Curated by ChEMBL
Affinity DataKd: 1.10nMAssay Description:Displacement of [3H]Ro5-4864 from TSPO in rat kainate lesioned striatumMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Brain And Mind Research Institute
Curated by ChEMBL
Brain And Mind Research Institute
Curated by ChEMBL
Affinity DataKd: 2nMAssay Description:Binding affinity constant for peripheral (mitochondrial) Benzodiazepine receptorMore data for this Ligand-Target Pair
Affinity DataKd: 2nMAssay Description:Binding affinity to human PBRMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Brain And Mind Research Institute
Curated by ChEMBL
Brain And Mind Research Institute
Curated by ChEMBL
Affinity DataKd: 3nMAssay Description:Displacement of [3H]SSR180575 from TSPO in rat cortexMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Brain And Mind Research Institute
Curated by ChEMBL
Brain And Mind Research Institute
Curated by ChEMBL
Affinity DataKd: 3.17nMAssay Description:Irreversible binding affinity to TSPO in rat kidney mitochondrial membraneMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Brain And Mind Research Institute
Curated by ChEMBL
Brain And Mind Research Institute
Curated by ChEMBL
Affinity DataKd: 3.5nMAssay Description:Binding affinity constant for Benzodiazepine receptor in rat RG-2 glioma cellsMore data for this Ligand-Target Pair
Affinity DataKd: 3.5nMAssay Description:Binding affinity to human PBRMore data for this Ligand-Target Pair
Affinity DataKd: 4nMAssay Description:Binding affinity to human PBRMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Brain And Mind Research Institute
Curated by ChEMBL
Brain And Mind Research Institute
Curated by ChEMBL
Affinity DataKd: 5.07nMAssay Description:Irreversible binding affinity to TSPO in rat kidney mitochondrial membraneMore data for this Ligand-Target Pair
Affinity DataKd: 6nMAssay Description:Binding affinity to human PBRMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Brain And Mind Research Institute
Curated by ChEMBL
Brain And Mind Research Institute
Curated by ChEMBL
Affinity DataKd: 8.31nMAssay Description:Irreversible binding affinity to TSPO in rat kidney mitochondrial membraneMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Brain And Mind Research Institute
Curated by ChEMBL
Brain And Mind Research Institute
Curated by ChEMBL
Affinity DataKd: >10nMAssay Description:Binding affinity constant for peripheral (mitochondrial) Benzodiazepine receptorMore data for this Ligand-Target Pair
Affinity DataKd: 11nMAssay Description:Inhibition concentration against human adenosine kinaseMore data for this Ligand-Target Pair
Affinity DataKd: 11nMAssay Description:Binding affinity to recombinant human TSPO by SPR assayMore data for this Ligand-Target Pair
Affinity DataKd: 40nMAssay Description:Binding affinity to C-terminal DDK-tagged human recombinant full-length TSPO expressed in HEK293 cells by SPR assayMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Brain And Mind Research Institute
Curated by ChEMBL
Brain And Mind Research Institute
Curated by ChEMBL
Affinity DataKd: 58nMAssay Description:Binding affinity constant for peripheral (mitochondrial) Benzodiazepine receptorMore data for this Ligand-Target Pair
Affinity DataKd: 61nMAssay Description:Binding affinity to C-terminal DDK-tagged human recombinant full-length TSPO expressed in HEK293 cells by SPR assayMore data for this Ligand-Target Pair
Affinity DataKd: 108nMAssay Description:Binding affinity to recombinant human TSPO by SPR assayMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Brain And Mind Research Institute
Curated by ChEMBL
Brain And Mind Research Institute
Curated by ChEMBL
Affinity DataKd: 213nMAssay Description:Binding affinity constant for peripheral (mitochondrial) Benzodiazepine receptorMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Brain And Mind Research Institute
Curated by ChEMBL
Brain And Mind Research Institute
Curated by ChEMBL
Affinity DataKd: 1.30E+3nMAssay Description:Binding affinity constant for Benzodiazepine receptor in normal rat brain homogenateMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Brain And Mind Research Institute
Curated by ChEMBL
Brain And Mind Research Institute
Curated by ChEMBL
Affinity DataKd: 4.00E+3nMAssay Description:Binding affinity constant for Benzodiazepine receptor in rat C6 glioma cellsMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Brain And Mind Research Institute
Curated by ChEMBL
Brain And Mind Research Institute
Curated by ChEMBL
Affinity DataKi: 0.0430nMAssay Description:In vitro binding affinity for PBR (peripheral benzodiazepine receptor) in rat brainMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Brain And Mind Research Institute
Curated by ChEMBL
Brain And Mind Research Institute
Curated by ChEMBL
Affinity DataKi: 0.0500nMAssay Description:Displacement of [3H]PK11195 from TSPO in Wistar rat heart incubated for 15 minsMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Brain And Mind Research Institute
Curated by ChEMBL
Brain And Mind Research Institute
Curated by ChEMBL
Affinity DataKi: 0.0500nMAssay Description:Displacement of [3H]PK11195 from TSPO in Wistar rat heart incubated for 15 minsMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Brain And Mind Research Institute
Curated by ChEMBL
Brain And Mind Research Institute
Curated by ChEMBL
Affinity DataKi: 0.0700nMAssay Description:Displacement of [11C](R)-PK1119 from Sprague-Dawley rat brain PBRMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Brain And Mind Research Institute
Curated by ChEMBL
Brain And Mind Research Institute
Curated by ChEMBL
Affinity DataKi: 0.0726nMAssay Description:Binding affinity to PBR in Sprague-Dawley rat mitochondrial tissueMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Brain And Mind Research Institute
Curated by ChEMBL
Brain And Mind Research Institute
Curated by ChEMBL
Affinity DataKi: 0.0726nMAssay Description:Displacement of [3H]PK11195 from rat PBR receptorMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Brain And Mind Research Institute
Curated by ChEMBL
Brain And Mind Research Institute
Curated by ChEMBL
Affinity DataKi: 0.0740nMAssay Description:Displacement of [11C](R)-PK1119 from Sprague-Dawley rat brain PBRMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Brain And Mind Research Institute
Curated by ChEMBL
Brain And Mind Research Institute
Curated by ChEMBL
Affinity DataKi: 0.0780nMAssay Description:In vitro inhibition of [11C]2 binding to Peripheral benzodiazepine receptor (PBR) in rat brainMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Brain And Mind Research Institute
Curated by ChEMBL
Brain And Mind Research Institute
Curated by ChEMBL
Affinity DataKi: 0.0800nMAssay Description:Displacement of [11C]DAA1106 from PBR receptor in rat brain membraneMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Brain And Mind Research Institute
Curated by ChEMBL
Brain And Mind Research Institute
Curated by ChEMBL
Affinity DataKi: 0.0978nMAssay Description:Binding affinity to PBR in Sprague-Dawley rat mitochondrial tissueMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Brain And Mind Research Institute
Curated by ChEMBL
Brain And Mind Research Institute
Curated by ChEMBL
Affinity DataKi: 0.0980nMAssay Description:Displacement of [11C](R)-PK1119 from Sprague-Dawley rat brain PBRMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Brain And Mind Research Institute
Curated by ChEMBL
Brain And Mind Research Institute
Curated by ChEMBL
Affinity DataKi: 0.100nMAssay Description:Displacement of [11C](R)-PK1119 from Sprague-Dawley rat brain PBRMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Brain And Mind Research Institute
Curated by ChEMBL
Brain And Mind Research Institute
Curated by ChEMBL
Affinity DataKi: 0.100nMAssay Description:Displacement of [11C](R)-PK1119 from Sprague-Dawley rat brain PBRMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Brain And Mind Research Institute
Curated by ChEMBL
Brain And Mind Research Institute
Curated by ChEMBL
Affinity DataKi: 0.100nMAssay Description:Inhibition of [3H]-Ro-5-4864 binding to mitochondrial rat testis Peripheral type benzodiazepine receptor (PBR)More data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Brain And Mind Research Institute
Curated by ChEMBL
Brain And Mind Research Institute
Curated by ChEMBL
Affinity DataKi: 0.110nMAssay Description:Inhibition of [3H]-PK11195 binding to Peripheral type benzodiazepine receptor (PBR) in rat cortex homogenate by 50%More data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Brain And Mind Research Institute
Curated by ChEMBL
Brain And Mind Research Institute
Curated by ChEMBL
Affinity DataKi: 0.130nMAssay Description:Displacement of [3H]PK11195 from TSPO in Wistar rat kidney mitochondrial fractions incubated for 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Brain And Mind Research Institute
Curated by ChEMBL
Brain And Mind Research Institute
Curated by ChEMBL
Affinity DataKi: 0.130nMAssay Description:Displacement of [3H]PK11195 from TSPO in Sprague-Dawley rat kidney mitochondria after 1 hr by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Brain And Mind Research Institute
Curated by ChEMBL
Brain And Mind Research Institute
Curated by ChEMBL
Affinity DataKi: 0.150nMAssay Description:Displacement of [3H]PK11195 from translocator protein in rat kidney mitochondrial membraneMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Brain And Mind Research Institute
Curated by ChEMBL
Brain And Mind Research Institute
Curated by ChEMBL
Affinity DataKi: 0.150nMAssay Description:Displacement of [3H]PK11195 from peripheral benzodiazepine receptor in Sprague-Dawley rat cerebral cortex membrane by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.150nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.150nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Brain And Mind Research Institute
Curated by ChEMBL
Brain And Mind Research Institute
Curated by ChEMBL
Affinity DataKi: 0.160nMAssay Description:In vitro inhibition of [11C]2 binding to Peripheral benzodiazepine receptor (PBR) in rat brainMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Brain And Mind Research Institute
Curated by ChEMBL
Brain And Mind Research Institute
Curated by ChEMBL
Affinity DataKi: 0.160nMAssay Description:Displacement of [11C]DAA1106 from Sprague-Dawley rat brain PBRMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Brain And Mind Research Institute
Curated by ChEMBL
Brain And Mind Research Institute
Curated by ChEMBL
Affinity DataKi: 0.170nMAssay Description:In vitro inhibition of [11C]2 binding to Peripheral benzodiazepine receptor (PBR) in rat brainMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Brain And Mind Research Institute
Curated by ChEMBL
Brain And Mind Research Institute
Curated by ChEMBL
Affinity DataKi: 0.180nMAssay Description:Inhibition of [3H]-PK11195 binding to Peripheral type benzodiazepine receptor (PBR) in rat cortex homogenate by 50%More data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Brain And Mind Research Institute
Curated by ChEMBL
Brain And Mind Research Institute
Curated by ChEMBL
Affinity DataKi: 0.180nMAssay Description:Displacement of [3H]PK11195 from rat PBR receptorMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Brain And Mind Research Institute
Curated by ChEMBL
Brain And Mind Research Institute
Curated by ChEMBL
Affinity DataKi: 0.180nMAssay Description:Displacement of [3H]PK11195 from translocator protein in rat kidney mitochondrial membraneMore data for this Ligand-Target Pair