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Found 14 Enz. Inhib. hit(s) with all data for entry = 916
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Tensha Therapeutics

US Patent
LigandPNGBDBM50365262((+)-JQ1 | (S)-JQ1 (1) | CHEMBL1957266 | JQ1 | US10...)
Affinity DataKd:  3.60E+3nMAssay Description:A BROMOscan binding assay was utilized to test the in vitro binding activity of (S)-Compounds 1, 2, 3, 4, 5 and 7 to the first and second bromodomain...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetIsoform C of Bromodomain-containing protein 4 (Short)(Homo sapiens (Human))
Tensha Therapeutics

US Patent
LigandPNGBDBM50365262((+)-JQ1 | (S)-JQ1 (1) | CHEMBL1957266 | JQ1 | US10...)
Affinity DataKd:  3.80E+3nMMore data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Tensha Therapeutics

US Patent
LigandPNGBDBM298346(US10124009, Compound 1)
Affinity DataKd:  1.30E+3nMAssay Description:A BROMOscan binding assay was utilized to test the in vitro binding activity of (S)-Compounds 1, 2, 3, 4, 5 and 7 to the first and second bromodomain...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetIsoform C of Bromodomain-containing protein 4 (Short)(Homo sapiens (Human))
Tensha Therapeutics

US Patent
LigandPNGBDBM298346(US10124009, Compound 1)
Affinity DataKd:  1.50E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Tensha Therapeutics

US Patent
LigandPNGBDBM298347(US10124009, Compound 2)
Affinity DataKd:  1.90E+3nMAssay Description:A BROMOscan binding assay was utilized to test the in vitro binding activity of (S)-Compounds 1, 2, 3, 4, 5 and 7 to the first and second bromodomain...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetIsoform C of Bromodomain-containing protein 4 (Short)(Homo sapiens (Human))
Tensha Therapeutics

US Patent
LigandPNGBDBM298347(US10124009, Compound 2)
Affinity DataKd:  1.90E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetIsoform C of Bromodomain-containing protein 4 (Short)(Homo sapiens (Human))
Tensha Therapeutics

US Patent
LigandPNGBDBM298351(US10124009, Compound 7)
Affinity DataKd:  2.10E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetIsoform C of Bromodomain-containing protein 4 (Short)(Homo sapiens (Human))
Tensha Therapeutics

US Patent
LigandPNGBDBM298348(US10124009, Compound 3)
Affinity DataKd:  1.20E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Tensha Therapeutics

US Patent
LigandPNGBDBM298349(US10124009, Compound 4)
Affinity DataKd:  1.10E+3nMAssay Description:A BROMOscan binding assay was utilized to test the in vitro binding activity of (S)-Compounds 1, 2, 3, 4, 5 and 7 to the first and second bromodomain...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetIsoform C of Bromodomain-containing protein 4 (Short)(Homo sapiens (Human))
Tensha Therapeutics

US Patent
LigandPNGBDBM298349(US10124009, Compound 4)
Affinity DataKd:  1.30E+3nMMore data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Tensha Therapeutics

US Patent
LigandPNGBDBM298350(US10124009, Compound 5)
Affinity DataKd:  430nMAssay Description:A BROMOscan binding assay was utilized to test the in vitro binding activity of (S)-Compounds 1, 2, 3, 4, 5 and 7 to the first and second bromodomain...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetIsoform C of Bromodomain-containing protein 4 (Short)(Homo sapiens (Human))
Tensha Therapeutics

US Patent
LigandPNGBDBM298350(US10124009, Compound 5)
Affinity DataKd:  400nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Tensha Therapeutics

US Patent
LigandPNGBDBM298351(US10124009, Compound 7)
Affinity DataKd:  1.50E+3nMAssay Description:A BROMOscan binding assay was utilized to test the in vitro binding activity of (S)-Compounds 1, 2, 3, 4, 5 and 7 to the first and second bromodomain...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Tensha Therapeutics

US Patent
LigandPNGBDBM298348(US10124009, Compound 3)
Affinity DataKd:  1.10E+3nMAssay Description:A BROMOscan binding assay was utilized to test the in vitro binding activity of (S)-Compounds 1, 2, 3, 4, 5 and 7 to the first and second bromodomain...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent