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Found 144 Enz. Inhib. hit(s) with Target = 'cGMP-dependent protein kinase 2'
TargetcGMP-dependent protein kinase 2(Homo sapiens (Human))
Baylor College Of Medicine

LigandPNGBDBM65501(8-pCP-cGMP | Cyclic GMP analogs | cGMP)
Affinity DataEC50:  257nMpH: 7.0Assay Description:Kinase activity was determined employing a microfluidic mobility-shift assay on a Caliper DeskTop Profiler (Caliper Life Sciences, PerkinElmer). The ...More data for this Ligand-Target Pair
TargetcGMP-dependent protein kinase 2 [41-418,G356E](Homo sapiens (Human))
Baylor College Of Medicine

LigandPNGBDBM65505(PET-cGMP)
Affinity DataEC50:  5.30nMpH: 7.0Assay Description:Kinase activity was determined employing a microfluidic mobility-shift assay on a Caliper DeskTop Profiler (Caliper Life Sciences, PerkinElmer). The ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase 2(Homo sapiens (Human))
Baylor College Of Medicine

LigandPNGBDBM65501(8-pCP-cGMP | Cyclic GMP analogs | cGMP)
Affinity DataEC50:  22nMpH: 7.0Assay Description:Kinase activity was determined employing a microfluidic mobility-shift assay on a Caliper DeskTop Profiler (Caliper Life Sciences, PerkinElmer). The ...More data for this Ligand-Target Pair
TargetcGMP-dependent protein kinase 2(Homo sapiens (Human))
Baylor College Of Medicine

LigandPNGBDBM65505(PET-cGMP)
Affinity DataEC50:  225nMpH: 7.0Assay Description:Kinase activity was determined employing a microfluidic mobility-shift assay on a Caliper DeskTop Profiler (Caliper Life Sciences, PerkinElmer). The ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase 2 [41-418](Homo sapiens (Human))
Baylor College Of Medicine

LigandPNGBDBM65501(8-pCP-cGMP | Cyclic GMP analogs | cGMP)
Affinity DataEC50:  96nMpH: 7.0Assay Description:Kinase activity was determined employing a microfluidic mobility-shift assay on a Caliper DeskTop Profiler (Caliper Life Sciences, PerkinElmer). The ...More data for this Ligand-Target Pair
TargetcGMP-dependent protein kinase 2 [41-418](Homo sapiens (Human))
Baylor College Of Medicine

LigandPNGBDBM65502(2-amino-8-bromo-9-[(2R,4aR,6R,7R,7aS)-2,7-dihydrox...)
Affinity DataEC50:  20nMpH: 7.0Assay Description:Kinase activity was determined employing a microfluidic mobility-shift assay on a Caliper DeskTop Profiler (Caliper Life Sciences, PerkinElmer). The ...More data for this Ligand-Target Pair
TargetcGMP-dependent protein kinase 2 [41-418](Homo sapiens (Human))
Baylor College Of Medicine

LigandPNGBDBM65501(8-pCP-cGMP | Cyclic GMP analogs | cGMP)
Affinity DataEC50:  5nMpH: 7.0Assay Description:Kinase activity was determined employing a microfluidic mobility-shift assay on a Caliper DeskTop Profiler (Caliper Life Sciences, PerkinElmer). The ...More data for this Ligand-Target Pair
TargetcGMP-dependent protein kinase 2 [41-418](Homo sapiens (Human))
Baylor College Of Medicine

LigandPNGBDBM65505(PET-cGMP)
Affinity DataEC50:  193nMpH: 7.0Assay Description:Kinase activity was determined employing a microfluidic mobility-shift assay on a Caliper DeskTop Profiler (Caliper Life Sciences, PerkinElmer). The ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase 2 [41-418,G232E](Homo sapiens (Human))
Baylor College Of Medicine

LigandPNGBDBM65501(8-pCP-cGMP | Cyclic GMP analogs | cGMP)
Affinity DataEC50:  184nMpH: 7.0Assay Description:Kinase activity was determined employing a microfluidic mobility-shift assay on a Caliper DeskTop Profiler (Caliper Life Sciences, PerkinElmer). The ...More data for this Ligand-Target Pair
TargetcGMP-dependent protein kinase 2 [41-418,G232E](Homo sapiens (Human))
Baylor College Of Medicine

LigandPNGBDBM65502(2-amino-8-bromo-9-[(2R,4aR,6R,7R,7aS)-2,7-dihydrox...)
Affinity DataEC50:  11nMpH: 7.0Assay Description:Kinase activity was determined employing a microfluidic mobility-shift assay on a Caliper DeskTop Profiler (Caliper Life Sciences, PerkinElmer). The ...More data for this Ligand-Target Pair
TargetcGMP-dependent protein kinase 2 [41-418,G232E](Homo sapiens (Human))
Baylor College Of Medicine

LigandPNGBDBM65501(8-pCP-cGMP | Cyclic GMP analogs | cGMP)
Affinity DataEC50:  116nMpH: 7.0Assay Description:Kinase activity was determined employing a microfluidic mobility-shift assay on a Caliper DeskTop Profiler (Caliper Life Sciences, PerkinElmer). The ...More data for this Ligand-Target Pair
TargetcGMP-dependent protein kinase 2 [41-418,G232E](Homo sapiens (Human))
Baylor College Of Medicine

LigandPNGBDBM65505(PET-cGMP)
Affinity DataEC50:  1.96E+3nMpH: 7.0Assay Description:Kinase activity was determined employing a microfluidic mobility-shift assay on a Caliper DeskTop Profiler (Caliper Life Sciences, PerkinElmer). The ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase 2 [41-418,G356E](Homo sapiens (Human))
Baylor College Of Medicine

LigandPNGBDBM65501(8-pCP-cGMP | Cyclic GMP analogs | cGMP)
Affinity DataEC50:  50nMpH: 7.0Assay Description:Kinase activity was determined employing a microfluidic mobility-shift assay on a Caliper DeskTop Profiler (Caliper Life Sciences, PerkinElmer). The ...More data for this Ligand-Target Pair
TargetcGMP-dependent protein kinase 2 [41-418,G356E](Homo sapiens (Human))
Baylor College Of Medicine

LigandPNGBDBM65502(2-amino-8-bromo-9-[(2R,4aR,6R,7R,7aS)-2,7-dihydrox...)
Affinity DataEC50:  30nMpH: 7.0Assay Description:Kinase activity was determined employing a microfluidic mobility-shift assay on a Caliper DeskTop Profiler (Caliper Life Sciences, PerkinElmer). The ...More data for this Ligand-Target Pair
TargetcGMP-dependent protein kinase 2 [41-418,G356E](Homo sapiens (Human))
Baylor College Of Medicine

LigandPNGBDBM65501(8-pCP-cGMP | Cyclic GMP analogs | cGMP)
Affinity DataEC50: <1nMpH: 7.0Assay Description:Kinase activity was determined employing a microfluidic mobility-shift assay on a Caliper DeskTop Profiler (Caliper Life Sciences, PerkinElmer). The ...More data for this Ligand-Target Pair
TargetcGMP-dependent protein kinase 2(Homo sapiens (Human))
Baylor College Of Medicine

LigandPNGBDBM65502(2-amino-8-bromo-9-[(2R,4aR,6R,7R,7aS)-2,7-dihydrox...)
Affinity DataEC50:  58nMpH: 7.0Assay Description:Kinase activity was determined employing a microfluidic mobility-shift assay on a Caliper DeskTop Profiler (Caliper Life Sciences, PerkinElmer). The ...More data for this Ligand-Target Pair
TargetcGMP-dependent protein kinase 2(Homo sapiens (Human))
Baylor College Of Medicine

LigandPNGBDBM31094(PKC-412 | cid_24202429)
Affinity DataKd:  7.40E+4nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetcGMP-dependent protein kinase 2(Homo sapiens (Human))
Baylor College Of Medicine

LigandPNGBDBM31096(CHEMBL290084 | Staurosporine | cid_451705)
Affinity DataKd:  1.60E+4nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetcGMP-dependent protein kinase 2(Homo sapiens (Human))
Baylor College Of Medicine

LigandPNGBDBM50326053(CHEMBL608533 | PKC-412)
Affinity DataKd:  74nMAssay Description:Binding affinity to PRKG2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase 2(Homo sapiens (Human))
Baylor College Of Medicine

LigandPNGBDBM50308060(16-hydroxy-16-(hydroxymethyl)-15-methyl-28-oxa-4,1...)
Affinity DataKd:  25nMAssay Description:Binding affinity to PRKG2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase 2(Homo sapiens (Human))
Baylor College Of Medicine

LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Affinity DataKd:  16nMAssay Description:Binding constant for PRKG2 kinase domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase 2(Homo sapiens (Human))
Baylor College Of Medicine

LigandPNGBDBM50026612(BIBF-1120 | Nintedanib | US10981896, Compound Nint...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PRKG2 kinase domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase 2(Homo sapiens (Human))
Baylor College Of Medicine

LigandPNGBDBM50326053(CHEMBL608533 | PKC-412)
Affinity DataKd:  74nMAssay Description:Binding constant for PRKG2 kinase domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase 2(Homo sapiens (Human))
Baylor College Of Medicine

LigandPNGBDBM50308060(16-hydroxy-16-(hydroxymethyl)-15-methyl-28-oxa-4,1...)
Affinity DataKd:  25nMAssay Description:Binding constant for PRKG2 kinase domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase 2(Homo sapiens (Human))
Baylor College Of Medicine

LigandPNGBDBM50326053(CHEMBL608533 | PKC-412)
Affinity DataKd:  74nMAssay Description:Binding constant for PRKG2 kinase domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase 2(Homo sapiens (Human))
Baylor College Of Medicine

LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Affinity DataKd:  16nMAssay Description:Binding constant for PRKG2 kinase domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase 2(Homo sapiens (Human))
Baylor College Of Medicine

LigandPNGBDBM50300690(1-(5-Tert-Butyl-1,2-Oxazol-3-Yl)-3-(4-{7-[2-(Morph...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to PRKG2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase 2(Homo sapiens (Human))
Baylor College Of Medicine

LigandPNGBDBM13535(4-[6-methoxy-7-(3-piperidin-1-ylpropoxy)quinazolin...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to PRKG2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase 2(Homo sapiens (Human))
Baylor College Of Medicine

LigandPNGBDBM16673(4-[4-({[4-chloro-3-(trifluoromethyl)phenyl]carbamo...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to PRKG2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase 2(Homo sapiens (Human))
Baylor College Of Medicine

LigandPNGBDBM50326054(CHEMBL1240703)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to PRKG2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase 2(Homo sapiens (Human))
Baylor College Of Medicine

LigandPNGBDBM4814(CHEMBL535 | N-[2-(diethylamino)ethyl]-5-[(Z)-(5-fl...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to PRKG2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase 2(Homo sapiens (Human))
Baylor College Of Medicine

LigandPNGBDBM5446(CHEMBL553 | ERLOTINIB HYDROCHLORIDE | Erlotinib | ...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PRKG2 kinase domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase 2(Homo sapiens (Human))
Baylor College Of Medicine

LigandPNGBDBM6568(6-(2,6-dichlorophenyl)-8-methyl-2-{[3-(methylsulfa...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PRKG2 kinase domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase 2(Homo sapiens (Human))
Baylor College Of Medicine

LigandPNGBDBM26300(2-{3-[(7-{3-[ethyl(2-hydroxyethyl)amino]propoxy}qu...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PRKG2 kinase domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase 2(Homo sapiens (Human))
Baylor College Of Medicine

LigandPNGBDBM50355496(CHEMBL1908397)
Affinity DataKd:  800nMAssay Description:Binding constant for PRKG2 kinase domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase 2(Homo sapiens (Human))
Baylor College Of Medicine

LigandPNGBDBM25617(N-[3-({5-chloro-1H-pyrrolo[2,3-b]pyridin-3-yl}carb...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PRKG2 kinase domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase 2(Homo sapiens (Human))
Baylor College Of Medicine

LigandPNGBDBM25121(4-{[(7R)-8-cyclopentyl-7-ethyl-5-methyl-6-oxo-5,6,...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PRKG2 kinase domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase 2(Homo sapiens (Human))
Baylor College Of Medicine

LigandPNGBDBM60665(BDBM50249542 | US9145414, R406 | US9212178, R406)
Affinity DataKd:  3.60E+3nMAssay Description:Binding constant for PRKG2 kinase domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase 2(Homo sapiens (Human))
Baylor College Of Medicine

LigandPNGBDBM50306682((R)-3-(1-(2,6-dichloro-3-fluorophenyl)ethoxy)-5-(1...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PRKG2 kinase domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase 2(Homo sapiens (Human))
Baylor College Of Medicine

LigandPNGBDBM13530(4-[(4-methylpiperazin-1-yl)methyl]-N-[4-methyl-3-[...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PRKG2 kinase domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase 2(Homo sapiens (Human))
Baylor College Of Medicine

LigandPNGBDBM24773(AMG 706 | AMG-706 | Motesanib | N-(3,3-dimethyl-1,...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PRKG2 kinase domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase 2(Homo sapiens (Human))
Baylor College Of Medicine

LigandPNGBDBM50193995(3-((3R,4R)-4-methyl-3-(methyl(7H-pyrrolo[2,3-d]pyr...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PRKG2 kinase domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase 2(Homo sapiens (Human))
Baylor College Of Medicine

LigandPNGBDBM25045(3-(4-morpholin-4-ylpyrido[2,3]furo[2,4-b]pyrimidin...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PRKG2 kinase domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase 2(Homo sapiens (Human))
Baylor College Of Medicine

LigandPNGBDBM50355495(CHEMBL1908391)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PRKG2 kinase domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase 2(Homo sapiens (Human))
Baylor College Of Medicine

LigandPNGBDBM50237710(4-methyl-N-[3-(4-methyl-1H-imidazol-1-yl)-5-(trifl...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PRKG2 kinase domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase 2(Homo sapiens (Human))
Baylor College Of Medicine

LigandPNGBDBM27817(2-{[2-({1-[2-(dimethylamino)acetyl]-5-methoxy-2,3-...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PRKG2 kinase domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase 2(Homo sapiens (Human))
Baylor College Of Medicine

LigandPNGBDBM31095(5-[(Z)-(5-fluoranyl-2-oxidanylidene-1H-indol-3-yli...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PRKG2 kinase domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase 2(Homo sapiens (Human))
Baylor College Of Medicine

LigandPNGBDBM5931(BMS-387072 | CHEMBL296468 | N-(5-{[(5-tert-butyl-1...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PRKG2 kinase domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase 2(Homo sapiens (Human))
Baylor College Of Medicine

LigandPNGBDBM50300690(1-(5-Tert-Butyl-1,2-Oxazol-3-Yl)-3-(4-{7-[2-(Morph...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PRKG2 kinase domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase 2(Homo sapiens (Human))
Baylor College Of Medicine

LigandPNGBDBM15244(5-(2,6-dichlorophenyl)-2-(2,4-difluorophenyl)sulfa...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PRKG2 kinase domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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